BRPI0612746A2 - derivados de benzofuranil como inibidores do receptor 5-ht6 - Google Patents
derivados de benzofuranil como inibidores do receptor 5-ht6 Download PDFInfo
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- BRPI0612746A2 BRPI0612746A2 BRPI0612746-0A BRPI0612746A BRPI0612746A2 BR PI0612746 A2 BRPI0612746 A2 BR PI0612746A2 BR PI0612746 A BRPI0612746 A BR PI0612746A BR PI0612746 A2 BRPI0612746 A2 BR PI0612746A2
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Landscapes
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| SE0501383-4 | 2005-06-17 | ||
| SE0501383 | 2005-06-17 | ||
| US70652305P | 2005-08-09 | 2005-08-09 | |
| US60/706,523 | 2005-08-09 | ||
| PCT/EP2006/063249 WO2006134150A1 (en) | 2005-06-17 | 2006-06-15 | Benzofuranyl derivatives as 5-ht6-receptor inhibitors |
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| BRPI0612746A2 true BRPI0612746A2 (pt) | 2010-11-30 |
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| BRPI0612746-0A BRPI0612746A2 (pt) | 2005-06-17 | 2006-06-15 | derivados de benzofuranil como inibidores do receptor 5-ht6 |
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| US (1) | US7582767B2 (enExample) |
| EP (1) | EP1896460B1 (enExample) |
| JP (1) | JP2008543813A (enExample) |
| KR (1) | KR20080017482A (enExample) |
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| AU (1) | AU2006259082B2 (enExample) |
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| CA (1) | CA2610383A1 (enExample) |
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| WO2014013014A1 (en) | 2012-07-18 | 2014-01-23 | Fundació Privada Centre De Regulació Genòmica (Crg) | Jak inhibitors for activation of epidermal stem cell populations |
| CN103880797B (zh) * | 2014-03-26 | 2015-12-02 | 沈阳大学 | 苯并呋喃类化合物及其医药用途 |
| WO2018041989A1 (en) | 2016-09-02 | 2018-03-08 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods for diagnosing and treating refractory celiac disease type 2 |
| US20210393621A1 (en) | 2018-10-26 | 2021-12-23 | The Research Foundation For The State University Of New York | Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia |
| WO2020201362A2 (en) | 2019-04-02 | 2020-10-08 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods of predicting and preventing cancer in patients having premalignant lesions |
| WO2020212395A1 (en) | 2019-04-16 | 2020-10-22 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Use of jak inhibitors for the treatment of painful conditions involving nav1.7 channels |
| US20250283174A1 (en) | 2022-05-16 | 2025-09-11 | Institut National de la Santé et de la Recherche Médicale | Methods for assessing the exhaustion of hematopoietic stem cells induced by chronic inflammation |
| WO2026093435A1 (en) | 2024-10-31 | 2026-05-07 | Institut National de la Santé et de la Recherche Médicale | Use of jak inhibitors for enhancing the potency of immunotherapy in the treament of cancer |
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|---|---|---|---|---|
| US3539573A (en) * | 1967-03-22 | 1970-11-10 | Jean Schmutz | 11-basic substituted dibenzodiazepines and dibenzothiazepines |
| AU767009B2 (en) | 1998-12-11 | 2003-10-30 | Virginia Commonwealth University | Selective 5-HT6 receptor ligands |
| CN100457726C (zh) | 2001-06-11 | 2009-02-04 | 比奥维特罗姆股份公开公司 | 取代的磺酰胺化合物、其制备方法及其作为治疗cns疾病、肥胖和ⅱ型糖尿病的药物的应用 |
| RS44204A (sr) * | 2001-11-22 | 2007-06-04 | Biovitrum Ab., | Inhibitori 11-beta- hidroksistereoidne dehidrogenaze tipa 1 |
| CN1662521A (zh) | 2002-06-20 | 2005-08-31 | 比奥维特罗姆股份公司 | 可用于治疗肥胖、ii型糖尿病和cns障碍的新化合物 |
| JP4754821B2 (ja) * | 2002-06-20 | 2011-08-24 | プロキシマゲン・リミテッド | 肥満症、ｉｉ型糖尿病およびｃｎｓ障害の治療に有用な新規化合物 |
| SE0303480D0 (sv) * | 2003-12-19 | 2003-12-19 | Biovitrum Ab | Benzofuranes |
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2006
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- 2006-06-15 AU AU2006259082A patent/AU2006259082B2/en not_active Ceased
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|---|---|
| KR20080017482A (ko) | 2008-02-26 |
| NO20080354L (no) | 2008-01-17 |
| NZ563510A (en) | 2011-01-28 |
| AU2006259082B2 (en) | 2011-07-14 |
| CN101193885B (zh) | 2011-07-27 |
| EA200800071A1 (ru) | 2008-10-30 |
| JP2008543813A (ja) | 2008-12-04 |
| WO2006134150A1 (en) | 2006-12-21 |
| EP1896460A1 (en) | 2008-03-12 |
| EP1896460B1 (en) | 2009-07-22 |
| CN101193885A (zh) | 2008-06-04 |
| EA015671B1 (ru) | 2011-10-31 |
| US20060293361A1 (en) | 2006-12-28 |
| ES2330145T3 (es) | 2009-12-04 |
| MX2007015988A (es) | 2008-03-07 |
| DE602006008002D1 (de) | 2009-09-03 |
| IL187575A (en) | 2012-12-31 |
| DK1896460T3 (da) | 2009-11-16 |
| US7582767B2 (en) | 2009-09-01 |
| IL187575A0 (en) | 2008-03-20 |
| AU2006259082A1 (en) | 2006-12-21 |
| HK1112918A1 (en) | 2008-09-19 |
| CA2610383A1 (en) | 2006-12-21 |
| ZA200710468B (en) | 2009-04-29 |
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