CA2192210A1 - 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors - Google Patents

3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors

Info

Publication number
CA2192210A1
CA2192210A1 CA002192210A CA2192210A CA2192210A1 CA 2192210 A1 CA2192210 A1 CA 2192210A1 CA 002192210 A CA002192210 A CA 002192210A CA 2192210 A CA2192210 A CA 2192210A CA 2192210 A1 CA2192210 A1 CA 2192210A1
Authority
CA
Canada
Prior art keywords
substituted
compound according
carbon atoms
argininal
gly
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002192210A
Other languages
English (en)
French (fr)
Inventor
Joseph Edward Semple
Robert J. Ardecky
Ruth F. Nutt
William Charles Ripka
David C. Rowley
Marguerita S. L. Lim-Wilby
Terence K. Brunck
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dendreon Pharmaceuticals LLC
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2192210A1 publication Critical patent/CA2192210A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
CA002192210A 1994-06-17 1995-06-19 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors Abandoned CA2192210A1 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US26137894A 1994-06-17 1994-06-17
US35683194A 1994-12-13 1994-12-13
US08/261,378 1994-12-13
US08/356,831 1994-12-13
US48700795A 1995-06-07 1995-06-07
US08/487,007 1995-06-07

Publications (1)

Publication Number Publication Date
CA2192210A1 true CA2192210A1 (en) 1995-12-28

Family

ID=27401400

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002192210A Abandoned CA2192210A1 (en) 1994-06-17 1995-06-19 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors

Country Status (8)

Country Link
EP (1) EP0802923A1 (zh)
CN (1) CN1151166A (zh)
AU (1) AU700808B2 (zh)
BR (1) BR9508048A (zh)
CA (1) CA2192210A1 (zh)
MX (1) MX9606566A (zh)
NO (1) NO965353L (zh)
NZ (1) NZ288940A (zh)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4192875A (en) * 1979-02-02 1980-03-11 Merck & Co., Inc. Cyclic hexapeptide

Also Published As

Publication number Publication date
NO965353D0 (no) 1996-12-13
AU700808B2 (en) 1999-01-14
EP0802923A1 (en) 1997-10-29
AU2863095A (en) 1996-01-15
NO965353L (no) 1997-02-17
MX9606566A (es) 1997-07-31
CN1151166A (zh) 1997-06-04
BR9508048A (pt) 1997-11-18
NZ288940A (en) 1999-01-28

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Legal Events

Date Code Title Description
FZDE Dead