NO754024L - - Google Patents

Info

Publication number
NO754024L
NO754024L NO754024A NO754024A NO754024L NO 754024 L NO754024 L NO 754024L NO 754024 A NO754024 A NO 754024A NO 754024 A NO754024 A NO 754024A NO 754024 L NO754024 L NO 754024L
Authority
NO
Norway
Application number
NO754024A
Other languages
Norwegian (no)
Other versions
NO145382B (no
NO145382C (no
Inventor
K H Mayer
S Petersen
E Klauke
F Hoffmeister
W Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO754024L publication Critical patent/NO754024L/no
Publication of NO145382B publication Critical patent/NO145382B/no
Publication of NO145382C publication Critical patent/NO145382C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
NO754024A 1974-12-13 1975-11-28 Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater. NO145382C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (3)

Publication Number Publication Date
NO754024L true NO754024L (enEXAMPLES) 1976-06-15
NO145382B NO145382B (no) 1981-11-30
NO145382C NO145382C (no) 1982-03-10

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
NO754024A NO145382C (no) 1974-12-13 1975-11-28 Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater.

Country Status (27)

Country Link
US (1) US4051252A (enEXAMPLES)
JP (1) JPS5182266A (enEXAMPLES)
AT (1) AT343653B (enEXAMPLES)
BE (1) BE836528A (enEXAMPLES)
CA (1) CA1059523A (enEXAMPLES)
CH (1) CH622250A5 (enEXAMPLES)
CS (1) CS189731B2 (enEXAMPLES)
DD (1) DD125484A5 (enEXAMPLES)
DE (1) DE2458965C3 (enEXAMPLES)
DK (1) DK137082C (enEXAMPLES)
ES (1) ES443429A1 (enEXAMPLES)
FI (1) FI753493A7 (enEXAMPLES)
FR (1) FR2293928A1 (enEXAMPLES)
GB (1) GB1490306A (enEXAMPLES)
HK (1) HK52580A (enEXAMPLES)
HU (1) HU173557B (enEXAMPLES)
IE (1) IE42208B1 (enEXAMPLES)
IL (1) IL48642A (enEXAMPLES)
KE (1) KE3078A (enEXAMPLES)
LU (1) LU73993A1 (enEXAMPLES)
NL (1) NL7514521A (enEXAMPLES)
NO (1) NO145382C (enEXAMPLES)
PL (1) PL99858B1 (enEXAMPLES)
SE (1) SE419645B (enEXAMPLES)
SU (1) SU604487A3 (enEXAMPLES)
YU (1) YU315275A (enEXAMPLES)
ZA (1) ZA757777B (enEXAMPLES)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
ZA200301703B (en) * 2000-09-15 2004-03-02 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
WO2002022602A2 (en) 2000-09-15 2002-03-21 Vertex Pharmaceuticals Incorporated Triazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6664247B2 (en) * 2000-12-21 2003-12-16 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
WO2003028720A1 (en) 2001-09-26 2003-04-10 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
MXPA04007697A (es) * 2002-02-06 2004-11-10 Vertex Pharma Compuestos de heteroarilo utiles como inhibidores de gsk-3.
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
WO2003078427A1 (en) 2002-03-15 2003-09-25 Vertex Pharmaceuticals, Inc. Azolylaminoazines as inhibitors of protein kinases
CA2486101C (en) 2002-05-17 2009-07-07 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
CA2494100C (en) 2002-08-02 2011-10-11 Vertex Pharmaceuticals Incorporated Pyrazole compositions useful as inhibitors of gsk-3
EP1556053A4 (en) * 2002-10-31 2006-04-19 Amgen Inc ANTI-INFLAMMATORY AGENTS
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
JP2007513184A (ja) * 2003-12-04 2007-05-24 バーテックス ファーマシューティカルズ インコーポレイテッド プロテインキナーゼのインヒビターとして有用なキノキサリン
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
JP2009504771A (ja) 2005-08-18 2009-02-05 バーテックス ファーマシューティカルズ インコーポレイテッド ピラジンキナーゼ阻害剤
AU2006311831C1 (en) 2005-11-03 2013-11-07 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CN101466374B (zh) * 2006-04-14 2012-03-21 雅培制药有限公司 制备抑制香草素亚型1(vr1)受体的吲唑基脲的方法
ATE457311T1 (de) 2006-11-02 2010-02-15 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyridine und aminopyrimidine
AU2007333650A1 (en) 2006-12-19 2008-06-26 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
WO2008112651A2 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
WO2008112642A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
WO2008112646A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyridines useful as inhibitors of protein kinases
MX2009011059A (es) 2007-04-13 2009-11-26 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasas.
WO2008137619A2 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
CA2694381A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CA2688584A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CA2687966A1 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
AR067762A1 (es) 2007-07-31 2009-10-21 Vertex Pharma Proceso para preparar 5-fluoro-1h-pirazolo (3,4-b) piridin-3-amina y derivados de la misma
CN102215816A (zh) * 2008-09-03 2011-10-12 沃泰克斯药物股份有限公司 共晶和包含所述共晶的药物制剂
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
EP2890684B1 (en) 2012-07-24 2018-02-14 Bial-Portela & CA, S.A. Urea compounds and their use as enzyme inhibitors
CA2880299A1 (en) * 2012-07-27 2014-01-30 Bial - Portela & Ca, S.A. Process for the synthesis of substituted urea compounds
PL3024825T3 (pl) 2013-07-24 2017-12-29 BIAL - PORTELA & Cª, S.A. Imidazolokarboksyamidy i ich zastosowanie jako inhibitorów faah

