OA11069A - Intranasal formulations for treating sexual disorders - Google Patents

Intranasal formulations for treating sexual disorders Download PDF

Info

Publication number
OA11069A
OA11069A OA9900137A OA9900137A OA11069A OA 11069 A OA11069 A OA 11069A OA 9900137 A OA9900137 A OA 9900137A OA 9900137 A OA9900137 A OA 9900137A OA 11069 A OA11069 A OA 11069A
Authority
OA
OAPI
Prior art keywords
intranasal
sildenafil
formulation
mesylate
solution
Prior art date
Application number
OA9900137A
Other languages
English (en)
Inventor
Ann Billotte
Peter James Dunn
Brian Thomas Henry
Peter Vallance Marshall
Joanna Jayne Woods
Original Assignee
Pfizer Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9813452.1A external-priority patent/GB9813452D0/en
Priority claimed from GBGB9820837.4A external-priority patent/GB9820837D0/en
Priority claimed from GBGB9903177.5A external-priority patent/GB9903177D0/en
Application filed by Pfizer Res & Dev filed Critical Pfizer Res & Dev
Publication of OA11069A publication Critical patent/OA11069A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Otolaryngology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
OA9900137A 1998-06-22 1999-06-18 Intranasal formulations for treating sexual disorders OA11069A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9813452.1A GB9813452D0 (en) 1998-06-22 1998-06-22 Pharmaceutical formulations
GBGB9820837.4A GB9820837D0 (en) 1998-09-24 1998-09-24 Pharmaceutical formulations
GBGB9903177.5A GB9903177D0 (en) 1999-02-13 1999-02-13 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
OA11069A true OA11069A (en) 2002-03-13

Family

ID=27269368

Family Applications (1)

Application Number Title Priority Date Filing Date
OA9900137A OA11069A (en) 1998-06-22 1999-06-18 Intranasal formulations for treating sexual disorders

Country Status (40)

Country Link
US (2) US20020040139A1 (bg)
EP (1) EP0967214B1 (bg)
JP (1) JP3263379B2 (bg)
KR (1) KR100345824B1 (bg)
AP (1) AP1178A (bg)
AR (1) AR016993A1 (bg)
AT (1) ATE269866T1 (bg)
AU (1) AU746865B2 (bg)
BG (1) BG64372B1 (bg)
BR (1) BR9903273A (bg)
CA (1) CA2275554C (bg)
CZ (1) CZ294856B6 (bg)
DE (1) DE69918222T2 (bg)
DK (1) DK0967214T3 (bg)
DZ (1) DZ2826A1 (bg)
EA (1) EA001903B1 (bg)
ES (1) ES2221733T3 (bg)
GT (1) GT199900095A (bg)
HN (1) HN1999000096A (bg)
HR (1) HRP990195B1 (bg)
HU (1) HUP9902076A3 (bg)
ID (1) ID23554A (bg)
IL (1) IL130539A0 (bg)
IS (1) IS5085A (bg)
MA (1) MA25089A1 (bg)
MY (1) MY117967A (bg)
NO (1) NO317365B1 (bg)
NZ (1) NZ336382A (bg)
OA (1) OA11069A (bg)
PA (1) PA8476301A1 (bg)
PE (1) PE20000702A1 (bg)
PT (1) PT967214E (bg)
SG (1) SG77246A1 (bg)
SI (1) SI0967214T1 (bg)
SK (1) SK284574B6 (bg)
TN (1) TNSN99129A1 (bg)
TR (1) TR199901444A2 (bg)
TW (1) TWI223598B (bg)
UA (1) UA59385C2 (bg)
YU (1) YU29699A (bg)

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Also Published As

Publication number Publication date
DE69918222D1 (de) 2004-07-29
PE20000702A1 (es) 2000-08-16
DE69918222T2 (de) 2005-07-28
PT967214E (pt) 2004-08-31
BR9903273A (pt) 2000-05-09
HUP9902076A3 (en) 2002-03-28
BG64372B1 (bg) 2004-12-30
AU3579499A (en) 2000-01-06
ES2221733T3 (es) 2005-01-01
JP2000034232A (ja) 2000-02-02
HU9902076D0 (en) 1999-08-30
EP0967214B1 (en) 2004-06-23
HN1999000096A (es) 2000-12-03
IL130539A0 (en) 2000-06-01
NZ336382A (en) 1999-11-29
SG77246A1 (en) 2000-12-19
SK284574B6 (sk) 2005-06-02
SK81999A3 (en) 2001-01-18
ID23554A (id) 2000-05-04
EA199900487A3 (ru) 2000-04-24
PA8476301A1 (es) 2000-09-29
HUP9902076A2 (hu) 2000-05-28
ATE269866T1 (de) 2004-07-15
EA199900487A2 (ru) 1999-12-29
JP3263379B2 (ja) 2002-03-04
SI0967214T1 (en) 2004-10-31
MY117967A (en) 2004-08-30
DK0967214T3 (da) 2004-09-27
HRP990195B1 (en) 2003-04-30
CA2275554A1 (en) 1999-12-22
TWI223598B (en) 2004-11-11
IS5085A (is) 1999-12-23
EA001903B1 (ru) 2001-10-22
AP9901585A0 (en) 1999-06-30
CZ294856B6 (cs) 2005-03-16
NO993051D0 (no) 1999-06-21
KR100345824B1 (ko) 2002-07-24
BG103510A (bg) 2000-01-31
GT199900095A (es) 2000-12-13
AP1178A (en) 2003-06-30
CZ9902257A3 (cs) 2000-11-15
NO317365B1 (no) 2004-10-18
US20030158206A1 (en) 2003-08-21
DZ2826A1 (fr) 2003-12-01
UA59385C2 (uk) 2003-09-15
CA2275554C (en) 2003-06-03
HRP990195A2 (en) 2000-02-29
MA25089A1 (fr) 2000-12-31
AR016993A1 (es) 2001-08-01
EP0967214A1 (en) 1999-12-29
AU746865B2 (en) 2002-05-02
KR20000006310A (ko) 2000-01-25
YU29699A (sh) 2003-02-28
US20020040139A1 (en) 2002-04-04
NO993051L (no) 1999-12-23
TR199901444A2 (xx) 2000-01-21
TNSN99129A1 (fr) 2005-11-10

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