OA06889A - Nouveaux dérivés du 4H-1,2,4-triazole, leur préparation, leur application comme médicament, les compositions les renfermant et les intermédiaires obtenus. - Google Patents

Nouveaux dérivés du 4H-1,2,4-triazole, leur préparation, leur application comme médicament, les compositions les renfermant et les intermédiaires obtenus.

Info

Publication number
OA06889A
OA06889A OA57482A OA57482A OA06889A OA 06889 A OA06889 A OA 06889A OA 57482 A OA57482 A OA 57482A OA 57482 A OA57482 A OA 57482A OA 06889 A OA06889 A OA 06889A
Authority
OA
OAPI
Prior art keywords
triazole
medicament
preparation
application
compositions containing
Prior art date
Application number
OA57482A
Other languages
English (en)
French (fr)
Inventor
Jean Meier
Francois Clemence
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of OA06889A publication Critical patent/OA06889A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C243/24Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids
    • C07C243/38Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
OA57482A 1980-08-22 1981-08-22 Nouveaux dérivés du 4H-1,2,4-triazole, leur préparation, leur application comme médicament, les compositions les renfermant et les intermédiaires obtenus. OA06889A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8018354A FR2488891A1 (fr) 1980-08-22 1980-08-22 Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament

Publications (1)

Publication Number Publication Date
OA06889A true OA06889A (fr) 1983-04-30

Family

ID=9245357

Family Applications (2)

Application Number Title Priority Date Filing Date
OA57482A OA06889A (fr) 1980-08-22 1981-08-22 Nouveaux dérivés du 4H-1,2,4-triazole, leur préparation, leur application comme médicament, les compositions les renfermant et les intermédiaires obtenus.
OA58106A OA07537A (fr) 1980-08-22 1983-09-22 Nouveaux dérivés du 4 H-1,2,4-triazole, leur préparation, leur application comme médicamment, les compositions les renfermant et les intermediaires obtenus.

Family Applications After (1)

Application Number Title Priority Date Filing Date
OA58106A OA07537A (fr) 1980-08-22 1983-09-22 Nouveaux dérivés du 4 H-1,2,4-triazole, leur préparation, leur application comme médicamment, les compositions les renfermant et les intermediaires obtenus.

Country Status (24)

Country Link
US (3) US4512997A (xx)
JP (1) JPS5770875A (xx)
AT (1) AT378957B (xx)
AU (1) AU543946B2 (xx)
BE (1) BE890035A (xx)
CA (1) CA1208226A (xx)
CH (1) CH649994A5 (xx)
DE (1) DE3133185A1 (xx)
DK (1) DK370781A (xx)
ES (2) ES504887A0 (xx)
FI (1) FI72971C (xx)
FR (1) FR2488891A1 (xx)
GB (1) GB2082581B (xx)
GR (1) GR75329B (xx)
HU (1) HU185647B (xx)
IE (1) IE51510B1 (xx)
IT (1) IT1171477B (xx)
LU (1) LU83576A1 (xx)
NL (1) NL8103903A (xx)
OA (2) OA06889A (xx)
PH (2) PH19890A (xx)
PT (1) PT73544B (xx)
SE (1) SE454173B (xx)
ZA (1) ZA815689B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2488891A1 (fr) * 1980-08-22 1982-02-26 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament
FR2539127B1 (fr) * 1983-01-10 1985-08-23 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicaments
US5278180A (en) * 1984-09-24 1994-01-11 Roussel Uclaf 4,5-bis(aryl) 4H-1,2,4-triazoles derivatives and analgesic use
FR2570699B1 (fr) * 1984-09-24 1987-08-28 Roussel Uclaf Nouveau procede de preparation de derives du 4h-1,2,4-triazole, nouveaux triazoles ainsi obtenus, leur application comme medicaments et les compositions pharmaceutiques les renfermant
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US6362342B1 (en) * 1999-06-29 2002-03-26 Lion Bioscience Ag Triazole compounds and methods of making same
US6770621B2 (en) 2000-05-02 2004-08-03 Theravance, Inc. Polyacid glycopeptide derivatives
JP2005521676A (ja) * 2002-02-07 2005-07-21 ザ キュレイターズ オブ ザ ユニバーシティ オブ ミズーリ オピオイドレセプター作動性4−(3−ヒドロキシフェニル)または4−(3−アルコキシフェニル)−1,2,4−トリアゾール化合物
KR102563713B1 (ko) 2017-04-26 2023-08-07 오티아이 루미오닉스 인크. 표면의 코팅을 패턴화하는 방법 및 패턴화된 코팅을 포함하는 장치
US11751415B2 (en) 2018-02-02 2023-09-05 Oti Lumionics Inc. Materials for forming a nucleation-inhibiting coating and devices incorporating same
KR20210149058A (ko) 2019-03-07 2021-12-08 오티아이 루미오닉스 인크. 핵생성 억제 코팅물 형성용 재료 및 이를 포함하는 디바이스
CN114072705A (zh) 2019-05-08 2022-02-18 Oti照明公司 用于形成成核抑制涂层的材料和结合所述成核抑制涂层的装置

