MA37872A1 - Benzothiazolone compound salts used as a beta-2-adrenoceptor agonist - Google Patents

Benzothiazolone compound salts used as a beta-2-adrenoceptor agonist

Info

Publication number
MA37872A1
MA37872A1 MA37872A MA37872A MA37872A1 MA 37872 A1 MA37872 A1 MA 37872A1 MA 37872 A MA37872 A MA 37872A MA 37872 A MA37872 A MA 37872A MA 37872 A1 MA37872 A1 MA 37872A1
Authority
MA
Morocco
Prior art keywords
beta
salts used
adrenoceptor agonist
compound salts
benzothiazolone compound
Prior art date
Application number
MA37872A
Other languages
French (fr)
Inventor
Arnaud Grandeury
Nicola Tufilli
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53386469&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA37872(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA37872A1 publication Critical patent/MA37872A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La présente invention concerne un composé de formule (i) sous forme de sel acétate (i), un procédé de fabrication du composé de l'invention et ses utilisations thérapeutiques. La présente invention concerne de plus une combinaison de principes pharmacologiquement actifs et des compositions pharmaceutiques.The present invention relates to a compound of formula (i) in acetate salt form (i), a process for producing the compound of the invention and its therapeutic uses. The present invention further relates to a combination of pharmacologically active principles and pharmaceutical compositions.

MA37872A 2012-08-30 2013-08-29 Benzothiazolone compound salts used as a beta-2-adrenoceptor agonist MA37872A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IQ23912 2012-08-30
PCT/IB2013/058109 WO2014033654A1 (en) 2012-08-30 2013-08-29 Salts of benzothiazolone compound as beta-2-adrenoceptor agonist

Publications (1)

Publication Number Publication Date
MA37872A1 true MA37872A1 (en) 2018-07-31

Family

ID=53386469

Family Applications (1)

Application Number Title Priority Date Filing Date
MA37872A MA37872A1 (en) 2012-08-30 2013-08-29 Benzothiazolone compound salts used as a beta-2-adrenoceptor agonist

Country Status (27)

Country Link
EP (2) EP3243817A1 (en)
KR (1) KR20150047586A (en)
CN (2) CN106146428A (en)
BR (1) BR112015004127A2 (en)
CA (1) CA2882877A1 (en)
CL (1) CL2015000461A1 (en)
CY (1) CY1120225T1 (en)
DK (1) DK2890687T3 (en)
EA (1) EA029946B1 (en)
ES (1) ES2642003T3 (en)
HK (1) HK1206015A1 (en)
HR (1) HRP20171362T1 (en)
HU (1) HUE033655T2 (en)
IL (1) IL237382A0 (en)
LT (1) LT2890687T (en)
MA (1) MA37872A1 (en)
MX (1) MX351741B (en)
MY (1) MY169038A (en)
NZ (1) NZ705319A (en)
PE (1) PE20150465A1 (en)
PL (1) PL2890687T3 (en)
PT (1) PT2890687T (en)
SA (1) SA515360076B1 (en)
SG (2) SG11201501293PA (en)
SI (1) SI2890687T1 (en)
TN (1) TN2015000058A1 (en)
WO (1) WO2014033654A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3192B1 (en) * 2011-09-06 2018-03-08 Novartis Ag Benzothiazolone compound

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR040962A1 (en) 2002-08-09 2005-04-27 Novartis Ag COMPOUNDS DERIVED FROM TIAZOL 1,3-2-ONA, PHARMACEUTICAL COMPOSITION AND COMPOSITE PREPARATION PROCESS
CA2514733A1 (en) 2003-02-28 2004-09-16 Transform Pharmaceuticals, Inc. Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen
WO2005110990A1 (en) 2004-05-13 2005-11-24 Boehringer Ingelheim International Gmbh Hydroxy-substituted benzo-condensed heterocycles for use as beta agonists in the treatment of respiratory diseases
GB0426164D0 (en) * 2004-11-29 2004-12-29 Novartis Ag Organic compounds
JO3192B1 (en) * 2011-09-06 2018-03-08 Novartis Ag Benzothiazolone compound
PL2961391T3 (en) * 2013-02-28 2017-10-31 Novartis Ag Formulation comprising benzothiazolone compound

