NZ337515A - Use of cholinesterase inhibitors to treat disorders of attention - Google Patents
Use of cholinesterase inhibitors to treat disorders of attentionInfo
- Publication number
- NZ337515A NZ337515A NZ337515A NZ33751598A NZ337515A NZ 337515 A NZ337515 A NZ 337515A NZ 337515 A NZ337515 A NZ 337515A NZ 33751598 A NZ33751598 A NZ 33751598A NZ 337515 A NZ337515 A NZ 337515A
- Authority
- NZ
- New Zealand
- Prior art keywords
- group
- attention
- groups
- preferable
- disorders
- Prior art date
Links
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- 125000001424 substituent group Chemical group 0.000 abstract description 19
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- NRNCYVBFPDDJNE-UHFFFAOYSA-N pemoline Chemical compound O1C(N)=NC(=O)C1C1=CC=CC=C1 NRNCYVBFPDDJNE-UHFFFAOYSA-N 0.000 description 1
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- XAEFZNCEHLXOMS-UHFFFAOYSA-M potassium benzoate Chemical compound [K+].[O-]C(=O)C1=CC=CC=C1 XAEFZNCEHLXOMS-UHFFFAOYSA-M 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Enzymes And Modification Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3983297P | 1997-03-03 | 1997-03-03 | |
| PCT/IB1998/000508 WO1998039000A1 (en) | 1997-03-03 | 1998-03-03 | Use of cholinesterase inhibitors to treat disorders of attention |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ337515A true NZ337515A (en) | 2002-07-26 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ337515A NZ337515A (en) | 1997-03-03 | 1998-03-03 | Use of cholinesterase inhibitors to treat disorders of attention |
Country Status (12)
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|---|---|
| US (2) | US6455544B1 (https=) |
| EP (1) | EP0971713B1 (https=) |
| JP (1) | JP4095676B2 (https=) |
| AT (1) | ATE241358T1 (https=) |
| AU (1) | AU743609B2 (https=) |
| CA (1) | CA2282654C (https=) |
| DE (1) | DE69815090T2 (https=) |
| DK (1) | DK0971713T3 (https=) |
| ES (1) | ES2200313T3 (https=) |
| NZ (1) | NZ337515A (https=) |
| PT (1) | PT971713E (https=) |
| WO (1) | WO1998039000A1 (https=) |
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| ES2200313T3 (es) * | 1997-03-03 | 2004-03-01 | Eisai Co., Ltd. | Uso de inhibidores de la colinesterasa para tratar trastornos de la atencion. |
| GB9716879D0 (en) * | 1997-08-08 | 1997-10-15 | Shire Int Licensing Bv | Treatment of attention deficit disorders |
| US6429207B1 (en) | 1997-11-21 | 2002-08-06 | Nps Pharmaceuticals, Inc. | Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
| US20030153598A1 (en) * | 2000-07-25 | 2003-08-14 | Raymond Pratt | Methods for treating Parkinson's disease with cholinesterase inhibitors |
| EP2133078A1 (en) * | 2000-03-03 | 2009-12-16 | Eisai R&D Management Co., Ltd. | Use of a cholinesterase inhibitor for the treatment of dementia and cognitive impairments |
| EP1764101A1 (en) * | 2000-03-03 | 2007-03-21 | Eisai R&D Management Co., Ltd. | Use of a cholinesterase inhibitor for the treatment of dementia and cognitive impairments |
| US20060183776A9 (en) * | 2000-03-03 | 2006-08-17 | Eisai Co., Ltd. | Liquid dosage formulations of donepezil |
| CA2428971A1 (en) * | 2000-11-14 | 2003-05-01 | New River Pharmaceuticals Inc. | Conjugates of a therapeutic agent and a peptide carrier |
| WO2004034963A2 (en) * | 2002-05-17 | 2004-04-29 | Eisai Co., Ltd. | Methods and compositions using cholinesterase inhibitors |
| US20070053976A1 (en) * | 2002-05-17 | 2007-03-08 | Eisai R & D Management Co., Ltd. | Novel combination of drugs as antidepressant |
| EP1531822B1 (en) * | 2002-06-12 | 2009-08-05 | ChemoCentryx Inc | 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders |
| US20050256130A1 (en) * | 2002-06-12 | 2005-11-17 | Chemocentryx, Inc. | Substituted piperazines |
