PE20141378A1 - Moduladores de receptores de glucocorticoides de pirimidina ciclohexilo - Google Patents

Moduladores de receptores de glucocorticoides de pirimidina ciclohexilo

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Publication number
PE20141378A1
PE20141378A1 PE2013002053A PE2013002053A PE20141378A1 PE 20141378 A1 PE20141378 A1 PE 20141378A1 PE 2013002053 A PE2013002053 A PE 2013002053A PE 2013002053 A PE2013002053 A PE 2013002053A PE 20141378 A1 PE20141378 A1 PE 20141378A1
Authority
PE
Peru
Prior art keywords
glucocorticoid receptors
alkyl
receptors modulators
modulators
pyrimidine
Prior art date
Application number
PE2013002053A
Other languages
English (en)
Inventor
Robin Clark
George Hynd
Nicholas Ray
Mohammad Sajad
Original Assignee
Corcept Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Corcept Therapeutics Inc filed Critical Corcept Therapeutics Inc
Publication of PE20141378A1 publication Critical patent/PE20141378A1/es

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Abstract

SE REFIERE A COMPUESTOS DE FORMULA (I) DONDE: LA LINEA DE GUIONES ESTA AUSENTE O ES UN ENLACE; X ES O Y S; R1 SE SELECCIONA DE CICLOALQUILO, HETEROCICLOALQUILO, ARILO Y HETEROARILO, OPCIONALMENTE SUSTITUIDO; R2 ES H, ALQUILO C1-6, ALQUILO C1-6-OR1b, ENTRE OTROS, R1b ES H Y ALQUILO C1-6; R3 SE SELECCIONA DE H Y ALQUILO C1-6; Ar ES ARILO OPCIONALMENTE SUSTITUIDO; L1 ES UN ENLACE O ALQUILENO C1-6; n ES UN NUMERO ENTERO DE 0 A 3. SE REFIERE TAMBIEN A UNA COMPOSICION FARMACEUTICA. DICHOS COMPUESTOS SON MODULADORES DE RECEPTORES DE GLUCOCORTICOIDES
PE2013002053A 2011-03-18 2012-03-16 Moduladores de receptores de glucocorticoides de pirimidina ciclohexilo PE20141378A1 (es)

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