PE20120654A1 - Formulaciones de 4-amino-2-(2,6-dioxopiperidin-1,3-il) isoindolin-1,3-diona - Google Patents

Formulaciones de 4-amino-2-(2,6-dioxopiperidin-1,3-il) isoindolin-1,3-diona

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Publication number
PE20120654A1
PE20120654A1 PE2011001611A PE2011001611A PE20120654A1 PE 20120654 A1 PE20120654 A1 PE 20120654A1 PE 2011001611 A PE2011001611 A PE 2011001611A PE 2011001611 A PE2011001611 A PE 2011001611A PE 20120654 A1 PE20120654 A1 PE 20120654A1
Authority
PE
Peru
Prior art keywords
diona
dioxopiperidin
isoindolin
formulations
amino
Prior art date
Application number
PE2011001611A
Other languages
English (en)
Inventor
Anthony Tutino
Michael T Kelly
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42635489&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20120654(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of PE20120654A1 publication Critical patent/PE20120654A1/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Pulmonology (AREA)
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  • Hematology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)

Abstract

REFERIDA A UNA FORMA DE DOSIFICACION ORAL QUE COMPRENDE: 1) POMALIDOMIDA O UNA SAL O SOLVATO FARMACEUTICAMENTE ACEPTABLE DE LA MISMA, EN UNA CANTIDAD QUE PROPORCIONA 0.5 mg-4 mg DE POTENCIA DE POLIDOMIDA; B) UN PORTADOR O EXCIPIENTE FARMACEUTICAMENTE ACEPTABLE SELECCIONADO DE ALMIDON PREGELATINIZADO, ESTEARILFUMARATO DE SODIO, MANITOL, ENTRE OTROS. DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE CANCER, DOLOR, TRASTORNO PULMONAR, ENFERMEDAD PARASITICA, ENTRE OTROS
PE2011001611A 2009-05-19 2010-05-19 Formulaciones de 4-amino-2-(2,6-dioxopiperidin-1,3-il) isoindolin-1,3-diona PE20120654A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17967809P 2009-05-19 2009-05-19

Publications (1)

Publication Number Publication Date
PE20120654A1 true PE20120654A1 (es) 2012-05-31

Family

ID=42635489

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PE2011001611A PE20120654A1 (es) 2009-05-19 2010-05-19 Formulaciones de 4-amino-2-(2,6-dioxopiperidin-1,3-il) isoindolin-1,3-diona

Country Status (34)

Country Link
US (6) US8828427B2 (es)
EP (3) EP3199149A1 (es)
JP (1) JP5752677B2 (es)
KR (1) KR101381060B1 (es)
CN (3) CN105640918A (es)
AU (1) AU2010249615B2 (es)
BR (1) BRPI1007855B1 (es)
CA (1) CA2752550C (es)
CL (1) CL2011001969A1 (es)
CO (1) CO6430422A2 (es)
CR (1) CR20110435A (es)
CY (2) CY1118632T1 (es)
DK (2) DK3351240T3 (es)
EC (1) ECSP11011317A (es)
ES (2) ES2728776T3 (es)
HR (2) HRP20170179T1 (es)
HU (2) HUE043862T2 (es)
IL (2) IL214644A (es)
LT (2) LT3351240T (es)
MX (2) MX342330B (es)
NI (1) NI201100158A (es)
NZ (1) NZ594557A (es)
PE (1) PE20120654A1 (es)
PH (1) PH12015501523A1 (es)
PL (2) PL2391355T3 (es)
PT (2) PT3351240T (es)
RU (1) RU2479307C1 (es)
SG (1) SG174137A1 (es)
SI (2) SI3351240T1 (es)
SM (1) SMT201700097B (es)
TR (1) TR201905423T4 (es)
UA (1) UA102582C2 (es)
WO (1) WO2010135396A2 (es)
ZA (1) ZA201105962B (es)

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