NO995030L - 5-(2-imidazolinylamino)benzimidazolforbindelser nyttige som <alfa>-2-adrenoseptoragonister - Google Patents

5-(2-imidazolinylamino)benzimidazolforbindelser nyttige som <alfa>-2-adrenoseptoragonister

Info

Publication number
NO995030L
NO995030L NO995030A NO995030A NO995030L NO 995030 L NO995030 L NO 995030L NO 995030 A NO995030 A NO 995030A NO 995030 A NO995030 A NO 995030A NO 995030 L NO995030 L NO 995030L
Authority
NO
Norway
Prior art keywords
imidazolinylamino
alpha
adrenoceptor agonists
compounds useful
benzimidazole compounds
Prior art date
Application number
NO995030A
Other languages
English (en)
Norwegian (no)
Other versions
NO995030D0 (no
Inventor
Thomas Lee Cupps
Sophie Eva Bogdan
Glen Edward Mieling
Nick Nikolaides
Raymond Todd Henry
Russell James Sheldon
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of NO995030D0 publication Critical patent/NO995030D0/no
Publication of NO995030L publication Critical patent/NO995030L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO995030A 1997-04-15 1999-10-15 5-(2-imidazolinylamino)benzimidazolforbindelser nyttige som <alfa>-2-adrenoseptoragonister NO995030L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4231697P 1997-04-15 1997-04-15
PCT/IB1998/000540 WO1998046595A1 (fr) 1997-04-15 1998-04-09 Composes de 5-(2-imidazolinylamino)benzimidazole utiles en tant qu'agonistes de l'adrenorecepteur alpha-2

Publications (2)

Publication Number Publication Date
NO995030D0 NO995030D0 (no) 1999-10-15
NO995030L true NO995030L (no) 1999-12-15

Family

ID=21921202

Family Applications (1)

Application Number Title Priority Date Filing Date
NO995030A NO995030L (no) 1997-04-15 1999-10-15 5-(2-imidazolinylamino)benzimidazolforbindelser nyttige som <alfa>-2-adrenoseptoragonister

Country Status (12)

Country Link
EP (1) EP0975627A1 (fr)
JP (1) JP2001519828A (fr)
KR (1) KR20010006440A (fr)
CN (1) CN1256691A (fr)
AU (1) AU6514498A (fr)
BR (1) BR9808904A (fr)
CA (1) CA2285610A1 (fr)
HU (1) HUP0002242A2 (fr)
ID (1) ID24081A (fr)
IL (1) IL132384A0 (fr)
NO (1) NO995030L (fr)
WO (1) WO1998046595A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996004270A1 (fr) 1994-08-04 1996-02-15 Synaptic Pharmaceutical Corporation Nouveaux derives de benzimidazole
US6495583B1 (en) 1997-03-25 2002-12-17 Synaptic Pharmaceutical Corporation Benzimidazole derivatives
WO1999026942A1 (fr) * 1997-11-24 1999-06-03 The Procter & Gamble Company 5-(2-imidazolinylamino)-benzimidazole, derives et procedes de preparation et d'utilisation de ces derniers en tant qu'agonistes du recepteur alpha-adrenergique ayant une meilleure stabilite metabolique
US20040167194A1 (en) * 2003-02-20 2004-08-26 Randall Jared Lynn Methods of making 6-[(4,5-Dihydro-1H-imidazol-2-yl)amino-]-7-methyl-1H-benzimidazole-4-carbonitrile and its preferred salt form
US8555875B2 (en) 2008-12-23 2013-10-15 Map Pharmaceuticals, Inc. Inhalation devices and related methods for administration of sedative hypnotic compounds
CN110540523B (zh) * 2018-07-05 2021-02-19 安徽圣诺贝化学科技有限公司 一种制备磺基取代苯并咪唑及其衍生物的方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5091528A (en) * 1990-09-12 1992-02-25 Allergan, Inc. 6- or 7- (2-imino-2-imidazolidine)-1,4-benzoxazines as α adrenergic agents
US5478858A (en) * 1993-12-17 1995-12-26 The Procter & Gamble Company 5-(2-imidazolinylamino) benzimidazole compounds useful as alpha-2 adrenoceptor agonists
WO1996004270A1 (fr) * 1994-08-04 1996-02-15 Synaptic Pharmaceutical Corporation Nouveaux derives de benzimidazole

Also Published As

Publication number Publication date
JP2001519828A (ja) 2001-10-23
NO995030D0 (no) 1999-10-15
HUP0002242A2 (hu) 2001-04-28
WO1998046595A1 (fr) 1998-10-22
BR9808904A (pt) 2005-02-22
IL132384A0 (en) 2001-03-19
EP0975627A1 (fr) 2000-02-02
AU6514498A (en) 1998-11-11
CA2285610A1 (fr) 1998-10-22
CN1256691A (zh) 2000-06-14
KR20010006440A (ko) 2001-01-26
ID24081A (id) 2000-07-06

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application