NO328499B1 - Kinuklidyl-N-fenyl-N-alkylkarbamater og anvendelse derav ved fremstilling av medikamenter - Google Patents
Kinuklidyl-N-fenyl-N-alkylkarbamater og anvendelse derav ved fremstilling av medikamenter Download PDFInfo
- Publication number
- NO328499B1 NO328499B1 NO20026211A NO20026211A NO328499B1 NO 328499 B1 NO328499 B1 NO 328499B1 NO 20026211 A NO20026211 A NO 20026211A NO 20026211 A NO20026211 A NO 20026211A NO 328499 B1 NO328499 B1 NO 328499B1
- Authority
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- Norway
- Prior art keywords
- quinuclidyl
- benzyl
- alkyl
- group
- crc4
- Prior art date
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- 230000002485 urinary effect Effects 0.000 description 1
- BDIAUFOIMFAIPU-UHFFFAOYSA-N valepotriate Natural products CC(C)CC(=O)OC1C=C(C(=COC2OC(=O)CC(C)C)COC(C)=O)C2C11CO1 BDIAUFOIMFAIPU-UHFFFAOYSA-N 0.000 description 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03B—APPARATUS OR ARRANGEMENTS FOR TAKING PHOTOGRAPHS OR FOR PROJECTING OR VIEWING THEM; APPARATUS OR ARRANGEMENTS EMPLOYING ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ACCESSORIES THEREFOR
- G03B27/00—Photographic printing apparatus
- G03B27/02—Exposure apparatus for contact printing
-
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03B—APPARATUS OR ARRANGEMENTS FOR TAKING PHOTOGRAPHS OR FOR PROJECTING OR VIEWING THEM; APPARATUS OR ARRANGEMENTS EMPLOYING ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ACCESSORIES THEREFOR
- G03B27/00—Photographic printing apparatus
- G03B27/02—Exposure apparatus for contact printing
- G03B27/14—Details
- G03B27/16—Illumination arrangements, e.g. positioning of lamps, positioning of reflectors
-
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03B—APPARATUS OR ARRANGEMENTS FOR TAKING PHOTOGRAPHS OR FOR PROJECTING OR VIEWING THEM; APPARATUS OR ARRANGEMENTS EMPLOYING ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ACCESSORIES THEREFOR
- G03B27/00—Photographic printing apparatus
- G03B27/02—Exposure apparatus for contact printing
- G03B27/14—Details
- G03B27/30—Details adapted to be combined with processing apparatus
- G03B27/303—Gas processing
-
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03D—APPARATUS FOR PROCESSING EXPOSED PHOTOGRAPHIC MATERIALS; ACCESSORIES THEREFOR
- G03D13/00—Processing apparatus or accessories therefor, not covered by groups G11B3/00 - G11B11/00
- G03D13/002—Heat development apparatus, e.g. Kalvar
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES200001661 | 2000-06-27 | ||
PCT/ES2001/000252 WO2002000652A1 (es) | 2000-06-27 | 2001-06-25 | Carbamatos derivados de arilalquilaminas |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20026211D0 NO20026211D0 (no) | 2002-12-23 |
NO20026211L NO20026211L (no) | 2003-02-26 |
NO328499B1 true NO328499B1 (no) | 2010-03-01 |
Family
ID=8494130
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20026211A NO328499B1 (no) | 2000-06-27 | 2002-12-23 | Kinuklidyl-N-fenyl-N-alkylkarbamater og anvendelse derav ved fremstilling av medikamenter |
Country Status (30)
Country | Link |
---|---|
US (2) | US6916828B2 (ja) |
EP (1) | EP1300407B2 (ja) |
JP (1) | JP5046465B2 (ja) |
KR (1) | KR100751981B1 (ja) |
CN (1) | CN1227251C (ja) |
AP (1) | AP1420A (ja) |
AT (1) | ATE260277T1 (ja) |
AU (2) | AU6610001A (ja) |
BG (1) | BG66102B1 (ja) |
