PE13395A1 - Composicion farmaceutica de imidazolil carbazolona - Google Patents

Composicion farmaceutica de imidazolil carbazolona

Info

Publication number
PE13395A1
PE13395A1 PE1994242905A PE24290594A PE13395A1 PE 13395 A1 PE13395 A1 PE 13395A1 PE 1994242905 A PE1994242905 A PE 1994242905A PE 24290594 A PE24290594 A PE 24290594A PE 13395 A1 PE13395 A1 PE 13395A1
Authority
PE
Peru
Prior art keywords
pharmaceutical composition
carbazolona
imidazolil
methyl
hydroxitriptamine
Prior art date
Application number
PE1994242905A
Other languages
English (en)
Inventor
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Lab Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Lab Sa filed Critical Glaxo Lab Sa
Publication of PE13395A1 publication Critical patent/PE13395A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/02Suppositories; Bougies; Bases therefor; Ovules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA PARA ADMINISTRACION RECTAL QUE COMPRENDE: 1) 1,2,3,9-TETRAHIDRO-9-METIL-3-((2-METIL-1H-IMIDAZOL-1-IL)-METIL)-4H-CARBAZOL-4-ONA DE FORMULA I; EN FORMA DE BASE LIBRE O UN SOLVATO A UNA CONCENTRACION DE 0,1 mg A 100 mg; PUDIENDO SER UTIL EN EL TRATAMIENTO DE LA NAUSEA Y EL VOMITO AL SER UN ANTAGONISTA DE LA 5-HIDROXITRIPTAMINA (5-HT); 2) EXCIPIENTES TALES COMO BASES GRASAS CON UN VALOR DE HIDROXILO DE 20 A 100, PUDIENDO PRESENTARSE EN UNA FORMA SOLIDA TAL COMO UN SUPOSITORIO
PE1994242905A 1993-05-25 1994-05-23 Composicion farmaceutica de imidazolil carbazolona PE13395A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939310756A GB9310756D0 (en) 1993-05-25 1993-05-25 Compositions

Publications (1)

Publication Number Publication Date
PE13395A1 true PE13395A1 (es) 1995-05-25

Family

ID=10736089

Family Applications (1)

Application Number Title Priority Date Filing Date
PE1994242905A PE13395A1 (es) 1993-05-25 1994-05-23 Composicion farmaceutica de imidazolil carbazolona

Country Status (38)

Country Link
US (1) US5741806A (es)
EP (1) EP0700290B1 (es)
JP (1) JP2965703B2 (es)
KR (1) KR100297212B1 (es)
CN (1) CN1106194C (es)
AP (1) AP544A (es)
AT (1) ATE183643T1 (es)
AU (1) AU680918B2 (es)
BE (1) BE1007158A3 (es)
BR (1) BR1100046A (es)
CA (1) CA2162919C (es)
CO (1) CO4230094A1 (es)
CY (1) CY2411B1 (es)
CZ (1) CZ291041B6 (es)
DE (1) DE69420266T2 (es)
DK (1) DK0700290T3 (es)
EC (1) ECSP941088A (es)
ES (1) ES2136198T3 (es)
FR (1) FR2705569B1 (es)
GB (2) GB9310756D0 (es)
GR (1) GR3031669T3 (es)
HR (2) HRP940315B1 (es)
HU (1) HU227121B1 (es)
IE (1) IE80632B1 (es)
IL (1) IL109749A (es)
IS (1) IS1868B (es)
IT (1) IT1272990B (es)
MY (1) MY111445A (es)
NO (1) NO306448B1 (es)
NZ (1) NZ267415A (es)
PE (1) PE13395A1 (es)
PL (1) PL175578B1 (es)
RU (1) RU2132684C1 (es)
SA (1) SA94150003B1 (es)
SG (1) SG48119A1 (es)
SI (1) SI0700290T1 (es)
WO (1) WO1994027599A1 (es)
ZA (1) ZA943593B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1468685A3 (en) * 1998-06-15 2004-12-15 Sepracor Inc. Use of optically pure (+)-norcisapride for treating apnea, bulimia and other disorders
EP1464333A3 (en) * 1998-06-15 2004-12-15 Sepracor Inc. Use of optically pure (-) norcisapride in the treatment of apnea, bulimia, and other disorders
TR200103757T2 (tr) * 1998-06-15 2002-06-21 Sepracor Inc. Apne, bulimi ve başka bozuklukların tedavi edilmesi için optik açıdan saf (-) norsisapridin kullanımı
IL140118A0 (en) * 1998-06-15 2002-02-10 Sepracor Inc Use of optically pure (+) norcisapride for treating apnea, bulimia and other disorders
US6353005B1 (en) 1999-03-02 2002-03-05 Sepracor, Inc. Method and compositions using (+) norcisapride in combination with proton pump inhibitors or H2 receptor antagonist
US6362202B1 (en) 1999-03-02 2002-03-26 Sepracor Inc. Methods and compositions using (−) norcisapride in combination with proton pump inhibitors or H2 receptor antagonists
BR0112969A (pt) * 2000-08-04 2004-06-22 Dmi Biosciences Inc Método de utilização de dicetopiperazinas e composições contendo-as