| US7842693B2 (en) * | 2002-06-12 | 2010-11-30 | Chemocentryx, Inc. | Substituted piperazines |
| US7589199B2 (en) | 2002-06-12 | 2009-09-15 | Chemocentryx, Inc. | Substituted piperazines |
| WO2005065645A2 (en) * | 2003-12-31 | 2005-07-21 | Actavis Group Hf | Donepezil formulations |
| US7435830B2 (en) | 2004-03-03 | 2008-10-14 | Chemocentryx, Inc. | Bicyclic and bridged nitrogen heterocycles |
| US7435831B2 (en) * | 2004-03-03 | 2008-10-14 | Chemocentryx, Inc. | Bicyclic and bridged nitrogen heterocycles |
| EP1741701A4 (en) * | 2004-04-28 | 2010-05-12 | Eisai R&D Man Co Ltd | PROCESS FOR THE PRODUCTION OF 1-BENZYL-4-¬ (5,6-DIMETHOXY-1INDANON) -2-YL METHYLPIPERIDINE AND HYDROCHLORIDE THEREOF |
| US7718674B2 (en) * | 2004-09-27 | 2010-05-18 | Bridge Pharma, Inc. | Methods of relieving neuropathic pain with the S-isomer of 2-{2[N-(2-indanyl)-N-phenylamino]ethyl}piperidine |
| WO2006037047A2 (en) * | 2004-09-27 | 2006-04-06 | Bridge Pharma, Inc. | The r-isomer of 2-{2-[n-(2-indanyl)-n-phenylamino]ethyl}piperidine and other dermal anesthetic agents |
| JP2008518955A (ja) | 2004-11-02 | 2008-06-05 | ノースウェスタン ユニバーシティ | ピリダジン化合物および方法 |
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| AU2006232517A1 (en) * | 2005-04-04 | 2006-10-12 | Eisai R&D Management Co., Ltd. | Dihydropyridine compounds and compositions for headaches |
| AU2006300492B2 (en) * | 2005-10-14 | 2011-08-25 | Eisai R & D Management Co., Ltd. | Process for producing 1-benzyl-4-[(5,6-dimethoxy-1indanon)-2-yl]methylpiperidine or hydrochloride thereof |
| AR058187A1 (es) * | 2005-11-14 | 2008-01-23 | Medichem Sa | Sintesis de un intermediario y formas polimorficas del mismo que se utilizan para la preparacion de clorhidrato de donepezilo. |
| US8158627B2 (en) | 2006-04-28 | 2012-04-17 | Northwestern University | Compositions and treatments using pyridazine compounds and cholinesterase inhibitors |
| CA2655809C (en) * | 2006-07-21 | 2013-10-01 | Bridge Pharma, Inc. | Dermal anesthetic compounds |
| US20100062045A1 (en) * | 2006-12-01 | 2010-03-11 | Nitto Denko Corporation | Method for suppressing coloring of adhesive prepartion containing donepezil and method for reducing amounts of donepezil-related substances formed |
| RU2452474C2 (ru) * | 2006-12-01 | 2012-06-10 | Нитто Денко Корпорейшн | Стабилизированная адгезивная композиция, содержащая донепезил |
| WO2008111590A2 (en) * | 2007-03-05 | 2008-09-18 | Eisai R & D Management Co., Ltd. | Ampa and nmda receptor antagonists for neurodegenerative diseases |
| WO2008139984A1 (en) * | 2007-04-26 | 2008-11-20 | Eisai R & D Management Co., Ltd. | Cinnamide compounds for dementia |
| KR100914691B1 (ko) * | 2007-08-10 | 2009-08-28 | 주식회사유한양행 | 도네페질 또는 그의 제조용 중간체의 제조방법 |
| CN102046171B (zh) * | 2008-05-30 | 2013-06-19 | 日东电工株式会社 | 经皮吸收制剂 |
| RU2481826C2 (ru) * | 2008-05-30 | 2013-05-20 | Нитто Денко Корпорейшн | Содержащий донепезил адгезивный препарат и упаковка для него |
| AU2011215870B2 (en) | 2010-02-09 | 2016-01-28 | The Johns Hopkins University | Methods and compositions for improving cognitive function |
| JP5951625B2 (ja) | 2010-11-24 | 2016-07-13 | ザ・トラスティーズ・オブ・コランビア・ユニバーシティー・イン・ザ・シティー・オブ・ニューヨークＴｈｅ Ｔｒｕｓｔｅｅｓ Ｏｆ Ｃｏｌｕｍｂｉａ Ｕｎｉｖｅｒｓｉｔｙ Ｉｎ Ｔｈｅ Ｃｉｔｙ Ｏｆ Ｎｅｗ Ｙｏｒｋ | 加齢性黄斑変性症およびシュタルガルト病の処置のための非レチノイドｒｂｐ４アンタゴニスト |
| US9333202B2 (en) | 2012-05-01 | 2016-05-10 | The Trustees Of Columbia University In The City Of New York | Non-retinoid antagonists for treatment of age-related macular degeneration and stargardt disease |
| US20140206667A1 (en) | 2012-11-14 | 2014-07-24 | Michela Gallagher | Methods and compositions for treating schizophrenia |
| US9265458B2 (en) | 2012-12-04 | 2016-02-23 | Sync-Think, Inc. | Application of smooth pursuit cognitive testing paradigms to clinical drug development |
