NO991023L - Stereospesifikk fremstilling av kirale 1-aryl- og 1-heteroaryl-2-substituerte etyl-2-aminer - Google Patents

Stereospesifikk fremstilling av kirale 1-aryl- og 1-heteroaryl-2-substituerte etyl-2-aminer

Info

Publication number
NO991023L
NO991023L NO991023A NO991023A NO991023L NO 991023 L NO991023 L NO 991023L NO 991023 A NO991023 A NO 991023A NO 991023 A NO991023 A NO 991023A NO 991023 L NO991023 L NO 991023L
Authority
NO
Norway
Prior art keywords
chiral
heteroaryl
amines
aryl
substituted ethyl
Prior art date
Application number
NO991023A
Other languages
English (en)
Norwegian (no)
Other versions
NO991023D0 (no
Inventor
Luc Grondard
Jean-Paul Casimir
Patrick Leon
Michael K O'brien
Matthew R Powers
Daniel Robin
Original Assignee
Rhone Poulenc Rorer Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Pharma filed Critical Rhone Poulenc Rorer Pharma
Publication of NO991023D0 publication Critical patent/NO991023D0/no
Publication of NO991023L publication Critical patent/NO991023L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/38—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reaction of ammonia or amines with sulfonic acids, or with esters, anhydrides, or halides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28—Halogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D203/22—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • C07D203/24—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO991023A 1996-09-12 1999-03-02 Stereospesifikk fremstilling av kirale 1-aryl- og 1-heteroaryl-2-substituerte etyl-2-aminer NO991023L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2600596P 1996-09-12 1996-09-12
PCT/US1997/015729 WO1998011064A1 (fr) 1996-09-12 1997-09-10 Preparation stereospecifique de 1-aryl- et 1-heteroaryl-2-substituees ethyl-2-amines chirales

Publications (2)

Publication Number Publication Date
NO991023D0 NO991023D0 (no) 1999-03-02
NO991023L true NO991023L (no) 1999-03-02

Family

ID=21829300

Family Applications (1)

Application Number Title Priority Date Filing Date
NO991023A NO991023L (no) 1996-09-12 1999-03-02 Stereospesifikk fremstilling av kirale 1-aryl- og 1-heteroaryl-2-substituerte etyl-2-aminer

Country Status (20)

Country Link
US (2) US6127550A (fr)
EP (1) EP0942900A4 (fr)
JP (1) JP2001501922A (fr)
KR (1) KR100317871B1 (fr)
CN (2) CN1112354C (fr)
AP (1) AP937A (fr)
AU (1) AU732332B2 (fr)
BG (1) BG103259A (fr)
BR (1) BR9711466A (fr)
CA (1) CA2265886A1 (fr)
EA (1) EA001364B1 (fr)
HK (1) HK1022296A1 (fr)
HU (1) HUP0000219A3 (fr)
IL (1) IL128813A0 (fr)
NO (1) NO991023L (fr)
OA (1) OA10991A (fr)
PL (1) PL331933A1 (fr)
SK (1) SK26999A3 (fr)
UA (1) UA54451C2 (fr)
WO (1) WO1998011064A1 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU225504B1 (en) * 1997-05-13 2007-01-29 Sanofi Aventis Novel halophenyl-(2-(2-thienyl)-ethylamino)-acetonitriles and process for producing them
SI1140933T1 (en) 1998-12-31 2005-02-28 Aventis Pharmaceuticals Inc. Process for preparing n6-substituted deaza-adenosine derivatives
KR100426030B1 (ko) * 2000-07-22 2004-04-03 (주) 한켐 락톤계 당화합물에서의 키랄성 전환방법
KR100440461B1 (ko) * 2000-08-19 2004-07-15 (주) 한켐 1,4-락톤을 이용한 ｌ-리보오스의 제조 방법
KR100433179B1 (ko) * 2001-11-10 2004-05-27 주식회사 삼천리제약 2-데옥시-ｌ-리보오스의 제조방법
CN100506919C (zh) * 2006-02-23 2009-07-01 中国科学院化学研究所 使用人血清蛋白对非手性菁染料聚集体进行手性诱导的方法
JP7229158B2 (ja) 2017-06-09 2023-02-27 中外製薬株式会社 Ｎ－置換アミノ酸を含むペプチドの合成方法
KR20210098476A (ko) * 2018-11-30 2021-08-10 추가이 세이야쿠 가부시키가이샤 펩티드 화합물 또는 아마이드 화합물의 탈보호법 및 고상 반응에 있어서의 탈수지 방법, 및 펩티드 화합물의 제조 방법

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3431152A (en) * 1967-03-23 1969-03-04 American Cyanamid Co Compositions containing aromatic sulfonyl aziridine as curing agents
US4933470A (en) * 1987-10-05 1990-06-12 Neorx Corporation Method of synthesis of vicinal diamines
ES2095960T3 (es) * 1990-09-25 1997-03-01 Rhone Poulenc Rorer Int Compuestos que tienen propiedades antihipertensivas y antiisquemicas.

Also Published As

Publication number Publication date
JP2001501922A (ja) 2001-02-13
HK1022296A1 (en) 2000-08-04
SK26999A3 (en) 1999-10-08
US6127550A (en) 2000-10-03
EP0942900A4 (fr) 2004-08-04
CN1388119A (zh) 2003-01-01
NO991023D0 (no) 1999-03-02
WO1998011064A1 (fr) 1998-03-19
BG103259A (bg) 2000-02-29
EA001364B1 (ru) 2001-02-26
OA10991A (en) 2001-11-07
CN1112354C (zh) 2003-06-25
AP937A (en) 2001-02-07
AU4256297A (en) 1998-04-02
US6433172B1 (en) 2002-08-13
HUP0000219A3 (en) 2001-04-28
CN1230176A (zh) 1999-09-29
CA2265886A1 (fr) 1998-03-19
BR9711466A (pt) 1999-08-24
AP9901476A0 (en) 1999-03-31
HUP0000219A2 (hu) 2000-12-28
EP0942900A1 (fr) 1999-09-22
KR20000036007A (ko) 2000-06-26
PL331933A1 (en) 1999-08-16
KR100317871B1 (ko) 2002-01-18
AU732332B2 (en) 2001-04-12
UA54451C2 (uk) 2003-03-17
EA199900281A1 (ru) 1999-08-26
IL128813A0 (en) 2000-01-31

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application