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (enEXAMPLES) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
HU173557B (hu) 1979-06-28
DK137082B (da) 1978-01-16
YU315275A (en) 1982-02-28
DE2458965A1 (de) 1976-06-16
SU604487A3 (ru) 1978-04-25
DK567275A (da) 1976-06-14
PL99858B1 (pl) 1978-08-31
LU73993A1 (enEXAMPLES) 1976-11-11
FR2293928A1 (fr) 1976-07-09
GB1490306A (en) 1977-11-02
DE2458965B2 (de) 1979-02-22
ZA757777B (en) 1976-11-24
IL48642A0 (en) 1976-02-29
DD125484A5 (enEXAMPLES) 1977-04-20
SE419645B (sv) 1981-08-17
DE2458965C3 (de) 1979-10-11
IL48642A (en) 1979-12-30
BE836528A (fr) 1976-06-11
CA1059523A (en) 1979-07-31
ES443429A1 (es) 1977-04-16
KE3078A (en) 1980-10-03
AU8717075A (en) 1977-06-09
ATA939775A (de) 1977-10-15
NL7514521A (nl) 1976-06-15
DK137082C (da) 1978-06-19
NO145382B (no) 1981-11-30
SE7513990L (sv) 1976-06-14
FI753493A7 (enEXAMPLES) 1976-06-14
IE42208B1 (en) 1980-06-18
CH622250A5 (enEXAMPLES) 1981-03-31
HK52580A (en) 1980-09-26
US4051252A (en) 1977-09-27
CS189731B2 (en) 1979-04-30
NO145382C (no) 1982-03-10
JPS5182266A (en) 1976-07-19
IE42208L (en) 1976-06-13
AT343653B (de) 1978-06-12
FR2293928B1 (enEXAMPLES) 1979-09-21

Similar Documents

Publication Publication Date Title
AU495028B2 (enEXAMPLES)
AU495920B2 (enEXAMPLES)
AR198841Q (enEXAMPLES)
AR203034Q (enEXAMPLES)
AU7474774A (enEXAMPLES)
AU6717074A (enEXAMPLES)
BG19713A1 (enEXAMPLES)
BG19772A1 (enEXAMPLES)
AU481044A (enEXAMPLES)
AU481375A (enEXAMPLES)
AU481457A (enEXAMPLES)
AU481580A (enEXAMPLES)
BG20011A1 (enEXAMPLES)
AU482043A (enEXAMPLES)
AU482294A (enEXAMPLES)
AU482309A (enEXAMPLES)
AU480463A (enEXAMPLES)
AU480145A (enEXAMPLES)
AU479987A (enEXAMPLES)
AU7253373A (enEXAMPLES)
AU479629A (enEXAMPLES)
BE828550A (enEXAMPLES)
BE830029A (enEXAMPLES)
BG19618A1 (enEXAMPLES)
BG20200A1 (enEXAMPLES)