NO965353L - 3-amino-2-okso-1-piperidineddiksyrederivater som enzyminhibitorer - Google Patents

3-amino-2-okso-1-piperidineddiksyrederivater som enzyminhibitorer

Info

Publication number
NO965353L
NO965353L NO965353A NO965353A NO965353L NO 965353 L NO965353 L NO 965353L NO 965353 A NO965353 A NO 965353A NO 965353 A NO965353 A NO 965353A NO 965353 L NO965353 L NO 965353L
Authority
NO
Norway
Prior art keywords
carbon atoms
alkyl
atoms
ring
amino
Prior art date
Application number
NO965353A
Other languages
English (en)
Norwegian (no)
Other versions
NO965353D0 (no
Inventor
Joseph Edward Semple
Robert John Ardecky
Ruth F Nutt
William Charles Ripka
David C Rowley
Marguerita S L Lim-Wilby
Terrence Brunck
Original Assignee
Corvas Int Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US1995/007661 external-priority patent/WO1995035311A1/en
Application filed by Corvas Int Inc filed Critical Corvas Int Inc
Publication of NO965353D0 publication Critical patent/NO965353D0/no
Publication of NO965353L publication Critical patent/NO965353L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO965353A 1994-06-17 1996-12-13 3-amino-2-okso-1-piperidineddiksyrederivater som enzyminhibitorer NO965353L (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US26137894A 1994-06-17 1994-06-17
US35683194A 1994-12-13 1994-12-13
US48700795A 1995-06-07 1995-06-07
PCT/US1995/007661 WO1995035311A1 (en) 1994-06-17 1995-06-19 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors

Publications (2)

Publication Number Publication Date
NO965353D0 NO965353D0 (no) 1996-12-13
NO965353L true NO965353L (no) 1997-02-17

Family

ID=27401400

Family Applications (1)

Application Number Title Priority Date Filing Date
NO965353A NO965353L (no) 1994-06-17 1996-12-13 3-amino-2-okso-1-piperidineddiksyrederivater som enzyminhibitorer

Country Status (8)

Country Link
EP (1) EP0802923A1 (zh)
CN (1) CN1151166A (zh)
AU (1) AU700808B2 (zh)
BR (1) BR9508048A (zh)
CA (1) CA2192210A1 (zh)
MX (1) MX9606566A (zh)
NO (1) NO965353L (zh)
NZ (1) NZ288940A (zh)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4192875A (en) * 1979-02-02 1980-03-11 Merck & Co., Inc. Cyclic hexapeptide

Also Published As

Publication number Publication date
NO965353D0 (no) 1996-12-13
AU700808B2 (en) 1999-01-14
EP0802923A1 (en) 1997-10-29
AU2863095A (en) 1996-01-15
CA2192210A1 (en) 1995-12-28
MX9606566A (es) 1997-07-31
CN1151166A (zh) 1997-06-04
BR9508048A (pt) 1997-11-18
NZ288940A (en) 1999-01-28

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