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2561244B1 (fr) * 1984-01-25 1988-03-04 Glaxo Group Ltd Composes heterocycliques du type tetrahydrocarbazolone, procede pour leur preparation et composition pharmaceutique les comprenant
US4695578A (en) * 1984-01-25 1987-09-22 Glaxo Group Limited 1,2,3,9-tetrahydro-3-imidazol-1-ylmethyl-4H-carbazol-4-ones, composition containing them, and method of using them to treat neuronal 5HT function disturbances
GB8627909D0 (en) * 1986-11-21 1986-12-31 Glaxo Group Ltd Medicaments
GB8816187D0 (en) * 1988-07-07 1988-08-10 Glaxo Group Ltd Medicaments
US5166145A (en) * 1990-09-10 1992-11-24 Alza Corporation Antiemetic therapy

Also Published As

Publication number Publication date
IE80632B1 (en) 1998-10-21
RU2132684C1 (ru) 1999-07-10
IT1272990B (it) 1997-07-01
DE69420266T2 (de) 1999-12-09
PL175578B1 (pl) 1999-01-29
CA2162919C (en) 1999-07-20
CO4230094A1 (es) 1995-10-19
GB2279008B (en) 1997-06-18
IL109749A (en) 1999-03-12
SA94150003B1 (ar) 2005-04-11
GB9310756D0 (en) 1993-07-14
GB9409835D0 (en) 1994-07-06
ES2136198T3 (es) 1999-11-16
CY2411B1 (en) 2004-11-12
IS1868B (is) 2003-05-02
GB2279008A (en) 1994-12-21
GR3031669T3 (en) 2000-02-29
IE940420A1 (en) 1994-11-30
EP0700290A1 (en) 1996-03-13
NO306448B1 (no) 1999-11-08
AP9400643A0 (en) 1994-07-31
IS4168A (is) 1994-11-26
DE69420266D1 (de) 1999-09-30
AU6970994A (en) 1994-12-20
CZ308595A3 (en) 1996-06-12
FR2705569B1 (fr) 1995-11-10
ATE183643T1 (de) 1999-09-15
SG48119A1 (en) 1998-04-17
FR2705569A1 (fr) 1994-12-02
EP0700290B1 (en) 1999-08-25
MY111445A (en) 2000-05-31
CN1124454A (zh) 1996-06-12
BE1007158A3 (fr) 1995-04-11
DK0700290T3 (da) 2000-03-13
HU227121B1 (en) 2010-07-28
ECSP941088A (es) 1994-11-16
SI0700290T1 (en) 1999-12-31
KR100297212B1 (ko) 2001-10-24
US5741806A (en) 1998-04-21
CN1106194C (zh) 2003-04-23
NO954783L (no) 1995-11-24
JP2965703B2 (ja) 1999-10-18
NZ267415A (en) 1997-10-24
NO954783D0 (no) 1995-11-24
IL109749A0 (en) 1994-08-26
HRP940315A2 (en) 1996-08-31
HUT74867A (en) 1997-02-28
PL311721A1 (en) 1996-03-04
CA2162919A1 (en) 1994-12-08
HU9503375D0 (en) 1996-01-29
CZ291041B6 (cs) 2002-12-11
AU680918B2 (en) 1997-08-14
ZA943593B (en) 1995-02-13
HRP940315B1 (en) 2000-12-31
HRP970315A2 (en) 1999-04-30
AP544A (en) 1996-10-11
ITRM940322A0 (it) 1994-05-24
BR1100046A (pt) 1999-11-23
ITRM940322A1 (it) 1995-11-24
WO1994027599A1 (en) 1994-12-08
JPH08510457A (ja) 1996-11-05

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