NZ563510A - Benzofuranyl derivatives as 5-HT6-receptor inhibitors - Google Patents
Benzofuranyl derivatives as 5-HT6-receptor inhibitorsInfo
- Publication number
- NZ563510A NZ563510A NZ563510A NZ56351006A NZ563510A NZ 563510 A NZ563510 A NZ 563510A NZ 563510 A NZ563510 A NZ 563510A NZ 56351006 A NZ56351006 A NZ 56351006A NZ 563510 A NZ563510 A NZ 563510A
- Authority
- NZ
- New Zealand
- Prior art keywords
- body weight
- disorders
- treatment
- compound according
- prophylaxis
- Prior art date
Links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Psychiatry (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Child & Adolescent Psychology (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Anesthesiology (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0501383 | 2005-06-17 | ||
| US70652305P | 2005-08-09 | 2005-08-09 | |
| PCT/EP2006/063249 WO2006134150A1 (en) | 2005-06-17 | 2006-06-15 | Benzofuranyl derivatives as 5-ht6-receptor inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ563510A true NZ563510A (en) | 2011-01-28 |
Family
ID=36659956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ563510A NZ563510A (en) | 2005-06-17 | 2006-06-15 | Benzofuranyl derivatives as 5-HT6-receptor inhibitors |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7582767B2 (enExample) |
| EP (1) | EP1896460B1 (enExample) |
| JP (1) | JP2008543813A (enExample) |
| KR (1) | KR20080017482A (enExample) |
| CN (1) | CN101193885B (enExample) |
| AU (1) | AU2006259082B2 (enExample) |
| BR (1) | BRPI0612746A2 (enExample) |
| CA (1) | CA2610383A1 (enExample) |
| DE (1) | DE602006008002D1 (enExample) |
| DK (1) | DK1896460T3 (enExample) |
| EA (1) | EA015671B1 (enExample) |
| ES (1) | ES2330145T3 (enExample) |
| IL (1) | IL187575A (enExample) |
| MX (1) | MX2007015988A (enExample) |
| NO (1) | NO20080354L (enExample) |
| NZ (1) | NZ563510A (enExample) |
| WO (1) | WO2006134150A1 (enExample) |
| ZA (1) | ZA200710468B (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0303480D0 (sv) * | 2003-12-19 | 2003-12-19 | Biovitrum Ab | Benzofuranes |
| WO2014013014A1 (en) | 2012-07-18 | 2014-01-23 | Fundació Privada Centre De Regulació Genòmica (Crg) | Jak inhibitors for activation of epidermal stem cell populations |
| CN103880797B (zh) * | 2014-03-26 | 2015-12-02 | 沈阳大学 | 苯并呋喃类化合物及其医药用途 |
| WO2018041989A1 (en) | 2016-09-02 | 2018-03-08 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods for diagnosing and treating refractory celiac disease type 2 |
| US20210393621A1 (en) | 2018-10-26 | 2021-12-23 | The Research Foundation For The State University Of New York | Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia |
| WO2020201362A2 (en) | 2019-04-02 | 2020-10-08 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods of predicting and preventing cancer in patients having premalignant lesions |
| WO2020212395A1 (en) | 2019-04-16 | 2020-10-22 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Use of jak inhibitors for the treatment of painful conditions involving nav1.7 channels |
| US20250283174A1 (en) | 2022-05-16 | 2025-09-11 | Institut National de la Santé et de la Recherche Médicale | Methods for assessing the exhaustion of hematopoietic stem cells induced by chronic inflammation |
| WO2026093435A1 (en) | 2024-10-31 | 2026-05-07 | Institut National de la Santé et de la Recherche Médicale | Use of jak inhibitors for enhancing the potency of immunotherapy in the treament of cancer |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3539573A (en) * | 1967-03-22 | 1970-11-10 | Jean Schmutz | 11-basic substituted dibenzodiazepines and dibenzothiazepines |