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1796403A (en) * 1931-03-17 Schaft
US3681374A (en) * 1970-08-11 1972-08-01 Asahi Chemical Ind Synthetic nacreous triazole crystals and method for production thereof
SU508198A3 (ru) * 1971-07-22 1976-03-25 Группо Лепетит С.П.А. (Фирма) Способ получени производных 1,2,4-триазола
AU7528974A (en) * 1973-11-13 1976-06-10 Commonwealth Scientific And Industrial Research Organization Triazoles
FR2269938A2 (en) * 1974-05-08 1975-12-05 Delalande Sa 5-Hydroxymethyl-3,4-diphenyl-1,2,4-triazoles - with anticholinergic, bronchodilator, antidepressant, analgesic, vasodilator activity, etc.
JPS56125376A (en) * 1980-03-07 1981-10-01 Mitsubishi Chem Ind Ltd Triazole derivative
FR2488891A1 (fr) * 1980-08-22 1982-02-26 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament

Also Published As

Publication number Publication date
CA1208226A (fr) 1986-07-22
SE8104515L (sv) 1982-02-23
IE51510B1 (en) 1987-01-07
ES8306730A1 (es) 1983-06-01
ES8307227A1 (es) 1983-06-16
ES515419A0 (es) 1983-06-16
US4512997A (en) 1985-04-23
AU543946B2 (en) 1985-05-09
LU83576A1 (fr) 1982-04-14
PT73544A (fr) 1981-09-01
NL8103903A (nl) 1982-03-16
FR2488891A1 (fr) 1982-02-26
FI72971B (fi) 1987-04-30
GB2082581A (en) 1982-03-10
JPH0261463B2 (xx) 1990-12-20
FI72971C (fi) 1987-08-10
IT1171477B (it) 1987-06-10
HU185647B (en) 1985-03-28
BE890035A (fr) 1982-02-22
ATA368281A (de) 1985-03-15
PT73544B (fr) 1983-07-14
PH19890A (en) 1986-08-13
GB2082581B (en) 1985-02-13
AT378957B (de) 1985-10-25
AU7442681A (en) 1982-02-25
DE3133185A1 (de) 1982-04-08
ZA815689B (en) 1982-08-25
FI812585L (fi) 1982-02-23
IE811923L (en) 1982-02-22
US4727084A (en) 1988-02-23
SE454173B (sv) 1988-04-11
DK370781A (da) 1982-02-23
IT8149147A0 (it) 1981-08-21
GR75329B (xx) 1984-07-13
OA07537A (fr) 1985-03-31
PH21567A (en) 1987-12-11
US4659729A (en) 1987-04-21
FR2488891B1 (xx) 1983-06-17
JPS5770875A (en) 1982-05-01
ES504887A0 (es) 1983-06-01
CH649994A5 (fr) 1985-06-28

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