MX342330B - Formulaciones de 4-amino-2-(2, 6-dioxopiperidin-3-il) isoindolin-1, 3-diona. - Google Patents

Formulaciones de 4-amino-2-(2, 6-dioxopiperidin-3-il) isoindolin-1, 3-diona.

Info

Publication number
MX342330B
MX342330B MX2014014182A MX2014014182A MX342330B MX 342330 B MX342330 B MX 342330B MX 2014014182 A MX2014014182 A MX 2014014182A MX 2014014182 A MX2014014182 A MX 2014014182A MX 342330 B MX342330 B MX 342330B
Authority
MX
Mexico
Prior art keywords
dioxopiperidine
isoindoline
dione
amino
formulations
Prior art date
Application number
MX2014014182A
Other languages
English (en)
Inventor
T Kelly Michael
Tutino Anthony
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42635489&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX342330(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of MX342330B publication Critical patent/MX342330B/es

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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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Abstract

Se proporcionan en la presente, composiciones farmacéuticas y formas de unidad de dosis sencilla de 4-amino-2-(2,6-dioxopiperidi na-3-il)isoindolin-1,3-diona, o un estereoisómero, profármaco, sal, solvato, hidrato o clatrato, farmacéuticamente aceptable. También se proporcionan métodos para tratar, manejar o prevenir varios trastornos, tales como cáncer o una enfermedad inflamatoria.
MX2014014182A 2009-05-19 2010-05-19 Formulaciones de 4-amino-2-(2, 6-dioxopiperidin-3-il) isoindolin-1, 3-diona. MX342330B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17967809P 2009-05-19 2009-05-19
PCT/US2010/035357 WO2010135396A2 (en) 2009-05-19 2010-05-19 Formulations of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione

Publications (1)

Publication Number Publication Date
MX342330B true MX342330B (es) 2016-09-26

Family

ID=42635489

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2014014182A MX342330B (es) 2009-05-19 2010-05-19 Formulaciones de 4-amino-2-(2, 6-dioxopiperidin-3-il) isoindolin-1, 3-diona.
MX2011008554A MX2011008554A (es) 2009-05-19 2010-05-19 Formulaciones de 4-amino-2-(2,6-dioxopiperidin-3-il) isoindolin-1,3-diona.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2011008554A MX2011008554A (es) 2009-05-19 2010-05-19 Formulaciones de 4-amino-2-(2,6-dioxopiperidin-3-il) isoindolin-1,3-diona.

Country Status (34)

Country Link
US (6) US8828427B2 (es)
EP (3) EP3199149A1 (es)
JP (1) JP5752677B2 (es)
KR (1) KR101381060B1 (es)
CN (3) CN105640918A (es)
AU (1) AU2010249615B2 (es)
BR (1) BRPI1007855B1 (es)
CA (1) CA2752550C (es)
CL (1) CL2011001969A1 (es)
CO (1) CO6430422A2 (es)
CR (1) CR20110435A (es)
CY (2) CY1118632T1 (es)
DK (2) DK3351240T3 (es)
EC (1) ECSP11011317A (es)
ES (2) ES2728776T3 (es)
HR (2) HRP20170179T1 (es)
HU (2) HUE043862T2 (es)
IL (2) IL214644A (es)
LT (2) LT3351240T (es)
MX (2) MX342330B (es)
NI (1) NI201100158A (es)
NZ (1) NZ594557A (es)
PE (1) PE20120654A1 (es)
PH (1) PH12015501523A1 (es)
PL (2) PL2391355T3 (es)
PT (2) PT3351240T (es)
RU (1) RU2479307C1 (es)
SG (1) SG174137A1 (es)
SI (2) SI3351240T1 (es)
SM (1) SMT201700097B (es)
TR (1) TR201905423T4 (es)
UA (1) UA102582C2 (es)
WO (1) WO2010135396A2 (es)
ZA (1) ZA201105962B (es)

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