BR112015004127A2 - sais de composto benzotiazolona como agonista de beta-2-adrenorreceptor - Google Patents
sais de composto benzotiazolona como agonista de beta-2-adrenorreceptorInfo
- Publication number
- BR112015004127A2 BR112015004127A2 BR112015004127A BR112015004127A BR112015004127A2 BR 112015004127 A2 BR112015004127 A2 BR 112015004127A2 BR 112015004127 A BR112015004127 A BR 112015004127A BR 112015004127 A BR112015004127 A BR 112015004127A BR 112015004127 A2 BR112015004127 A2 BR 112015004127A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- salts
- beta
- present
- adrenoreceptor agonist
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
abstract the present invention provides a compound of formula (i) in acetate salt form (i) a method for manufacturing the compound of the invention, and its therapeutic uses. the present invention further provides a combination of pharmacologically active agents and pharmaceutical compositions. tradução do resumo resumo patente de invenção: "sais de composto benzotiazolona como agonista de beta-2-adrenorreceptor". a presente invenção refere-se a um composto de fórmula (i) em forma de sal de acetato (i), um método para fabricação do composto da invenção e seus usos terapêuticos. a presente invenção provê ainda uma combinação de agentes farmacologicamente ativos e composições farmacêuticas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IQ23912 | 2012-08-30 | ||
PCT/IB2013/058109 WO2014033654A1 (en) | 2012-08-30 | 2013-08-29 | Salts of benzothiazolone compound as beta-2-adrenoceptor agonist |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112015004127A2 true BR112015004127A2 (pt) | 2017-07-04 |
Family
ID=53386469
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015004127A BR112015004127A2 (pt) | 2012-08-30 | 2013-08-29 | sais de composto benzotiazolona como agonista de beta-2-adrenorreceptor |
Country Status (27)
Country | Link |
---|---|
EP (2) | EP2890687B1 (pt) |
KR (1) | KR20150047586A (pt) |
CN (2) | CN106146428A (pt) |
BR (1) | BR112015004127A2 (pt) |
CA (1) | CA2882877A1 (pt) |
CL (1) | CL2015000461A1 (pt) |
CY (1) | CY1120225T1 (pt) |
DK (1) | DK2890687T3 (pt) |
EA (1) | EA029946B1 (pt) |
ES (1) | ES2642003T3 (pt) |
HK (1) | HK1206015A1 (pt) |
HR (1) | HRP20171362T1 (pt) |
HU (1) | HUE033655T2 (pt) |
IL (1) | IL237382A0 (pt) |
LT (1) | LT2890687T (pt) |
MA (1) | MA37872A1 (pt) |
MX (1) | MX351741B (pt) |
MY (1) | MY169038A (pt) |
NZ (1) | NZ705319A (pt) |
PE (1) | PE20150465A1 (pt) |
PL (1) | PL2890687T3 (pt) |
PT (1) | PT2890687T (pt) |
SA (1) | SA515360076B1 (pt) |
SG (2) | SG10201704377PA (pt) |
SI (1) | SI2890687T1 (pt) |
TN (1) | TN2015000058A1 (pt) |
WO (1) | WO2014033654A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JO3192B1 (ar) * | 2011-09-06 | 2018-03-08 | Novartis Ag | مركب بنزوثيازولون |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20050130A1 (es) | 2002-08-09 | 2005-03-29 | Novartis Ag | Compuestos organicos |
EP1631260A2 (en) | 2003-02-28 | 2006-03-08 | Transform Pharmaceuticals, Inc. | Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen |
WO2005110990A1 (de) | 2004-05-13 | 2005-11-24 | Boehringer Ingelheim International Gmbh | Hydroxy-substituierte benzkondensierte heterozyklen als betaagonisten zur behandlung von atemwegserkrankungen |
GB0426164D0 (en) * | 2004-11-29 | 2004-12-29 | Novartis Ag | Organic compounds |
JO3192B1 (ar) * | 2011-09-06 | 2018-03-08 | Novartis Ag | مركب بنزوثيازولون |
