BE890035A - Nouveaux derives du 4h-1,2,4-triazole, leur preparation, leur application comme medicament, les compositions les renfermant et les intermediaires obtenus - Google Patents

Nouveaux derives du 4h-1,2,4-triazole, leur preparation, leur application comme medicament, les compositions les renfermant et les intermediaires obtenus

Info

Publication number
BE890035A
BE890035A BE0/205731A BE205731A BE890035A BE 890035 A BE890035 A BE 890035A BE 0/205731 A BE0/205731 A BE 0/205731A BE 205731 A BE205731 A BE 205731A BE 890035 A BE890035 A BE 890035A
Authority
BE
Belgium
Prior art keywords
medicaments
preparation
new
application
compositions containing
Prior art date
Application number
BE0/205731A
Other languages
English (en)
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of BE890035A publication Critical patent/BE890035A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C243/24Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids
    • C07C243/38Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BE0/205731A 1980-08-22 1981-08-21 Nouveaux derives du 4h-1,2,4-triazole, leur preparation, leur application comme medicament, les compositions les renfermant et les intermediaires obtenus BE890035A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8018354A FR2488891A1 (fr) 1980-08-22 1980-08-22 Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament

Publications (1)

Publication Number Publication Date
BE890035A true BE890035A (fr) 1982-02-22

Family

ID=9245357

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/205731A BE890035A (fr) 1980-08-22 1981-08-21 Nouveaux derives du 4h-1,2,4-triazole, leur preparation, leur application comme medicament, les compositions les renfermant et les intermediaires obtenus

Country Status (24)

Country Link
US (3) US4512997A (fr)
JP (1) JPS5770875A (fr)
AT (1) AT378957B (fr)
AU (1) AU543946B2 (fr)
BE (1) BE890035A (fr)
CA (1) CA1208226A (fr)
CH (1) CH649994A5 (fr)
DE (1) DE3133185A1 (fr)
DK (1) DK370781A (fr)
ES (2) ES8306730A1 (fr)
FI (1) FI72971C (fr)
FR (1) FR2488891A1 (fr)
GB (1) GB2082581B (fr)
GR (1) GR75329B (fr)
HU (1) HU185647B (fr)
IE (1) IE51510B1 (fr)
IT (1) IT1171477B (fr)
LU (1) LU83576A1 (fr)
NL (1) NL8103903A (fr)
OA (2) OA06889A (fr)
PH (2) PH19890A (fr)
PT (1) PT73544B (fr)
SE (1) SE454173B (fr)
ZA (1) ZA815689B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4659729A (en) * 1980-08-22 1987-04-21 Roussel Uclaf Novel 4H-1,2,4-triazole derivatives

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2539127B1 (fr) * 1983-01-10 1985-08-23 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicaments
US5278180A (en) * 1984-09-24 1994-01-11 Roussel Uclaf 4,5-bis(aryl) 4H-1,2,4-triazoles derivatives and analgesic use
FR2570699B1 (fr) * 1984-09-24 1987-08-28 Roussel Uclaf Nouveau procede de preparation de derives du 4h-1,2,4-triazole, nouveaux triazoles ainsi obtenus, leur application comme medicaments et les compositions pharmaceutiques les renfermant
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US6362342B1 (en) * 1999-06-29 2002-03-26 Lion Bioscience Ag Triazole compounds and methods of making same
AU2001259298A1 (en) * 2000-05-02 2001-11-12 Advanced Medicine, Inc. Polyacid glycopeptide derivatives
ES2311711T3 (es) * 2002-02-07 2009-02-16 The Curators Of The University Of Missouri Compuestos de 4-(3-hidroxifenil) o 4-(3-alcoxifenil)-1,2,4-triazol activos como receptores de opioides.
KR20230117645A (ko) 2017-04-26 2023-08-08 오티아이 루미오닉스 인크. 표면의 코팅을 패턴화하는 방법 및 패턴화된 코팅을포함하는 장치
US11751415B2 (en) 2018-02-02 2023-09-05 Oti Lumionics Inc. Materials for forming a nucleation-inhibiting coating and devices incorporating same
WO2020178804A1 (fr) 2019-03-07 2020-09-10 Oti Lumionics Inc. Matériaux pour formation de revêtement inhibant la nucléation et dispositifs les incorporant

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1796403A (en) * 1931-03-17 Schaft
US3681374A (en) * 1970-08-11 1972-08-01 Asahi Chemical Ind Synthetic nacreous triazole crystals and method for production thereof
SU508198A3 (ru) * 1971-07-22 1976-03-25 Группо Лепетит С.П.А. (Фирма) Способ получени производных 1,2,4-триазола
AU7528974A (en) * 1973-11-13 1976-06-10 Commonwealth Scientific And Industrial Research Organization Triazoles
FR2269938A2 (en) * 1974-05-08 1975-12-05 Delalande Sa 5-Hydroxymethyl-3,4-diphenyl-1,2,4-triazoles - with anticholinergic, bronchodilator, antidepressant, analgesic, vasodilator activity, etc.
JPS56125376A (en) * 1980-03-07 1981-10-01 Mitsubishi Chem Ind Ltd Triazole derivative
FR2488891A1 (fr) * 1980-08-22 1982-02-26 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4659729A (en) * 1980-08-22 1987-04-21 Roussel Uclaf Novel 4H-1,2,4-triazole derivatives

Also Published As

Publication number Publication date
FI72971C (fi) 1987-08-10
CA1208226A (fr) 1986-07-22
AT378957B (de) 1985-10-25
PT73544B (fr) 1983-07-14
US4727084A (en) 1988-02-23
OA07537A (fr) 1985-03-31
AU543946B2 (en) 1985-05-09
JPH0261463B2 (fr) 1990-12-20
NL8103903A (nl) 1982-03-16
IT8149147A0 (it) 1981-08-21
PH19890A (en) 1986-08-13
IT1171477B (it) 1987-06-10
LU83576A1 (fr) 1982-04-14
ES504887A0 (es) 1983-06-01
PT73544A (fr) 1981-09-01
ES8306730A1 (es) 1983-06-01
ES8307227A1 (es) 1983-06-16
GB2082581B (en) 1985-02-13
SE454173B (sv) 1988-04-11
CH649994A5 (fr) 1985-06-28
PH21567A (en) 1987-12-11
OA06889A (fr) 1983-04-30
ATA368281A (de) 1985-03-15
DK370781A (da) 1982-02-23
JPS5770875A (en) 1982-05-01
IE811923L (en) 1982-02-22
GB2082581A (en) 1982-03-10
FI812585L (fi) 1982-02-23
SE8104515L (sv) 1982-02-23
GR75329B (fr) 1984-07-13
FR2488891A1 (fr) 1982-02-26
US4512997A (en) 1985-04-23
ZA815689B (en) 1982-08-25
DE3133185A1 (de) 1982-04-08
ES515419A0 (es) 1983-06-16
IE51510B1 (en) 1987-01-07
US4659729A (en) 1987-04-21
HU185647B (en) 1985-03-28
FI72971B (fi) 1987-04-30
AU7442681A (en) 1982-02-25
FR2488891B1 (fr) 1983-06-17

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: ROUSSEL-UCLAF

Effective date: 19900831