BR (1) | BR0112297A (ja) |
CA (1) | CA2414514C (ja) |
CR (1) | CR6889A (ja) |
CZ (1) | CZ294251B6 (ja) |
DE (2) | DE20122417U1 (ja) |
DK (1) | DK1300407T4 (ja) |
EA (1) | EA005520B1 (ja) |
ES (1) | ES2213703T5 (ja) |
HK (1) | HK1054934A1 (ja) |
HU (1) | HU229306B1 (ja) |
IL (1) | IL153707A0 (ja) |
MX (1) | MXPA03000141A (ja) |
NO (1) | NO328499B1 (ja) |
OA (1) | OA12300A (ja) |
PL (1) | PL201530B1 (ja) |
PT (1) | PT1300407E (ja) |
SI (1) | SI1300407T2 (ja) |
TR (1) | TR200400420T4 (ja) |
UA (1) | UA72632C2 (ja) |
WO (1) | WO2002000652A1 (ja) |
ZA (1) | ZA200300644B (ja) |
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GB9913083D0 (en) | 1999-06-04 | 1999-08-04 | Novartis Ag | Organic compounds |
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MXPA03005583A (es) * | 2000-12-22 | 2004-05-05 | Almirall Prodesfarma Ag | Derivados de carbamato de quinuclidina y su uso como antagonistas m3. |
KR100869721B1 (ko) | 2000-12-28 | 2008-11-21 | 알미랄 에이쥐 | 신규한 퀴누클리딘 유도체 및 그를 함유한 의약 조성물 |
NZ554913A (en) | 2001-12-14 | 2009-01-31 | Targacept Inc | Methods and compositions for the treatment of central nervous system disorders |
EA006505B1 (ru) * | 2001-12-20 | 2005-12-29 | Лабораториос С.А.Л.В.А.Т.,С.А. | Производные карбамата 1-алкил-1-азониабицикло[2.2.2]октана и их применение в качестве антагонистов мускаринового рецептора |
ES2203327B1 (es) * | 2002-06-21 | 2005-06-16 | Almirall Prodesfarma, S.A. | Nuevos carbamatos de quinuclidina y composiciones farmaceuticas que los contienen. |
ES2204295B1 (es) | 2002-07-02 | 2005-08-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de quinuclidina-amida. |
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AR044519A1 (es) | 2003-05-02 | 2005-09-14 | Novartis Ag | Derivados de piridin-tiazol amina y de pirimidin-tiazol amina |
GB0401334D0 (en) | 2004-01-21 | 2004-02-25 | Novartis Ag | Organic compounds |
GB0411056D0 (en) | 2004-05-18 | 2004-06-23 | Novartis Ag | Organic compounds |
ES2246170B1 (es) * | 2004-07-29 | 2007-04-01 | Almirall Prodesfarma, S.A. | Nuevo procedimiento para preparar derivados de carbamato de quinuclidinio. |
GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
GB0424284D0 (en) | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
GB0426164D0 (en) | 2004-11-29 | 2004-12-29 | Novartis Ag | Organic compounds |
GB0507577D0 (en) | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
GB0510390D0 (en) | 2005-05-20 | 2005-06-29 | Novartis Ag | Organic compounds |
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BRPI0710573A2 (pt) | 2006-04-21 | 2012-02-28 | Novartis Ag | compostos orgánicos, usos e processos para a preparação dos referidos compostos, bem como composição farmacêutica compreendendo os mesmos |
EP1882691A1 (en) | 2006-07-26 | 2008-01-30 | CHIESI FARMACEUTICI S.p.A. | Quinuclidine derivatives as M3 antagonists |
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US3287471A (en) | 1964-05-05 | 1966-11-22 | Searle & Co | Pyrrolidinyl nu-phenyl-nu-benzylcarbamates |
JPH0495071A (ja) | 1990-08-10 | 1992-03-27 | Kyorin Pharmaceut Co Ltd | カルバミン酸誘導体 |
WO1995006635A1 (fr) * | 1993-09-02 | 1995-03-09 | Yamanouchi Pharmaceutical Co., Ltd. | Derive de carbamate et medicament le contenant |
WO1995021820A1 (fr) * | 1994-02-10 | 1995-08-17 | Yamanouchi Pharmaceutical Co., Ltd. | Nouveau derive du carbamate et composition correspondante |
