OA07178A - Nouveaux dérivés de la méthyl-4 phényl-6 pyridazine actifs sur le système nerveux central. - Google Patents

Nouveaux dérivés de la méthyl-4 phényl-6 pyridazine actifs sur le système nerveux central.

Info

Publication number
OA07178A
OA07178A OA57770A OA57770A OA07178A OA 07178 A OA07178 A OA 07178A OA 57770 A OA57770 A OA 57770A OA 57770 A OA57770 A OA 57770A OA 07178 A OA07178 A OA 07178A
Authority
OA
OAPI
Prior art keywords
methyl
pyridazine
phenyl
active
nervous system
Prior art date
Application number
OA57770A
Other languages
English (en)
French (fr)
Inventor
Camille Wermuth
Kathleen Biziere
Horace Davi
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of OA07178A publication Critical patent/OA07178A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/22Nitrogen and oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20Nitrogen atoms
OA57770A 1981-08-10 1982-08-10 Nouveaux dérivés de la méthyl-4 phényl-6 pyridazine actifs sur le système nerveux central. OA07178A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8115435A FR2510997A1 (fr) 1981-08-10 1981-08-10 Nouveaux derives de la methyl-4 phenyl-6 pyridazine, procede pour leur preparation et medicaments actifs sur le systeme nerveux central en contenant

Publications (1)

Publication Number Publication Date
OA07178A true OA07178A (fr) 1984-04-30

Family

ID=9261319

Family Applications (1)

Application Number Title Priority Date Filing Date
OA57770A OA07178A (fr) 1981-08-10 1982-08-10 Nouveaux dérivés de la méthyl-4 phényl-6 pyridazine actifs sur le système nerveux central.

Country Status (29)

Country Link
US (3) US4576946A (ja)
EP (1) EP0072299B1 (ja)
JP (1) JPS5838262A (ja)
KR (1) KR880002710B1 (ja)
AT (1) ATE24317T1 (ja)
AU (1) AU548029B2 (ja)
CA (1) CA1180704A (ja)
CS (1) CS241052B2 (ja)
DD (3) DD209453A5 (ja)
DE (1) DE3274737D1 (ja)
DK (1) DK148654C (ja)
EG (1) EG15922A (ja)
ES (1) ES514854A0 (ja)
FI (1) FI74462C (ja)
FR (1) FR2510997A1 (ja)
GR (1) GR76235B (ja)
HU (1) HU190695B (ja)
IE (1) IE53611B1 (ja)
IL (1) IL66423A0 (ja)
MA (1) MA19561A1 (ja)
NO (1) NO157141C (ja)
NZ (1) NZ201530A (ja)
OA (1) OA07178A (ja)
PH (1) PH17883A (ja)
PL (3) PL137201B1 (ja)
PT (1) PT75371B (ja)
SU (2) SU1366056A3 (ja)
YU (3) YU171782A (ja)
ZA (1) ZA825516B (ja)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2539741A1 (fr) * 1983-01-21 1984-07-27 Sanofi Sa Composes a noyau heterocyclique diazote, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent
FR2540113A1 (fr) * 1983-01-27 1984-08-03 Sanofi Sa Acides derives de la pyridazine actifs sur le systeme nerveux central
US4565814A (en) * 1983-01-28 1986-01-21 Sanofi Pyridazine derivatives having a psychotropic action and compositions
FR2601011B1 (fr) * 1986-07-03 1988-10-28 Sanofi Sa Nouveaux derives tricycliques agonistes des recepteurs cholinergiques et medicaments en contenant
US5106973A (en) * 1987-11-23 1992-04-21 Janssen Pharmaceutica N.V. Pyridzainamine derivatives
PT93060B (pt) 1989-02-07 1995-12-29 Sanofi Sa Processo para a obtencao de derivados de piridazina e de composicoes farmaceuticas que os contem
FR2642648B1 (fr) * 1989-02-07 1991-06-21 Sanofi Sa Utilisation de derives d'alkyl-5 pyridazine comme medicaments actifs sur le systeme cholinergique
US5631255A (en) * 1989-02-07 1997-05-20 Sanofi Pyridazine derivatives
JP3553142B2 (ja) * 1994-07-29 2004-08-11 花王株式会社 4級アンモニウム塩の製造方法及び中間体ジアミノアルコール
EP1745039A4 (en) * 2004-05-08 2009-07-22 Neurogen Corp 3-ARYL-5,6-DISUBSTITUTED PYRIDAZINES
EP1741709A1 (en) * 2005-06-28 2007-01-10 Sanofi-Aventis Deutschland GmbH Heteroaryl-substituted amides comprising a saturated linker group, and their use as pharmaceuticals
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
AR081626A1 (es) 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
MA41598A (fr) * 2015-02-25 2018-01-02 Constellation Pharmaceuticals Inc Composés thérapeutiques de pyridazine et leurs utilisations
AR119731A1 (es) 2019-05-17 2022-01-05 Novartis Ag Inhibidores del inflamasoma nlrp3