Also Published As

Publication number Publication date
ES2642003T3 (en) 2017-11-14
PE20150465A1 (en) 2015-04-22
BR112015004127A2 (en) 2017-07-04
LT2890687T (en) 2017-09-11
MY169038A (en) 2019-02-07
EA201590452A1 (en) 2015-07-30
SG11201501293PA (en) 2015-03-30
HK1206015A1 (en) 2015-12-31
WO2014033654A1 (en) 2014-03-06
CN104736525A (en) 2015-06-24
CN106146428A (en) 2016-11-23
CL2015000461A1 (en) 2015-05-04
PL2890687T3 (en) 2017-11-30
CA2882877A1 (en) 2014-03-06
HRP20171362T1 (en) 2017-11-03
EP2890687A1 (en) 2015-07-08
MX2015002656A (en) 2015-05-20
EP2890687B1 (en) 2017-06-28
IL237382A0 (en) 2015-04-30
DK2890687T3 (en) 2017-10-09
EP3243817A1 (en) 2017-11-15
PT2890687T (en) 2017-10-05
CN104736525B (en) 2016-08-24
NZ705319A (en) 2018-05-25
SA515360076B1 (en) 2016-03-20
SG10201704377PA (en) 2017-06-29
SI2890687T1 (en) 2017-10-30
HUE033655T2 (en) 2017-12-28
MX351741B (en) 2017-10-26
CY1120225T1 (en) 2018-12-12
KR20150047586A (en) 2015-05-04
EA029946B1 (en) 2018-06-29
TN2015000058A1 (en) 2016-06-29

Similar Documents

Publication Publication Date Title
CY1124882T1 (en) 1,4-DI-CONSTITUTED PYRIDAZINE ANALOGUES AND METHODS FOR THERAPEUTIC TREATMENT OF CONDITIONS RELATED TO SMN DEFICIENCY
MA37477A1 (en) Modulators of complement pathways and their uses
MA37405A1 (en) Heterocyclyl compounds
MA34837B1 (en) INDOLIC COMPOUNDS OR ANALOGS THEREFOR USEFUL IN THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION (AMD)
MA35275B1 (en) Compounds of tetrahydropyridopyridine and tetrahydropyridopyrimidine and their use as c5a receptor modulators
EA201592255A1 (en) DERIVATIVES OF PYRAZOLOPIRROLIDIN-4-IT AS A BET INHIBITOR AND THEIR APPLICATION IN THE TREATMENT OF THE DISEASE
MA33364B1 (en) SUBSTITUTED AMINOBUTYRIC DERIVATIVES AS NEPRILYSIN INHIBITORS
EA201592256A1 (en) DERIVATIVES OF IMIDAZOPIRROLIDINONE AND THEIR APPLICATION IN THE TREATMENT OF DISEASES
MD20160078A2 (en) Syk inhibitors
MA35032B1 (en) GLYCOSIDE DERIVATIVES AND THEIR USES IN THE TREATMENT OF DIABETES
MA38330A1 (en) Butanoic phosphonic acid derivatives of bisphenol substituted as nep inhibitors (neutral endopeptidase)
EA201690247A1 (en) AMINOMETHYBYRIL DERIVATIVES-INHIBITORS OF COMPLEX D FACTOR AND USE
EA201492023A1 (en) REGULATORS OF THE COMPLEX WAY AND THEIR APPLICATION
PH12015502802A1 (en) Formulation comprising a hypolipidemic agent
MA39983A (en) CARBOXAMIDE DERIVATIVES
MX2021010046A (en) A new therapeutical composition containing apomorphine as active ingredient.
UA103329C2 (en) Normal;heading 1;heading 2;heading 3;SALTS OF HIV INHIBITOR COMPOUNDS
IN2014DN05972A (en)
EA201490573A1 (en) CONTAINING BENZOTHIAZOLONE
MA37872A1 (en) Benzothiazolone compound salts used as a beta-2-adrenoceptor agonist
EA201591487A1 (en) DERIVATIVES OF SUBSTITUTED BISFENILBUTANIC ACID AS NEP INHIBITORS WITH IMPROVED IN VIVO EFFICIENCY
IN2014MN02433A (en)
MA37879B1 (en) Stabilized amorphous form of agomelatine, process for its preparation and pharmaceutical compositions containing it
EA201490342A1 (en) DERIVATIVES OF PYRAZOLINE AND THEIR APPLICATION AS A SELECTIVE MODULATOR OF THE ANDROGEN RECEPTOR
MA34462B1 (en) 2,3,5-TRISUBSTITUTED THIOPHENE COMPOUNDS AND USES THEREOF