NO2005012I1 (no) * | 1994-12-28 | 2005-06-06 | Debio Rech Pharma Sa | Triptorelin og farmasoytisk akseptable salter derav |
JPH08198751A (ja) * | 1995-01-19 | 1996-08-06 | Yamanouchi Pharmaceut Co Ltd | カルバメート誘導体 |
UA72632C2 (uk) * | 2000-06-27 | 2005-03-15 | Лабораторіос С.А.Л.В.А.Т., С.А. | Карбамати, похідні від арилалкіламінів |
MXPA03005583A (es) * | 2000-12-22 | 2004-05-05 | Almirall Prodesfarma Ag | Derivados de carbamato de quinuclidina y su uso como antagonistas m3. |
EA006505B1 (ru) * | 2001-12-20 | 2005-12-29 | Лабораториос С.А.Л.В.А.Т.,С.А. | Производные карбамата 1-алкил-1-азониабицикло[2.2.2]октана и их применение в качестве антагонистов мускаринового рецептора |
-
2001
- 2001-06-25 UA UA2003010718A patent/UA72632C2/uk unknown
- 2001-06-25 AU AU6610001A patent/AU6610001A/xx not_active Withdrawn
- 2001-06-25 WO PCT/ES2001/000252 patent/WO2002000652A1/es active IP Right Grant
- 2001-06-25 AP APAP/P/2003/002722A patent/AP1420A/en active
- 2001-06-25 PT PT01943553T patent/PT1300407E/pt unknown
- 2001-06-25 ES ES01943553T patent/ES2213703T5/es not_active Expired - Lifetime
- 2001-06-25 CZ CZ2003261A patent/CZ294251B6/cs not_active IP Right Cessation
- 2001-06-25 TR TR2004/00420T patent/TR200400420T4/xx unknown
- 2001-06-25 US US10/312,227 patent/US6916828B2/en not_active Expired - Fee Related
- 2001-06-25 JP JP2002505776A patent/JP5046465B2/ja not_active Expired - Fee Related
- 2001-06-25 DK DK01943553.6T patent/DK1300407T4/da active
- 2001-06-25 BR BR0112297-5A patent/BR0112297A/pt active Search and Examination
- 2001-06-25 SI SI200130075T patent/SI1300407T2/sl unknown
- 2001-06-25 CA CA002414514A patent/CA2414514C/en not_active Expired - Fee Related
- 2001-06-25 PL PL359333A patent/PL201530B1/pl unknown
- 2001-06-25 HU HU0301414A patent/HU229306B1/hu not_active IP Right Cessation
- 2001-06-25 AU AU2001266100A patent/AU2001266100B9/en not_active Ceased
- 2001-06-25 OA OA1200200393A patent/OA12300A/en unknown
- 2001-06-25 DE DE20122417U patent/DE20122417U1/de not_active Expired - Lifetime
- 2001-06-25 AT AT01943553T patent/ATE260277T1/de active
- 2001-06-25 EA EA200300072A patent/EA005520B1/ru not_active IP Right Cessation
- 2001-06-25 DE DE60102160T patent/DE60102160T3/de not_active Expired - Lifetime
- 2001-06-25 EP EP01943553A patent/EP1300407B2/en not_active Expired - Lifetime
- 2001-06-25 IL IL15370701A patent/IL153707A0/xx not_active IP Right Cessation
- 2001-06-25 KR KR1020027017706A patent/KR100751981B1/ko not_active IP Right Cessation
- 2001-06-25 MX MXPA03000141A patent/MXPA03000141A/es active IP Right Grant
- 2001-06-25 CN CNB018148042A patent/CN1227251C/zh not_active Expired - Fee Related
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2002
- 2002-12-23 NO NO20026211A patent/NO328499B1/no not_active IP Right Cessation
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2003
- 2003-01-17 BG BG107474A patent/BG66102B1/bg unknown
- 2003-01-20 CR CR6889A patent/CR6889A/es not_active Application Discontinuation
- 2003-01-23 ZA ZA200300644A patent/ZA200300644B/en unknown
- 2003-10-06 HK HK03107175A patent/HK1054934A1/xx not_active IP Right Cessation
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2004
- 2004-06-23 US US10/875,592 patent/US7115629B2/en not_active Expired - Fee Related
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