MA37872A1 - Sels de composé benzothiazolone utilisés en tant qu'agoniste de beta-2-adrenoceptor - Google Patents

Sels de composé benzothiazolone utilisés en tant qu'agoniste de beta-2-adrenoceptor

Info

Publication number
MA37872A1
MA37872A1 MA37872A MA37872A MA37872A1 MA 37872 A1 MA37872 A1 MA 37872A1 MA 37872 A MA37872 A MA 37872A MA 37872 A MA37872 A MA 37872A MA 37872 A1 MA37872 A1 MA 37872A1
Authority
MA
Morocco
Prior art keywords
beta
salts used
adrenoceptor agonist
compound salts
benzothiazolone compound
Prior art date
Application number
MA37872A
Other languages
English (en)
Inventor
Arnaud Grandeury
Nicola Tufilli
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53386469&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA37872(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA37872A1 publication Critical patent/MA37872A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La présente invention concerne un composé de formule (i) sous forme de sel acétate (i), un procédé de fabrication du composé de l'invention et ses utilisations thérapeutiques. La présente invention concerne de plus une combinaison de principes pharmacologiquement actifs et des compositions pharmaceutiques.
MA37872A 2012-08-30 2013-08-29 Sels de composé benzothiazolone utilisés en tant qu'agoniste de beta-2-adrenoceptor MA37872A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IQ23912 2012-08-30
PCT/IB2013/058109 WO2014033654A1 (fr) 2012-08-30 2013-08-29 Sels de composé benzothiazolone utilisés en tant qu'agoniste de beta-2-adrenoceptor

Publications (1)

Publication Number Publication Date
MA37872A1 true MA37872A1 (fr) 2018-07-31

Family

ID=53386469

Family Applications (1)

Application Number Title Priority Date Filing Date
MA37872A MA37872A1 (fr) 2012-08-30 2013-08-29 Sels de composé benzothiazolone utilisés en tant qu'agoniste de beta-2-adrenoceptor

Country Status (27)

Country Link
EP (2) EP3243817A1 (fr)
KR (1) KR20150047586A (fr)
CN (2) CN106146428A (fr)
BR (1) BR112015004127A2 (fr)
CA (1) CA2882877A1 (fr)
CL (1) CL2015000461A1 (fr)
CY (1) CY1120225T1 (fr)
DK (1) DK2890687T3 (fr)
EA (1) EA029946B1 (fr)
ES (1) ES2642003T3 (fr)
HK (1) HK1206015A1 (fr)
HR (1) HRP20171362T1 (fr)
HU (1) HUE033655T2 (fr)
IL (1) IL237382A0 (fr)
LT (1) LT2890687T (fr)
MA (1) MA37872A1 (fr)
MX (1) MX351741B (fr)
MY (1) MY169038A (fr)
NZ (1) NZ705319A (fr)
PE (1) PE20150465A1 (fr)
PL (1) PL2890687T3 (fr)
PT (1) PT2890687T (fr)
SA (1) SA515360076B1 (fr)
SG (2) SG11201501293PA (fr)
SI (1) SI2890687T1 (fr)
TN (1) TN2015000058A1 (fr)
WO (1) WO2014033654A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3192B1 (ar) 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR040962A1 (es) 2002-08-09 2005-04-27 Novartis Ag Compuestos derivados de tiazol 1,3-2-ona, composicion farmaceutica y proceso de preparacion del compuesto
CA2514733A1 (fr) 2003-02-28 2004-09-16 Transform Pharmaceuticals, Inc. Compositions pharmaceutiques a base d'un co-cristal
JP2007537187A (ja) 2004-05-13 2007-12-20 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 呼吸器疾患の治療においてβアゴニストとして使用するためのヒドロキシ置換ベンゾ縮合ヘテロ環化合物
GB0426164D0 (en) * 2004-11-29 2004-12-29 Novartis Ag Organic compounds
JO3192B1 (ar) * 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
AU2014222362B2 (en) * 2013-02-28 2016-07-21 Novartis Ag Formulation comprising benzothiazolone compound

Also Published As

Publication number Publication date
LT2890687T (lt) 2017-09-11
NZ705319A (en) 2018-05-25
PT2890687T (pt) 2017-10-05
BR112015004127A2 (pt) 2017-07-04
HRP20171362T1 (hr) 2017-11-03
CN104736525B (zh) 2016-08-24
SG11201501293PA (en) 2015-03-30
MX351741B (es) 2017-10-26
KR20150047586A (ko) 2015-05-04
SI2890687T1 (sl) 2017-10-30
CN104736525A (zh) 2015-06-24
TN2015000058A1 (en) 2016-06-29
PL2890687T3 (pl) 2017-11-30
MY169038A (en) 2019-02-07
EA201590452A1 (ru) 2015-07-30
MX2015002656A (es) 2015-05-20
ES2642003T3 (es) 2017-11-14
EP3243817A1 (fr) 2017-11-15
HUE033655T2 (en) 2017-12-28
HK1206015A1 (en) 2015-12-31
SA515360076B1 (ar) 2016-03-20
EA029946B1 (ru) 2018-06-29
IL237382A0 (en) 2015-04-30
WO2014033654A1 (fr) 2014-03-06
SG10201704377PA (en) 2017-06-29
DK2890687T3 (en) 2017-10-09
CL2015000461A1 (es) 2015-05-04
EP2890687B1 (fr) 2017-06-28
CA2882877A1 (fr) 2014-03-06
EP2890687A1 (fr) 2015-07-08
PE20150465A1 (es) 2015-04-22
CY1120225T1 (el) 2018-12-12
CN106146428A (zh) 2016-11-23

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