OA09835A - Nouveaux dérivés p-substitués de phnényl 4-oxybutane amine leurs procédés de préparation et les compositions pharmaceutiques n renfermant - Google Patents

Nouveaux dérivés p-substitués de phnényl 4-oxybutane amine leurs procédés de préparation et les compositions pharmaceutiques n renfermant

Info

Publication number
OA09835A
OA09835A OA60229A OA60229A OA09835A OA 09835 A OA09835 A OA 09835A OA 60229 A OA60229 A OA 60229A OA 60229 A OA60229 A OA 60229A OA 09835 A OA09835 A OA 09835A
Authority
OA
OAPI
Prior art keywords
phnenyl
oxybutane
amine
new
pharmaceutical compositions
Prior art date
Application number
OA60229A
Other languages
English (en)
Inventor
Paule Bonnet
Remi Delansorne
Maurice Faure
Michel Lanquetin
Serge Zunino
Original Assignee
Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theramex filed Critical Theramex
Publication of OA09835A publication Critical patent/OA09835A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline
OA60229A 1990-10-17 1992-06-17 Nouveaux dérivés p-substitués de phnényl 4-oxybutane amine leurs procédés de préparation et les compositions pharmaceutiques n renfermant OA09835A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR909012562A FR2668150B1 (fr) 1990-10-17 1990-10-17 Nouveaux derives du terbutylphenyl 1-amino 4-hydroxybutane, leurs procedes de preparation et les compositions pharmaceutiques en renfermant.

Publications (1)

Publication Number Publication Date
OA09835A true OA09835A (fr) 1994-08-15

Family

ID=9401134

Family Applications (1)

Application Number Title Priority Date Filing Date
OA60229A OA09835A (fr) 1990-10-17 1992-06-17 Nouveaux dérivés p-substitués de phnényl 4-oxybutane amine leurs procédés de préparation et les compositions pharmaceutiques n renfermant

Country Status (23)

Country Link
US (1) US5461059A (fr)
EP (1) EP0505543A1 (fr)
JP (1) JPH05503298A (fr)
KR (1) KR927003589A (fr)
AP (1) AP282A (fr)
BG (1) BG60680B1 (fr)
BR (1) BR9106188A (fr)
CA (1) CA2071911A1 (fr)
CZ (1) CZ182292A3 (fr)
FI (1) FI922773A (fr)
FR (2) FR2668150B1 (fr)
HU (1) HUT61297A (fr)
IE (1) IE913636A1 (fr)
IL (1) IL99776A0 (fr)
MA (1) MA22321A1 (fr)
NO (1) NO922358L (fr)
NZ (1) NZ240274A (fr)
OA (1) OA09835A (fr)
PL (2) PL169022B1 (fr)
PT (1) PT99266A (fr)
RO (1) RO108241B1 (fr)
WO (1) WO1992006977A1 (fr)
ZA (1) ZA918282B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2048109B1 (es) * 1992-07-20 1994-12-16 Espanola Prod Quimicos Procedimiento de preparacion de nuevos derivados piperidicos del bencimidazol.
WO1994027973A1 (fr) * 1993-05-20 1994-12-08 Kissei Pharmaceutical Co., Ltd. Derive 1-(2-benzimidazolyl)-1,5-diazacyclooctane
ES2072193B1 (es) * 1993-05-21 1996-02-16 Espanola Prod Quimicos Nuevos derivados del1-fenilmetil bencimidazol piperacinas.
US5691323A (en) * 1995-05-12 1997-11-25 Merck & Co., Inc. Muscarine antagonists
FR2727865B1 (fr) * 1994-12-08 1997-07-18 Esteve Labor Dr Utilisation des derives de 2-(4-(azolybutyl)-piperazinyl- (methyl))-benzimidazole et analogues ainsi que de leurs sels, pour la preparation de medicaments destines au traitement ou a la prophylaxie de l'asthme
AU707139B2 (en) * 1996-04-03 1999-07-01 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
HUP0301622A3 (en) * 2000-07-04 2006-05-29 Novo Nordisk As Purine derivatives inhibiting the enzyme dipeptidyl petidase iv (dpp-iv) and pharmaceutical compositions containing them
WO2004009091A1 (fr) * 2002-06-17 2004-01-29 Glaxo Group Limited Agonistes des recepteurs x du foie

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL137020C (fr) * 1962-08-31
US3161645A (en) * 1962-12-18 1964-12-15 Res Lab Dr C Janssen N V 1-(1-aroylpropyl-4-piperidyl)-2-benzimidazolinones and related compounds
US3491103A (en) * 1963-12-19 1970-01-20 Sandoz Ag Certain 4h-benzo(4,5)cyclohepta-(1,2-b) thiophenes
US4219559A (en) * 1979-01-10 1980-08-26 Janssen Pharmaceutica N.V. N-Heterocyclyl-4-piperidinamines
JPS5879983A (ja) * 1981-11-06 1983-05-13 Kanebo Ltd 新規なベンズイミダゾ−ル誘導体、その製造法およびその医薬組成物
US4695575A (en) * 1984-11-13 1987-09-22 Janssen Pharmaceutica, N.V. 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines
NZ223654A (en) * 1987-03-09 1990-03-27 Janssen Pharmaceutica Nv 1-alkyl-substituted-benzimidazole-4-piperidinamines and pharmaceutical compositions
EP0339978B1 (fr) * 1988-04-28 1996-08-21 Schering Corporation Composés polycycliques condensés, compositions, procédés de préparation et leur utilisation comme agents PAF antagonistiques, antihistaminiques et/ou anti-inflammatoires
US4908372A (en) * 1988-10-13 1990-03-13 Merrell Dow Pharmaceuticals Inc. Antihistaminic piperidinyl benzimidazoles
PH30434A (en) * 1989-04-07 1997-05-09 Janssen Pharmaceutica Nv Hydroxyalkylfuranyl derivatives
US5217980A (en) * 1990-07-19 1993-06-08 Janssen Pharmaceutica N.V. Oxazolyl and piperidinyl substituted benimidazolyl compounds

