BR9508048A - Derivados 3-amino 2-oxo 1-piperidina acéticos como inibidores de enzimas - Google Patents

Derivados 3-amino 2-oxo 1-piperidina acéticos como inibidores de enzimas

Info

Publication number
BR9508048A
BR9508048A BR9508048A BR9508048A BR9508048A BR 9508048 A BR9508048 A BR 9508048A BR 9508048 A BR9508048 A BR 9508048A BR 9508048 A BR9508048 A BR 9508048A BR 9508048 A BR9508048 A BR 9508048A
Authority
BR
Brazil
Prior art keywords
oxo
acetic
amino
enzyme inhibitors
piperidine derivatives
Prior art date
Application number
BR9508048A
Other languages
English (en)
Portuguese (pt)
Inventor
Joseph Edward Semple
Robert J Ardecky
Ruth F Nutt
William Charles Ripka
David Scott Rowley
Marquerida S L Lim-Wilby
Terence K Brunck
Original Assignee
Corvas Int Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Corvas Int Inc filed Critical Corvas Int Inc
Priority claimed from PCT/US1995/007661 external-priority patent/WO1995035311A1/en
Publication of BR9508048A publication Critical patent/BR9508048A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
BR9508048A 1994-06-17 1995-06-19 Derivados 3-amino 2-oxo 1-piperidina acéticos como inibidores de enzimas BR9508048A (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US26137894A 1994-06-17 1994-06-17
US35683194A 1994-12-13 1994-12-13
US48700795A 1995-06-07 1995-06-07
PCT/US1995/007661 WO1995035311A1 (en) 1994-06-17 1995-06-19 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors

Publications (1)

Publication Number Publication Date
BR9508048A true BR9508048A (pt) 1997-11-18

Family

ID=27401400

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9508048A BR9508048A (pt) 1994-06-17 1995-06-19 Derivados 3-amino 2-oxo 1-piperidina acéticos como inibidores de enzimas

Country Status (8)

Country Link
EP (1) EP0802923A1 (zh)
CN (1) CN1151166A (zh)
AU (1) AU700808B2 (zh)
BR (1) BR9508048A (zh)
CA (1) CA2192210A1 (zh)
MX (1) MX9606566A (zh)
NO (1) NO965353L (zh)
NZ (1) NZ288940A (zh)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4192875A (en) * 1979-02-02 1980-03-11 Merck & Co., Inc. Cyclic hexapeptide

Also Published As

Publication number Publication date
NO965353D0 (no) 1996-12-13
AU700808B2 (en) 1999-01-14
EP0802923A1 (en) 1997-10-29
AU2863095A (en) 1996-01-15
CA2192210A1 (en) 1995-12-28
NO965353L (no) 1997-02-17
MX9606566A (es) 1997-07-31
CN1151166A (zh) 1997-06-04
NZ288940A (en) 1999-01-28

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Legal Events

Date Code Title Description
B06A Notification to applicant to reply to the report for non-patentability or inadequacy of the application according art. 36 industrial patent law
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements
B08F Application fees: dismissal - article 86 of industrial property law