LT2961391T (lt) * | 2013-02-28 | 2017-07-25 | Novartis Ag | Kompozicija, apimanti benzotiazolono junginį |
-
2013
- 2013-08-29 CN CN201610537241.9A patent/CN106146428A/zh active Pending
- 2013-08-29 EP EP13812075.3A patent/EP2890687B1/en active Active
- 2013-08-29 DK DK13812075.3T patent/DK2890687T3/en active
- 2013-08-29 ES ES13812075.3T patent/ES2642003T3/es active Active
- 2013-08-29 MA MA37872A patent/MA37872A1/fr unknown
- 2013-08-29 PT PT138120753T patent/PT2890687T/pt unknown
- 2013-08-29 BR BR112015004127A patent/BR112015004127A2/pt not_active Application Discontinuation
- 2013-08-29 PL PL13812075T patent/PL2890687T3/pl unknown
- 2013-08-29 SG SG10201704377PA patent/SG10201704377PA/en unknown
- 2013-08-29 KR KR1020157007573A patent/KR20150047586A/ko not_active Application Discontinuation
- 2013-08-29 EP EP17171708.5A patent/EP3243817A1/en not_active Withdrawn
- 2013-08-29 EA EA201590452A patent/EA029946B1/ru not_active IP Right Cessation
- 2013-08-29 CA CA2882877A patent/CA2882877A1/en not_active Abandoned
- 2013-08-29 NZ NZ705319A patent/NZ705319A/en not_active IP Right Cessation
- 2013-08-29 MY MYPI2015000453A patent/MY169038A/en unknown
- 2013-08-29 SG SG11201501293PA patent/SG11201501293PA/en unknown
- 2013-08-29 SI SI201330750T patent/SI2890687T1/sl unknown
- 2013-08-29 WO PCT/IB2013/058109 patent/WO2014033654A1/en active Application Filing
- 2013-08-29 PE PE2015000275A patent/PE20150465A1/es not_active Application Discontinuation
- 2013-08-29 CN CN201380055093.1A patent/CN104736525B/zh not_active Expired - Fee Related
- 2013-08-29 HU HUE13812075A patent/HUE033655T2/en unknown
- 2013-08-29 MX MX2015002656A patent/MX351741B/es active IP Right Grant
- 2013-08-29 LT LTEP13812075.3T patent/LT2890687T/lt unknown
-
2015
- 2015-02-20 TN TNP2015000058A patent/TN2015000058A1/fr unknown
- 2015-02-23 IL IL237382A patent/IL237382A0/en unknown
- 2015-02-25 CL CL2015000461A patent/CL2015000461A1/es unknown
- 2015-02-26 SA SA515360076A patent/SA515360076B1/ar unknown
- 2015-07-08 HK HK15106522.7A patent/HK1206015A1/xx not_active IP Right Cessation
-
2017
- 2017-09-11 HR HRP20171362TT patent/HRP20171362T1/hr unknown
- 2017-09-13 CY CY20171100967T patent/CY1120225T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
IL237382A0 (en) | 2015-04-30 |
DK2890687T3 (en) | 2017-10-09 |
WO2014033654A1 (en) | 2014-03-06 |
HK1206015A1 (en) | 2015-12-31 |
CA2882877A1 (en) | 2014-03-06 |
HUE033655T2 (en) | 2017-12-28 |
CN106146428A (zh) | 2016-11-23 |
TN2015000058A1 (en) | 2016-06-29 |
CL2015000461A1 (es) | 2015-05-04 |
CY1120225T1 (el) | 2018-12-12 |
EA029946B1 (ru) | 2018-06-29 |
SG11201501293PA (en) | 2015-03-30 |
HRP20171362T1 (hr) | 2017-11-03 |
EP3243817A1 (en) | 2017-11-15 |
EP2890687A1 (en) | 2015-07-08 |
EP2890687B1 (en) | 2017-06-28 |
MX351741B (es) | 2017-10-26 |
ES2642003T3 (es) | 2017-11-14 |
EA201590452A1 (ru) | 2015-07-30 |
NZ705319A (en) | 2018-05-25 |
PL2890687T3 (pl) | 2017-11-30 |
MA37872A1 (fr) | 2018-07-31 |
LT2890687T (lt) | 2017-09-11 |
SI2890687T1 (sl) | 2017-10-30 |
PT2890687T (pt) | 2017-10-05 |
MY169038A (en) | 2019-02-07 |
SA515360076B1 (ar) | 2016-03-20 |
PE20150465A1 (es) | 2015-04-22 |
CN104736525B (zh) | 2016-08-24 |
MX2015002656A (es) | 2015-05-20 |
CN104736525A (zh) | 2015-06-24 |
SG10201704377PA (en) | 2017-06-29 |
KR20150047586A (ko) | 2015-05-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
B11E | Dismissal acc. art. 34 of ipl - requirements for examination incomplete | ||
B11T | Dismissal of application maintained [chapter 11.20 patent gazette] |