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1345880A (en) * 1971-06-18 1974-02-06 Cepbepe Pyridazine derivatives
FR2388799A1 (fr) * 1977-04-28 1978-11-24 Rolland Sa A Derives de pyridazinone, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
IL66423A0 (en) 1982-11-30
FI74462B (fi) 1987-10-30
IE53611B1 (en) 1988-12-21
PL237837A1 (en) 1984-05-07
AU548029B2 (en) 1985-11-21
JPH0417950B2 (ja) 1992-03-26
NZ201530A (en) 1985-05-31
AU8661982A (en) 1983-02-17
NO822705L (no) 1983-02-11
DK357482A (da) 1983-02-11
ES8305735A1 (es) 1983-05-01
FI822767A0 (fi) 1982-08-09
PL137262B1 (en) 1986-05-31
SU1366056A3 (ru) 1988-01-07
PL243376A1 (en) 1984-04-24
NO157141B (no) 1987-10-19
PL137265B1 (en) 1986-05-31
JPS5838262A (ja) 1983-03-05
US4514397A (en) 1985-04-30
EP0072299B1 (fr) 1986-12-17
PL137201B1 (en) 1986-05-31
MA19561A1 (fr) 1983-04-01
NO157141C (no) 1988-01-27
YU209684A (en) 1985-04-30
EG15922A (en) 1986-06-30
EP0072299A3 (en) 1984-01-11
DK148654C (da) 1986-02-17
GR76235B (ja) 1984-08-04
DD209453A5 (de) 1984-05-09
PT75371B (en) 1984-12-10
EP0072299A2 (fr) 1983-02-16
ES514854A0 (es) 1983-05-01
KR840001146A (ko) 1984-03-28
FR2510997A1 (fr) 1983-02-11
FI822767L (fi) 1983-02-11
SU1356961A3 (ru) 1987-11-30
FR2510997B1 (ja) 1984-02-10
US4677106A (en) 1987-06-30
PL243377A1 (en) 1984-04-24
US4576946A (en) 1986-03-18
CA1180704A (en) 1985-01-08
YU171782A (en) 1985-04-30
DK148654B (da) 1985-08-26
PH17883A (en) 1985-01-21
IE821821L (en) 1983-02-10
ATE24317T1 (de) 1987-01-15
ZA825516B (en) 1983-06-29
HU190695B (en) 1986-10-28
DD213213A5 (de) 1984-09-05
DD213212A5 (de) 1984-09-05
CS241052B2 (en) 1986-03-13
YU209784A (en) 1985-04-30
DE3274737D1 (en) 1987-01-29
PT75371A (en) 1982-09-01
FI74462C (fi) 1988-02-08
CS591282A2 (en) 1985-06-13
KR880002710B1 (ko) 1988-12-26

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