PE20141993A1 - Compuestos de benzotiazolona - Google Patents

Compuestos de benzotiazolona

Info

Publication number
PE20141993A1
PE20141993A1 PE2014000312A PE2014000312A PE20141993A1 PE 20141993 A1 PE20141993 A1 PE 20141993A1 PE 2014000312 A PE2014000312 A PE 2014000312A PE 2014000312 A PE2014000312 A PE 2014000312A PE 20141993 A1 PE20141993 A1 PE 20141993A1
Authority
PE
Peru
Prior art keywords
benzothiazolone compounds
benzothiazolone
compounds
caquexia
butoxiphenil
Prior art date
Application number
PE2014000312A
Other languages
English (en)
Inventor
Jun Cao
Bernhard Erb
Robin Alec Fairhurst
Arnaud Grandeury
Shinji Hatakeyama
Magdalena Koziczak-Holbro
Xinzhong Lai
Phillip Lustenberger
Bernd Riebesehl
Nicola Tufilli
Thomas Ullrich
Xiang Wu
Jianguang Zhou
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47010668&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20141993(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PE20141993A1 publication Critical patent/PE20141993A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/08—Acetic acid
    • C07C53/10—Salts thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

REFERIDO A UN COMPUESTO DE FORMULA (R)-7-(2-(1-(4-BUTOXIFENIL)-2-METILPROPAN-2-ILAMINO)-1-HIDROXIETIL)-5-HIDROXIBENZO[D]TIAZOL-2(3H)-ONA. SE REFIERE TAMBIEN A UNA COMPOSICION FARMACEUTICA, CARACTERIZADA POR SU APLICACION PARA EL TRATAMIENTO O LA PREVENCION DE LA DISTROFIA MUSCULAR, CAQUEXIA O SARCOPENIA
PE2014000312A 2011-09-06 2012-09-05 Compuestos de benzotiazolona PE20141993A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN2011079379 2011-09-06

Publications (1)

Publication Number Publication Date
PE20141993A1 true PE20141993A1 (es) 2014-12-17

Family

ID=47010668

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2014000312A PE20141993A1 (es) 2011-09-06 2012-09-05 Compuestos de benzotiazolona

Country Status (38)

Country Link
US (6) US8933108B2 (es)
EP (1) EP2753609B1 (es)
JP (2) JP6130835B2 (es)
KR (2) KR101800140B1 (es)
CN (2) CN106187942B (es)
AP (1) AP3830A (es)
AR (1) AR087787A1 (es)
AU (1) AU2013200422C1 (es)
BR (1) BR112014004732A2 (es)
CA (1) CA2845766A1 (es)
CL (1) CL2014000493A1 (es)
CO (1) CO6900147A2 (es)
CR (1) CR20140114A (es)
CU (1) CU24303B1 (es)
CY (1) CY1118585T1 (es)
DK (1) DK2753609T3 (es)
EA (1) EA022909B1 (es)
ES (1) ES2615052T3 (es)
GT (1) GT201400042A (es)
HR (1) HRP20170075T1 (es)
HU (1) HUE030530T2 (es)
IL (1) IL231235A (es)
JO (1) JO3192B1 (es)
LT (1) LT2753609T (es)
MX (1) MX345405B (es)
MY (1) MY163301A (es)
PE (1) PE20141993A1 (es)
PL (1) PL2753609T3 (es)
PT (1) PT2753609T (es)
RS (1) RS55468B1 (es)
SG (1) SG2014013114A (es)
SI (1) SI2753609T1 (es)
TN (1) TN2014000060A1 (es)
TW (1) TWI555738B (es)
UA (1) UA114295C2 (es)
UY (1) UY34312A (es)
WO (1) WO2013035047A1 (es)
ZA (2) ZA201401112B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA117092C2 (uk) 2011-09-06 2018-06-25 Байєр Інтеллектуал Проперті Гмбх Амінозаміщені імідазопіридазини
JO3192B1 (ar) 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
BR112015004127A2 (pt) * 2012-08-30 2017-07-04 Novartis Ag sais de composto benzotiazolona como agonista de beta-2-adrenorreceptor
JP2015537017A (ja) 2012-11-19 2015-12-24 バイエル ファーマ アクチエンゲゼルシャフト アミノイミダゾピリダジン類
WO2014132205A1 (en) * 2013-02-28 2014-09-04 Novartis Ag Formulation comprising benzothiazolone compound
US10967119B1 (en) 2019-04-01 2021-04-06 Azizi Bilal Wearable medication injecting device

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Also Published As

Publication number Publication date
SI2753609T1 (sl) 2017-03-31
US8933108B2 (en) 2015-01-13
GT201400042A (es) 2015-02-19
KR101628585B1 (ko) 2016-06-08
CN103781771A (zh) 2014-05-07
IL231235A0 (en) 2014-04-30
CN106187942B (zh) 2020-06-26
CL2014000493A1 (es) 2014-10-03
CR20140114A (es) 2014-05-06
PT2753609T (pt) 2017-02-08
CA2845766A1 (en) 2013-03-14
JO3192B1 (ar) 2018-03-08
MX345405B (es) 2017-01-30
PL2753609T3 (pl) 2017-05-31
HUE030530T2 (en) 2017-05-29
JP6340103B2 (ja) 2018-06-06
CU24303B1 (es) 2018-01-10
TWI555738B (zh) 2016-11-01
UA114295C2 (uk) 2017-05-25
MX2014002688A (es) 2014-04-14
CN106187942A (zh) 2016-12-07
US9913828B2 (en) 2018-03-13
US20160075670A1 (en) 2016-03-17
LT2753609T (lt) 2017-01-10
IL231235A (en) 2017-09-28
WO2013035047A1 (en) 2013-03-14
US20160279107A1 (en) 2016-09-29
KR20160038079A (ko) 2016-04-06
RS55468B1 (sr) 2017-04-28
SG2014013114A (en) 2014-07-30
KR20140057382A (ko) 2014-05-12
TN2014000060A1 (en) 2015-07-01
CU20140028A7 (es) 2014-05-27
HRP20170075T1 (hr) 2017-03-24
JP6130835B2 (ja) 2017-05-17
TW201317221A (zh) 2013-05-01
MY163301A (en) 2017-09-15
EP2753609A1 (en) 2014-07-16
AU2013200422B2 (en) 2014-08-07
JP2014525472A (ja) 2014-09-29
CN103781771B (zh) 2016-08-24
AP3830A (en) 2016-09-30
US20180140582A1 (en) 2018-05-24
AU2013200422C1 (en) 2015-01-15
ZA201500790B (en) 2017-04-26
EA201490573A1 (ru) 2014-06-30
AR087787A1 (es) 2014-04-16
CY1118585T1 (el) 2017-07-12
US20150094346A1 (en) 2015-04-02
US20130245080A1 (en) 2013-09-19
ZA201401112B (en) 2016-01-27
US20150336914A1 (en) 2015-11-26
AU2013200422A1 (en) 2013-03-21
EA022909B1 (ru) 2016-03-31
BR112014004732A2 (pt) 2017-03-28
EP2753609B1 (en) 2016-11-09
JP2017132781A (ja) 2017-08-03
UY34312A (es) 2013-04-30
KR101800140B1 (ko) 2017-11-21
CO6900147A2 (es) 2014-03-20
DK2753609T3 (en) 2017-02-06
US10251868B2 (en) 2019-04-09
ES2615052T3 (es) 2017-06-05
NZ621089A (en) 2015-07-31
AP2014007462A0 (en) 2014-02-28

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