| US9380976B2 (en) | 2013-03-11 | 2016-07-05 | Sync-Think, Inc. | Optical neuroinformatics |
| WO2014152018A1 (en) | 2013-03-14 | 2014-09-25 | The Trustees Of Columbia University In The City Of New York | Octahydrocyclopentapyrroles, their preparation and use |
| US9944644B2 (en) | 2013-03-14 | 2018-04-17 | The Trustees Of Columbia University In The City Of New York | Octahydropyrrolopyrroles their preparation and use |
| EP3495357B1 (en) | 2013-03-14 | 2021-05-05 | The Trustees of Columbia University in the City of New York | 4-phenylpiperidines, their preparation and use |
| US9938291B2 (en) | 2013-03-14 | 2018-04-10 | The Trustess Of Columbia University In The City Of New York | N-alkyl-2-phenoxyethanamines, their preparation and use |
| JP6433482B2 (ja) | 2013-03-15 | 2018-12-05 | エージンバイオ， インコーポレイテッド | 認知機能を改善するための方法および組成物 |
| WO2014144663A1 (en) | 2013-03-15 | 2014-09-18 | The Johns Hopkins University | Methods and compositions for improving cognitive function |
| SG11201608943VA (en) | 2014-04-30 | 2016-11-29 | Univ Columbia | Substituted 4-phenylpiperidines, their preparaiton and use |
| KR101732776B1 (ko) * | 2014-10-08 | 2017-05-04 | 영남대학교 산학협력단 | 신규한 인데노 피리디니움 유도체 화합물 및 이의 제조방법 |
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| FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
| US5064858A (en) * | 1988-08-17 | 1991-11-12 | Spectrum Pharmaceutical Corporation | Protected complex of procaine for the treatment of symptoms from narcotics addiction, tinnitus and Alzheimer's disease |
| WO1997003671A1 (en) * | 1995-07-14 | 1997-02-06 | Medeva Europe Limited | Composition comprising d-threo-methylphenidate and another drug |
| SK285312B6 (sk) | 1996-06-07 | 2006-10-05 | Eisai Co., Ltd. | Polymorf (III) donepezil hydrochloridu, spôsob jeho výroby a terapeutický prostriedok s jeho obsahom |
| ES2200313T3 (es) * | 1997-03-03 | 2004-03-01 | Eisai Co., Ltd. | Uso de inhibidores de la colinesterasa para tratar trastornos de la atencion. |
-
1998
- 1998-03-03 ES ES98905121T patent/ES2200313T3/es not_active Expired - Lifetime
- 1998-03-03 DE DE69815090T patent/DE69815090T2/de not_active Expired - Lifetime
- 1998-03-03 US US09/033,880 patent/US6455544B1/en not_active Expired - Lifetime
- 1998-03-03 DK DK98905121T patent/DK0971713T3/da active
- 1998-03-03 PT PT98905121T patent/PT971713E/pt unknown
- 1998-03-03 NZ NZ337515A patent/NZ337515A/en not_active IP Right Cessation
- 1998-03-03 JP JP53831598A patent/JP4095676B2/ja not_active Expired - Lifetime
- 1998-03-03 AU AU73215/98A patent/AU743609B2/en not_active Ceased
- 1998-03-03 EP EP98905121A patent/EP0971713B1/en not_active Expired - Lifetime
- 1998-03-03 CA CA002282654A patent/CA2282654C/en not_active Expired - Fee Related
- 1998-03-03 AT AT98905121T patent/ATE241358T1/de active
- 1998-03-03 WO PCT/IB1998/000508 patent/WO1998039000A1/en not_active Ceased
-
2002
- 2002-09-24 US US10/253,731 patent/US7105540B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| DE69815090D1 (de) | 2003-07-03 |
| DK0971713T3 (da) | 2003-09-22 |
| AU743609B2 (en) | 2002-01-31 |
| JP2001515480A (ja) | 2001-09-18 |
| US7105540B2 (en) | 2006-09-12 |
| AU7321598A (en) | 1998-09-22 |
| ES2200313T3 (es) | 2004-03-01 |
| WO1998039000A1 (en) | 1998-09-11 |
| US6455544B1 (en) | 2002-09-24 |
| EP0971713A1 (en) | 2000-01-19 |
| US20030055040A1 (en) | 2003-03-20 |
| JP4095676B2 (ja) | 2008-06-04 |
| CA2282654A1 (en) | 1998-09-11 |
| ATE241358T1 (de) | 2003-06-15 |
| CA2282654C (en) | 2009-02-03 |
| DE69815090T2 (de) | 2004-02-19 |
| EP0971713B1 (en) | 2003-05-28 |
| PT971713E (pt) | 2003-09-30 |
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