| AU767009B2 (en) | 1998-12-11 | 2003-10-30 | Virginia Commonwealth University | Selective 5-HT6 receptor ligands |
| CN100457726C (zh) | 2001-06-11 | 2009-02-04 | 比奥维特罗姆股份公开公司 | 取代的磺酰胺化合物、其制备方法及其作为治疗cns疾病、肥胖和ⅱ型糖尿病的药物的应用 |
| RS44204A (sr) * | 2001-11-22 | 2007-06-04 | Biovitrum Ab., | Inhibitori 11-beta- hidroksistereoidne dehidrogenaze tipa 1 |
| CN1662521A (zh) | 2002-06-20 | 2005-08-31 | 比奥维特罗姆股份公司 | 可用于治疗肥胖、ii型糖尿病和cns障碍的新化合物 |
| JP4754821B2 (ja) * | 2002-06-20 | 2011-08-24 | プロキシマゲン・リミテッド | 肥満症、ｉｉ型糖尿病およびｃｎｓ障害の治療に有用な新規化合物 |
| SE0303480D0 (sv) * | 2003-12-19 | 2003-12-19 | Biovitrum Ab | Benzofuranes |
-
2006
- 2006-06-05 US US11/447,524 patent/US7582767B2/en not_active Expired - Fee Related
- 2006-06-15 NZ NZ563510A patent/NZ563510A/en not_active IP Right Cessation
- 2006-06-15 CA CA002610383A patent/CA2610383A1/en not_active Abandoned
- 2006-06-15 ZA ZA200710468A patent/ZA200710468B/xx unknown
- 2006-06-15 DK DK06763743T patent/DK1896460T3/da active
- 2006-06-15 KR KR1020087001242A patent/KR20080017482A/ko not_active Ceased
- 2006-06-15 EP EP06763743A patent/EP1896460B1/en not_active Expired - Lifetime
- 2006-06-15 MX MX2007015988A patent/MX2007015988A/es active IP Right Grant
- 2006-06-15 BR BRPI0612746-0A patent/BRPI0612746A2/pt not_active IP Right Cessation
- 2006-06-15 DE DE602006008002T patent/DE602006008002D1/de not_active Expired - Lifetime
- 2006-06-15 ES ES06763743T patent/ES2330145T3/es not_active Expired - Lifetime
- 2006-06-15 AU AU2006259082A patent/AU2006259082B2/en not_active Ceased
- 2006-06-15 JP JP2008516325A patent/JP2008543813A/ja not_active Withdrawn
- 2006-06-15 WO PCT/EP2006/063249 patent/WO2006134150A1/en not_active Ceased
- 2006-06-15 CN CN2006800201432A patent/CN101193885B/zh not_active Expired - Fee Related
- 2006-06-15 EA EA200800071A patent/EA015671B1/ru not_active IP Right Cessation
-
2007
- 2007-11-22 IL IL187575A patent/IL187575A/en not_active IP Right Cessation
-
2008
- 2008-01-17 NO NO20080354A patent/NO20080354L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20080017482A (ko) | 2008-02-26 |
| NO20080354L (no) | 2008-01-17 |
| AU2006259082B2 (en) | 2011-07-14 |
| CN101193885B (zh) | 2011-07-27 |
| EA200800071A1 (ru) | 2008-10-30 |
| JP2008543813A (ja) | 2008-12-04 |
| WO2006134150A1 (en) | 2006-12-21 |
| EP1896460A1 (en) | 2008-03-12 |
| EP1896460B1 (en) | 2009-07-22 |
| CN101193885A (zh) | 2008-06-04 |
| EA015671B1 (ru) | 2011-10-31 |
| US20060293361A1 (en) | 2006-12-28 |
| ES2330145T3 (es) | 2009-12-04 |
| MX2007015988A (es) | 2008-03-07 |
| DE602006008002D1 (de) | 2009-09-03 |
| BRPI0612746A2 (pt) | 2010-11-30 |
| IL187575A (en) | 2012-12-31 |
| DK1896460T3 (da) | 2009-11-16 |
| US7582767B2 (en) | 2009-09-01 |
| IL187575A0 (en) | 2008-03-20 |
| AU2006259082A1 (en) | 2006-12-21 |
| HK1112918A1 (en) | 2008-09-19 |
| CA2610383A1 (en) | 2006-12-21 |
| ZA200710468B (en) | 2009-04-29 |
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Legal Events
| Date | Code | Title | Description |
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| ASS | Change of ownership |
Owner name: PROXIMAGEN LIMITED, GB Free format text: OLD OWNER(S): BIOVITRUM AB |
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| PSEA | Patent sealed | ||
| RENW | Renewal (renewal fees accepted) | ||
| LAPS | Patent lapsed |