OA12961A - Substituted aryl thioureas and related compounds, inhibitors of viral replication. - Google Patents
Substituted aryl thioureas and related compounds, inhibitors of viral replication. Download PDFInfo
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- OA12961A OA12961A OA1200500150A OA1200500150A OA12961A OA 12961 A OA12961 A OA 12961A OA 1200500150 A OA1200500150 A OA 1200500150A OA 1200500150 A OA1200500150 A OA 1200500150A OA 12961 A OA12961 A OA 12961A
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- OA
- OAPI
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- phenyl
- thiourea
- carbonyl
- c4alkyl
- amino
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
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- C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C335/04—Derivatives of thiourea
- C07C335/24—Derivatives of thiourea containing any of the groups, X being a hetero atom, Y being any atom
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- C07C335/04—Derivatives of thiourea
- C07C335/24—Derivatives of thiourea containing any of the groups, X being a hetero atom, Y being any atom
- C07C335/26—Y being a hydrogen or a carbon atom, e.g. benzoylthioureas
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
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- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Pyrane Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Furan Compounds (AREA)
- Pyrrole Compounds (AREA)
- Pyridine Compounds (AREA)
- Quinoline Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
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OA1200500150A OA12961A (en) | 2002-11-19 | 2003-11-18 | Substituted aryl thioureas and related compounds, inhibitors of viral replication. |
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US (2) | US7094807B2 (fr) |
EP (1) | EP1562895A1 (fr) |
JP (2) | JP4206382B2 (fr) |
KR (1) | KR20050111306A (fr) |
CN (1) | CN1738797A (fr) |
AP (1) | AP2005003319A0 (fr) |
AU (1) | AU2003295605A1 (fr) |
BR (1) | BR0316397A (fr) |
CA (1) | CA2506415A1 (fr) |
EA (1) | EA200500846A1 (fr) |
MX (1) | MXPA05005379A (fr) |
NO (1) | NO20052546L (fr) |
NZ (1) | NZ540033A (fr) |
OA (1) | OA12961A (fr) |
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US7148357B2 (en) | 2002-07-31 | 2006-12-12 | Schering Ag | VEGFR-2 and VEGFR-3 inhibitory anthranilamide pyridines |
CA2506415A1 (fr) * | 2002-11-19 | 2004-06-03 | Achillion Pharmaceuticals, Inc. | Aryl thio-urees substituees et composes analogues, inhibiteurs de la replication virale |
-
2003
- 2003-11-18 CA CA002506415A patent/CA2506415A1/fr not_active Abandoned
- 2003-11-18 WO PCT/US2003/036809 patent/WO2004046095A1/fr active Application Filing
- 2003-11-18 BR BR0316397-0A patent/BR0316397A/pt not_active IP Right Cessation
- 2003-11-18 US US10/716,175 patent/US7094807B2/en not_active Expired - Fee Related
- 2003-11-18 AU AU2003295605A patent/AU2003295605A1/en not_active Abandoned
- 2003-11-18 AP AP2005003319A patent/AP2005003319A0/xx unknown
- 2003-11-18 OA OA1200500150A patent/OA12961A/en unknown
- 2003-11-18 MX MXPA05005379A patent/MXPA05005379A/es unknown
- 2003-11-18 JP JP2004553861A patent/JP4206382B2/ja not_active Expired - Fee Related
- 2003-11-18 EP EP03786803A patent/EP1562895A1/fr not_active Withdrawn
- 2003-11-18 KR KR1020057009112A patent/KR20050111306A/ko not_active Application Discontinuation
- 2003-11-18 NZ NZ540033A patent/NZ540033A/en not_active IP Right Cessation
- 2003-11-18 CN CNA2003801087106A patent/CN1738797A/zh active Pending
- 2003-11-18 EA EA200500846A patent/EA200500846A1/ru unknown
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2004
- 2004-12-17 US US11/015,300 patent/US7476686B2/en not_active Expired - Fee Related
-
2005
- 2005-05-26 NO NO20052546A patent/NO20052546L/no not_active Application Discontinuation
-
2006
- 2006-10-03 JP JP2006272359A patent/JP2007084548A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
AP2005003319A0 (en) | 2005-06-30 |
NO20052546D0 (no) | 2005-05-26 |
MXPA05005379A (es) | 2006-02-17 |
JP2006506439A (ja) | 2006-02-23 |
AU2003295605A1 (en) | 2004-06-15 |
JP2007084548A (ja) | 2007-04-05 |
JP4206382B2 (ja) | 2009-01-07 |
EP1562895A1 (fr) | 2005-08-17 |
WO2004046095A1 (fr) | 2004-06-03 |
KR20050111306A (ko) | 2005-11-24 |
CA2506415A1 (fr) | 2004-06-03 |
US7476686B2 (en) | 2009-01-13 |
CN1738797A (zh) | 2006-02-22 |
US20060014836A1 (en) | 2006-01-19 |
EA200500846A1 (ru) | 2005-12-29 |
US7094807B2 (en) | 2006-08-22 |
BR0316397A (pt) | 2005-09-27 |
NZ540033A (en) | 2007-05-31 |
NO20052546L (no) | 2005-07-18 |
US20040138205A1 (en) | 2004-07-15 |
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