OA10189A - Use of indole derivatives as 5htl agonists - Google Patents

Use of indole derivatives as 5htl agonists Download PDF

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Publication number
OA10189A
OA10189A OA60728A OA60728A OA10189A OA 10189 A OA10189 A OA 10189A OA 60728 A OA60728 A OA 60728A OA 60728 A OA60728 A OA 60728A OA 10189 A OA10189 A OA 10189A
Authority
OA
OAPI
Prior art keywords
indole
ylmethyl
methylaminosulfonylmethyl
treating
ranging
Prior art date
Application number
OA60728A
Other languages
English (en)
Inventor
John Eugene Macor
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of OA10189A publication Critical patent/OA10189A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
OA60728A 1993-04-27 1995-10-27 Use of indole derivatives as 5htl agonists OA10189A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5393093A 1993-04-27 1993-04-27

Publications (1)

Publication Number Publication Date
OA10189A true OA10189A (en) 1996-12-18

Family

ID=21987528

Family Applications (1)

Application Number Title Priority Date Filing Date
OA60728A OA10189A (en) 1993-04-27 1995-10-27 Use of indole derivatives as 5htl agonists

Country Status (29)

Country Link
EP (1) EP0696194B1 (es)
JP (1) JP2922307B2 (es)
KR (1) KR960701636A (es)
CN (3) CN1121689A (es)
AP (1) AP486A (es)
AT (1) ATE222492T1 (es)
AU (1) AU689469B2 (es)
BG (1) BG61898B1 (es)
BR (1) BR9406435A (es)
CA (1) CA2161533C (es)
CO (1) CO4230093A1 (es)
CZ (1) CZ290416B6 (es)
DE (1) DE69431201T2 (es)
DK (1) DK0696194T3 (es)
ES (1) ES2180573T3 (es)
HU (1) HU222488B1 (es)
IL (1) IL109376A (es)
MX (1) MX9403088A (es)
NO (1) NO308236B1 (es)
NZ (1) NZ263614A (es)
OA (1) OA10189A (es)
PL (1) PL175156B1 (es)
PT (1) PT696194E (es)
RO (1) RO117760B1 (es)
RU (1) RU2132683C1 (es)
SG (1) SG43951A1 (es)
SK (1) SK283353B6 (es)
WO (1) WO1994025023A1 (es)
ZA (1) ZA942805B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5559129A (en) * 1990-10-15 1996-09-24 Pfizer Inc Indole derivatives
US5545644A (en) * 1990-10-15 1996-08-13 Pfizer Inc. Indole derivatives
US5559246A (en) * 1990-10-15 1996-09-24 Pfizer Inc. Indole derivatives
US5578612A (en) * 1990-10-15 1996-11-26 Pfizer Inc. Indole derivatives
US5607951A (en) * 1990-10-15 1997-03-04 Pfizer Inc Indole derivatives
KR100191973B1 (ko) * 1993-08-31 1999-06-15 디. 제이. 우드, 스피겔 알렌 제이 5-아릴인돌 유도체
GB9417310D0 (en) 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
WO1996011923A1 (en) * 1994-10-12 1996-04-25 Pfizer Limited Indole derivative for the treatment of migraine
GB9424471D0 (en) * 1994-12-03 1995-01-18 Pfizer Ltd Treatment of emesis
GB9510223D0 (en) * 1995-05-20 1995-07-19 Pfizer Ltd Therapeutic agent
US5945118A (en) * 1995-09-29 1999-08-31 Pfizer Inc Indole derivative for the treatment of migraine
US5773015A (en) * 1996-11-27 1998-06-30 Elizabeth Arden Co., Division Of Conopco, Inc. Method for controlling skin oils and grease
GB9706089D0 (en) * 1997-03-24 1997-05-14 Scherer Ltd R P Pharmaceutical composition
US5994352A (en) * 1998-11-13 1999-11-30 Pfizer Inc. 5-arylindole derivatives
ES2199086B1 (es) * 2002-07-31 2005-06-01 Cepa Schwarz Pharma Sl Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
MX2022009528A (es) * 2020-02-04 2022-11-14 Mindset Pharma Inc Derivados de 3-pirrolidina-indol como agentes psicodélicos serotoninérgicos para el tratamiento de trastornos del snc.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2095360C1 (ru) * 1990-10-15 1997-11-10 Пфайзер Инк. Производные индола, их оптические изомеры и фармацевтически приемлемые соли
GB9102579D0 (en) * 1991-01-24 1991-03-27 Glaxo Group Ltd Compositions
GB9103770D0 (en) * 1991-02-22 1991-04-10 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
PL311266A1 (en) 1996-02-05
EP0696194A1 (en) 1996-02-14
CZ290416B6 (cs) 2002-07-17
CN1121689A (zh) 1996-05-01
ATE222492T1 (de) 2002-09-15
AU6436094A (en) 1994-11-21
HU222488B1 (hu) 2003-07-28
KR960701636A (ko) 1996-03-28
PT696194E (pt) 2002-11-29
CA2161533A1 (en) 1994-11-10
BR9406435A (pt) 1996-01-09
JPH08504829A (ja) 1996-05-28
EP0696194B1 (en) 2002-08-21
NZ263614A (en) 1998-02-26
ZA942805B (en) 1995-10-23
CN1509713A (zh) 2004-07-07
DE69431201T2 (de) 2002-12-05
AP9400633A0 (en) 1994-04-30
AP486A (en) 1996-04-16
CN1515252A (zh) 2004-07-28
BG100093A (bg) 1996-04-30
HU9503089D0 (en) 1995-12-28
HUT73670A (en) 1996-09-30
SK133295A3 (en) 1997-01-08
RO117760B1 (ro) 2002-07-30
CZ9502802A3 (en) 1996-04-17
IL109376A (en) 2000-10-31
SK283353B6 (sk) 2003-06-03
NO954287L (no) 1995-10-26
IL109376A0 (en) 1994-07-31
PL175156B1 (pl) 1998-11-30
DK0696194T3 (da) 2002-10-07
SG43951A1 (en) 1997-11-14
AU689469B2 (en) 1998-04-02
MX9403088A (es) 1997-02-28
BG61898B1 (bg) 1998-09-30
CA2161533C (en) 1998-08-04
CO4230093A1 (es) 1995-10-19
JP2922307B2 (ja) 1999-07-19
NO308236B1 (no) 2000-08-21
RU2132683C1 (ru) 1999-07-10
NO954287D0 (no) 1995-10-26
WO1994025023A1 (en) 1994-11-10
DE69431201D1 (de) 2002-09-26
ES2180573T3 (es) 2003-02-16

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