DK3351240T3 - Formuleringer af 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindolin-1,3-dion - Google Patents

Formuleringer af 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindolin-1,3-dion Download PDF

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Publication number
DK3351240T3
DK3351240T3 DK18160247.5T DK18160247T DK3351240T3 DK 3351240 T3 DK3351240 T3 DK 3351240T3 DK 18160247 T DK18160247 T DK 18160247T DK 3351240 T3 DK3351240 T3 DK 3351240T3
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Prior art keywords
dioxopiperidin
isoindolin
dion
formulations
amino
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DK18160247.5T
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English (en)
Inventor
Anthony Tutino
Michael T Kelly
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Celgene Corp
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
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    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
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    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
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    • A61K9/4866Organic macromolecular compounds
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
DK18160247.5T 2009-05-19 2010-05-19 Formuleringer af 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindolin-1,3-dion DK3351240T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17967809P 2009-05-19 2009-05-19
EP17151178.5A EP3199149A1 (en) 2009-05-19 2010-05-19 Formulations of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione

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DK3351240T3 true DK3351240T3 (da) 2019-06-17

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DK18160247.5T DK3351240T3 (da) 2009-05-19 2010-05-19 Formuleringer af 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindolin-1,3-dion
DK10720107.1T DK2391355T3 (da) 2009-05-19 2010-05-19 Formuleringer af 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindolin-1,3-dion

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US (6) US8828427B2 (da)
EP (3) EP2391355B1 (da)
JP (1) JP5752677B2 (da)
KR (1) KR101381060B1 (da)
CN (3) CN106176662A (da)
AU (1) AU2010249615B2 (da)
BR (1) BRPI1007855B1 (da)
CA (1) CA2752550C (da)
CL (1) CL2011001969A1 (da)
CO (1) CO6430422A2 (da)
CR (1) CR20110435A (da)
CY (2) CY1118632T1 (da)
DK (2) DK3351240T3 (da)
EC (1) ECSP11011317A (da)
ES (2) ES2615511T3 (da)
HR (2) HRP20170179T1 (da)
HU (2) HUE033115T2 (da)
IL (2) IL214644A (da)
LT (2) LT3351240T (da)
MX (2) MX342330B (da)
NI (1) NI201100158A (da)
NZ (1) NZ594557A (da)
PE (1) PE20120654A1 (da)
PH (1) PH12015501523A1 (da)
PL (2) PL3351240T3 (da)
PT (2) PT3351240T (da)
RU (1) RU2479307C1 (da)
SG (1) SG174137A1 (da)
SI (2) SI3351240T1 (da)
SM (1) SMT201700097B (da)
TR (1) TR201905423T4 (da)
UA (1) UA102582C2 (da)
WO (1) WO2010135396A2 (da)
ZA (1) ZA201105962B (da)

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