UY34312A - Compuesto de benzotiazolona - Google Patents

Compuesto de benzotiazolona

Info

Publication number
UY34312A
UY34312A UY0001034312A UY34312A UY34312A UY 34312 A UY34312 A UY 34312A UY 0001034312 A UY0001034312 A UY 0001034312A UY 34312 A UY34312 A UY 34312A UY 34312 A UY34312 A UY 34312A
Authority
UY
Uruguay
Prior art keywords
benzotiazolona
composite
reivindicación
pág
fórmula
Prior art date
Application number
UY0001034312A
Other languages
English (en)
Inventor
Tufilli Nicola
Cao Jun
Erb Bernhard
Robin Alec Fairhurst
Grandeury Arnaud
Hatakeyama Shinji
Lai Xinzhong
Lustenberger Philipp
Riebesehl Bernd
Ullrich Thomas
Wu Xiang
Zhou Jianguang
Koziczakholbro Magdalena
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47010668&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY34312(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of UY34312A publication Critical patent/UY34312A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/08—Acetic acid
    • C07C53/10—Salts thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

La presente invención proporciona un compuesto de la fórmula (I) en forma libre o en forma de una sal farmacéuticamente aceptable un método para fabricar el compuesto de la invención, y sus usos terapéuticos. La presente invención proporciona además una combinación de agentes farmacológicamente activos y composiciones farmacéuticas.
UY0001034312A 2011-09-06 2012-09-05 Compuesto de benzotiazolona UY34312A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN2011079379 2011-09-06

Publications (1)

Publication Number Publication Date
UY34312A true UY34312A (es) 2013-04-30

Family

ID=47010668

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034312A UY34312A (es) 2011-09-06 2012-09-05 Compuesto de benzotiazolona

Country Status (38)

Country Link
US (6) US8933108B2 (es)
EP (1) EP2753609B1 (es)
JP (2) JP6130835B2 (es)
KR (2) KR101628585B1 (es)
CN (2) CN106187942B (es)
AP (1) AP3830A (es)
AR (1) AR087787A1 (es)
AU (1) AU2013200422C1 (es)
BR (1) BR112014004732A2 (es)
CA (1) CA2845766A1 (es)
CL (1) CL2014000493A1 (es)
CO (1) CO6900147A2 (es)
CR (1) CR20140114A (es)
CU (1) CU24303B1 (es)
CY (1) CY1118585T1 (es)
DK (1) DK2753609T3 (es)
EA (1) EA022909B1 (es)
ES (1) ES2615052T3 (es)
GT (1) GT201400042A (es)
HR (1) HRP20170075T1 (es)
HU (1) HUE030530T2 (es)
IL (1) IL231235A (es)
JO (1) JO3192B1 (es)
LT (1) LT2753609T (es)
MX (1) MX345405B (es)
MY (1) MY163301A (es)
PE (1) PE20141993A1 (es)
PL (1) PL2753609T3 (es)
PT (1) PT2753609T (es)
RS (1) RS55468B1 (es)
SG (1) SG2014013114A (es)
SI (1) SI2753609T1 (es)
TN (1) TN2014000060A1 (es)
TW (1) TWI555738B (es)
UA (1) UA114295C2 (es)
UY (1) UY34312A (es)
WO (1) WO2013035047A1 (es)
ZA (2) ZA201401112B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA117092C2 (uk) 2011-09-06 2018-06-25 Байєр Інтеллектуал Проперті Гмбх Амінозаміщені імідазопіридазини
JO3192B1 (ar) 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
DK2890687T3 (en) * 2012-08-30 2017-10-09 Novartis Ag Salts of benzothiazolone compound as beta-2-adrenoceptor agonist
CN104797585B (zh) 2012-11-19 2017-08-15 拜耳医药股份公司 氨基咪唑并哒嗪
WO2014132205A1 (en) 2013-02-28 2014-09-04 Novartis Ag Formulation comprising benzothiazolone compound
US10967119B1 (en) 2019-04-01 2021-04-06 Azizi Bilal Wearable medication injecting device

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DK2890687T3 (en) * 2012-08-30 2017-10-09 Novartis Ag Salts of benzothiazolone compound as beta-2-adrenoceptor agonist
WO2014132205A1 (en) 2013-02-28 2014-09-04 Novartis Ag Formulation comprising benzothiazolone compound

Also Published As

Publication number Publication date
JP2014525472A (ja) 2014-09-29
US10251868B2 (en) 2019-04-09
BR112014004732A2 (pt) 2017-03-28
SG2014013114A (en) 2014-07-30
AP3830A (en) 2016-09-30
ZA201401112B (en) 2016-01-27
IL231235A0 (en) 2014-04-30
CA2845766A1 (en) 2013-03-14
DK2753609T3 (en) 2017-02-06
IL231235A (en) 2017-09-28
MX2014002688A (es) 2014-04-14
CN106187942B (zh) 2020-06-26
HUE030530T2 (en) 2017-05-29
US20130245080A1 (en) 2013-09-19
UA114295C2 (uk) 2017-05-25
GT201400042A (es) 2015-02-19
PT2753609T (pt) 2017-02-08
AU2013200422A1 (en) 2013-03-21
TW201317221A (zh) 2013-05-01
CU24303B1 (es) 2018-01-10
CN103781771B (zh) 2016-08-24
US20150094346A1 (en) 2015-04-02
HRP20170075T1 (hr) 2017-03-24
CU20140028A7 (es) 2014-05-27
KR101800140B1 (ko) 2017-11-21
LT2753609T (lt) 2017-01-10
CN103781771A (zh) 2014-05-07
MY163301A (en) 2017-09-15
AU2013200422B2 (en) 2014-08-07
TN2014000060A1 (en) 2015-07-01
NZ621089A (en) 2015-07-31
US9913828B2 (en) 2018-03-13
ZA201500790B (en) 2017-04-26
TWI555738B (zh) 2016-11-01
US20150336914A1 (en) 2015-11-26
US20180140582A1 (en) 2018-05-24
KR20160038079A (ko) 2016-04-06
RS55468B1 (sr) 2017-04-28
JP6130835B2 (ja) 2017-05-17
CN106187942A (zh) 2016-12-07
KR20140057382A (ko) 2014-05-12
US20160075670A1 (en) 2016-03-17
KR101628585B1 (ko) 2016-06-08
ES2615052T3 (es) 2017-06-05
CL2014000493A1 (es) 2014-10-03
CO6900147A2 (es) 2014-03-20
AP2014007462A0 (en) 2014-02-28
CY1118585T1 (el) 2017-07-12
EA201490573A1 (ru) 2014-06-30
SI2753609T1 (sl) 2017-03-31
PE20141993A1 (es) 2014-12-17
US8933108B2 (en) 2015-01-13
US20160279107A1 (en) 2016-09-29
JP6340103B2 (ja) 2018-06-06
JO3192B1 (ar) 2018-03-08
CR20140114A (es) 2014-05-06
EP2753609B1 (en) 2016-11-09
MX345405B (es) 2017-01-30
PL2753609T3 (pl) 2017-05-31
JP2017132781A (ja) 2017-08-03
AU2013200422C1 (en) 2015-01-15
EA022909B1 (ru) 2016-03-31
EP2753609A1 (en) 2014-07-16
WO2013035047A1 (en) 2013-03-14
AR087787A1 (es) 2014-04-16

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Legal Events

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Effective date: 20201020