Also Published As

Publication number Publication date
WO1992006977A1 (fr) 1992-04-30
HU9202176D0 (en) 1992-10-28
FI922773A0 (fi) 1992-06-16
FR2670783B1 (fr) 1994-11-18
CA2071911A1 (fr) 1992-04-18
NO922358L (no) 1992-08-11
BR9106188A (pt) 1993-03-16
CZ182292A3 (en) 1993-01-13
KR927003589A (ko) 1992-12-18
AP282A (en) 1993-09-08
RO108241B1 (ro) 1994-03-31
JPH05503298A (ja) 1993-06-03
PL169022B1 (pl) 1996-05-31
FR2668150A1 (fr) 1992-04-24
NZ240274A (en) 1995-07-26
NO922358D0 (no) 1992-06-16
PT99266A (pt) 1992-08-31
IL99776A0 (en) 1992-08-18
MA22321A1 (fr) 1992-07-01
BG60680B1 (bg) 1995-12-29
IE913636A1 (en) 1992-04-22
ZA918282B (en) 1992-07-29
EP0505543A1 (fr) 1992-09-30
PL169452B1 (pl) 1996-07-31
AP9100328A0 (en) 1991-10-31
FR2670783A1 (fr) 1992-06-26
FI922773A (fi) 1992-06-16
HUT61297A (en) 1992-12-28
US5461059A (en) 1995-10-24
FR2668150B1 (fr) 1994-11-18

Similar Documents

Publication Publication Date Title
FR2569404B1 (fr) Nouveaux derives de 1,2-benzisothiazol-3-ylpiperazine, compositions pharmaceutiques contenant de tels composes et leurs procedes de preparation
MA23632A1 (fr) Procede de preparation de composes nouveaux et de compostions pharmaceutiques les contenant
DE69131813D1 (de) Amido-3-Pyrazol-Derivate, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen
OA09378A (fr) "Nouveaux dérivés de la pipéridine, de la tétrahydropyridine et de la pyrrolidine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent".
FR2466248B1 (fr) Derives d'agents anti-inflammatoires non steroides, procede de preparation et compositions pharmaceutiques les contenant
PT84171A (pt) Procede de preparation de derives des n alpha-arylsulfonylaminoacyl-p-amidinophenylalaninamides leurs derives de synthese et leurs compositions pharmaceutiques les contenant
FR2694004B1 (fr) Nouvelles 3-(Hydroxybenzylidényl)-indoline-2-ones et 3-(hydroxybenzylidényl)-indoline-2-thiones, leurs procédés de préparation, et les compositions pharmaceutiques qui les contiennent.
FR2703051B1 (fr) Nouvelles pyridothiadiazines, leurs procédés de préparation, et les compositions pharmaceutiques qui les contiennent.
FR2714907B1 (fr) Nouveaux dérivés de l'Adénosine, leurs procédés de préparation, compositions pharmaceutiques les contenant.
PT72631B (fr) Procede pour la preparation de nouveaux derives de guanidine et de compositions pharmaceutiques qui les contiennent
BE887970A (fr) Nouveaux derives d'ocytocine et compositions pharmaceutiques contenant ces derives
DZ2550A1 (fr) Dérivés d'azétidinylpropylpipéridine procédé pour leur préparation et compositions pharmaceutiques les contenant.
DE19975037I2 (de) 3H-Imidazo-5,1-d-1,2,3,5-tetrazin-4-on-Derivate Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammensetzungen
FR2714059B1 (fr) Dérivés amino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
OA09835A (fr) Nouveaux dérivés p-substitués de phnényl 4-oxybutane amine leurs procédés de préparation et les compositions pharmaceutiques n renfermant
OA09137A (fr) Nouveaux dérivés de la benzoxazolinone, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
FR2740134B1 (fr) Derives d'amines cycliques d'aryl-piperazines, leur preparation et les compositions pharmaceutiques les contenant
PT84452A (fr) Procede de preparation de derives de n-](hydroxy-2 phenyl) (phenyl) methylene"amino-2 ethyl"acetamide et de compositions pharmaceutiques les contenant
PT87699A (pt) Process for the preparation of tricyclic pyridone derivatives and of pharmaceutical compositions containing the same
FR2686339B1 (fr) Nouveaux amides et sulfonamides naphtaleniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
PT83593A (fr) Procede de preparation de 7-acyl-benzoxazinones et leurs derives et de compositions pharmaceutiques les contenant
OA09439A (fr) "Nouveaux dérivés benzoxazolinoniques, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent".
FR2689509B1 (fr) Nouveaux derives spiraniques du 3-amino chromane, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
PT84933B (fr) Procede de preparation de cyclodepsipeptides et compositions pharmaceutiques qui les contiennent
PT87202A (pt) Process for the preparation of novel acyl derivatives and of pharmaceutical compositions containing the same