NO974151L - 6-substituerte pyrazolo [3,4-d] pyrimidin-4-oner og preparater og fremgangsmåter for anvendelse derav - Google Patents

6-substituerte pyrazolo [3,4-d] pyrimidin-4-oner og preparater og fremgangsmåter for anvendelse derav

Info

Publication number
NO974151L
NO974151L NO974151A NO974151A NO974151L NO 974151 L NO974151 L NO 974151L NO 974151 A NO974151 A NO 974151A NO 974151 A NO974151 A NO 974151A NO 974151 L NO974151 L NO 974151L
Authority
NO
Norway
Prior art keywords
pyrimidin
methods
substituted pyrazolo
preparations
ones
Prior art date
Application number
NO974151A
Other languages
English (en)
Norwegian (no)
Other versions
NO974151D0 (no
Inventor
Edward R Bacon
Sol J Daum
Baldev Singh
Original Assignee
Sanofi Winthrop Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Winthrop Inc filed Critical Sanofi Winthrop Inc
Publication of NO974151D0 publication Critical patent/NO974151D0/no
Publication of NO974151L publication Critical patent/NO974151L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO974151A 1995-03-10 1997-09-09 6-substituerte pyrazolo [3,4-d] pyrimidin-4-oner og preparater og fremgangsmåter for anvendelse derav NO974151L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/402,268 US5656629A (en) 1995-03-10 1995-03-10 6-substituted pyrazolo (3,4-d)pyrimidin-4-ones and compositions and methods of use thereof
PCT/US1996/002971 WO1996028429A1 (en) 1995-03-10 1996-03-05 6-SUBSTITUTED PYRAZOLO [3,4-d] PYRIMIDIN-4-ONES AND COMPOSITIONS AND METHODS OF USE THEREOF

Publications (2)

Publication Number Publication Date
NO974151D0 NO974151D0 (no) 1997-09-09
NO974151L true NO974151L (no) 1997-11-04

Family

ID=23591222

Family Applications (1)

Application Number Title Priority Date Filing Date
NO974151A NO974151L (no) 1995-03-10 1997-09-09 6-substituerte pyrazolo [3,4-d] pyrimidin-4-oner og preparater og fremgangsmåter for anvendelse derav

Country Status (13)

Country Link
US (2) US5656629A (de)
EP (1) EP0813527A4 (de)
JP (1) JPH11501923A (de)
KR (1) KR19980702891A (de)
AU (1) AU708750B2 (de)
CA (1) CA2211669A1 (de)
CZ (1) CZ280597A3 (de)
HU (1) HUP9801336A3 (de)
NO (1) NO974151L (de)
NZ (1) NZ306035A (de)
PL (1) PL322380A1 (de)
WO (1) WO1996028429A1 (de)
ZA (1) ZA961947B (de)

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CN101906106A (zh) * 2003-09-18 2010-12-08 康福玛医药公司 作为hsp90-抑制剂的新的杂环化合物
US7572799B2 (en) 2003-11-24 2009-08-11 Pfizer Inc Pyrazolo[4,3-d]pyrimidines as Phosphodiesterase Inhibitors
DE102004001873A1 (de) * 2004-01-14 2005-09-29 Bayer Healthcare Ag Cyanopyrimidinone
MXPA06009462A (es) * 2004-02-27 2007-03-15 Hoffmann La Roche Derivados pirazolo heteroaril fusionados.
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MX2008002385A (es) * 2005-08-25 2008-03-18 Hoffmann La Roche Inhibidores de proteinas cinasas activads por mitogenos p38 y metodos para utilizarlos.
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US8648085B2 (en) * 2007-11-30 2014-02-11 Boehringer Ingelheim International Gmbh 1, 5-dihydro-pyrazolo (3, 4-D) pyrimidin-4-one derivatives and their use as PDE9A mudulators for the treatment of CNS disorders
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JP5894148B2 (ja) 2010-05-31 2016-03-23 イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． 有機化合物
JP5879336B2 (ja) 2010-05-31 2016-03-08 イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． 有機化合物
BR112013003097B1 (pt) 2010-08-12 2021-03-16 Boehringer Ingelheim International Gmbh 6-cicloalquil-pirazolopirimidinonas e composição farmacêutica
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Also Published As

Publication number Publication date
ZA961947B (en) 1996-10-07
JPH11501923A (ja) 1999-02-16
AU708750B2 (en) 1999-08-12
AU5418896A (en) 1996-10-02
US5977118A (en) 1999-11-02
CA2211669A1 (en) 1996-09-19
KR19980702891A (ko) 1998-08-05
EP0813527A4 (de) 1998-09-09
NZ306035A (en) 1999-07-29
HUP9801336A2 (hu) 1998-10-28
MX9706876A (es) 1998-06-28
US5656629A (en) 1997-08-12
EP0813527A1 (de) 1997-12-29
NO974151D0 (no) 1997-09-09
CZ280597A3 (cs) 1998-04-15
HUP9801336A3 (en) 2000-07-28
WO1996028429A1 (en) 1996-09-19
PL322380A1 (en) 1998-01-19

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