NO326546B1 - Pyridinderivater, fremgangsmate for fremstilling derav samt farmasoytisk preparat omfattende en slik forbindelse - Google Patents
Pyridinderivater, fremgangsmate for fremstilling derav samt farmasoytisk preparat omfattende en slik forbindelse Download PDFInfo
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- NO326546B1 NO326546B1 NO20034122A NO20034122A NO326546B1 NO 326546 B1 NO326546 B1 NO 326546B1 NO 20034122 A NO20034122 A NO 20034122A NO 20034122 A NO20034122 A NO 20034122A NO 326546 B1 NO326546 B1 NO 326546B1
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- Prior art keywords
- compound
- hydrogen
- formula
- phenyl
- chlorophenyl
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0107505A GB0107505D0 (en) | 2001-03-26 | 2001-03-26 | Organic compounds |
| US33828101P | 2001-12-06 | 2001-12-06 | |
| PCT/EP2002/003332 WO2002076946A2 (en) | 2001-03-26 | 2002-03-25 | Fused pyridine derivatives for use as vanilloid receptor antagonists for treating pain. |
Publications (3)
| Publication Number | Publication Date |
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| NO20034122D0 NO20034122D0 (no) | 2003-09-16 |
| NO20034122L NO20034122L (no) | 2003-09-16 |
| NO326546B1 true NO326546B1 (no) | 2009-01-05 |
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| NO20034122A NO326546B1 (no) | 2001-03-26 | 2003-09-16 | Pyridinderivater, fremgangsmate for fremstilling derav samt farmasoytisk preparat omfattende en slik forbindelse |
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| Country | Link |
|---|---|
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| EP (1) | EP1377576A2 (es) |
| JP (1) | JP4205430B2 (es) |
| KR (1) | KR20030083755A (es) |
| CN (1) | CN1500089A (es) |
| BR (1) | BR0208338A (es) |
| CA (1) | CA2441599A1 (es) |
| CZ (1) | CZ20032561A3 (es) |
| HU (1) | HUP0303623A2 (es) |
| IL (1) | IL157815A0 (es) |
| MX (1) | MXPA03008754A (es) |
| NO (1) | NO326546B1 (es) |
| PE (1) | PE20021161A1 (es) |
| PL (1) | PL363907A1 (es) |
| RU (1) | RU2003130221A (es) |
| SK (1) | SK11952003A3 (es) |
| WO (1) | WO2002076946A2 (es) |
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| JP2004506714A (ja) | 2000-08-21 | 2004-03-04 | パシフィック コーポレーション | 新規チオ尿素化合物及びこれを含有する薬学的組成物 |
| ATE393141T1 (de) | 2000-08-21 | 2008-05-15 | Pacific Corp | Neue thiourea-derivate und pharmazeutische zusammensetzungen die diese enthalten |
| KR20040085151A (ko) | 2002-01-17 | 2004-10-07 | 뉴로젠 코포레이션 | 캡사이신 조절자로서의 치환된 퀴나졸린-4-일 아민 유사체 |
| JP4583760B2 (ja) | 2002-02-01 | 2010-11-17 | ユーロ−セルティーク エス．エイ． | 疼痛の治療に有用な治療薬 |
| US6864261B2 (en) | 2002-05-02 | 2005-03-08 | Euro-Celtique S.A. | Therapeutic agents useful for treating pain |
| GB0229808D0 (en) * | 2002-12-20 | 2003-01-29 | Glaxo Group Ltd | Novel compositions |
| ATE450533T1 (de) * | 2003-02-14 | 2009-12-15 | Glaxo Group Ltd | Carboxamidderivate |
| ATE556067T1 (de) | 2003-05-20 | 2012-05-15 | Ajinomoto Kk | Modulatoren des vanilloid rezeptors |
| GB0319150D0 (en) | 2003-08-14 | 2003-09-17 | Glaxo Group Ltd | Novel compounds |
| US20070135454A1 (en) | 2003-11-14 | 2007-06-14 | Tracy Bayliss | Bicyclic pyrimidin-4(3h)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1-receptor(vr1) |
| GB0412769D0 (en) | 2004-06-08 | 2004-07-07 | Novartis Ag | Organic compounds |
| WO2006019965A2 (en) * | 2004-07-16 | 2006-02-23 | Takeda San Diego, Inc. | Dipeptidyl peptidase inhibitors |
| JP2008508190A (ja) | 2004-07-19 | 2008-03-21 | ノボ ノルディスク アクティーゼルスカブ | 肥満または肥満に関連する疾患および障害の治療におけるカプサイシン受容体の活性の阻害 |
| DE102004039373A1 (de) | 2004-08-12 | 2006-02-23 | Grünenthal GmbH | Para-Alkyl-substituierte N-(4-Hydroxy-3-methoxy-benzyl)-zimtsäureamide und deren Verwendung zur Herstellung von Arzneimitteln |
| KR20060087386A (ko) | 2005-01-28 | 2006-08-02 | 주식회사 대웅제약 | 신규 벤조이미다졸 유도체 및 이를 함유하는 약제학적조성물 |
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Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2749344A (en) * | 1953-01-02 | 1956-06-05 | Burroughs Wellcome Co | Pyrimidine compounds |
| US5958930A (en) * | 1991-04-08 | 1999-09-28 | Duquesne University Of The Holy Ghost | Pyrrolo pyrimidine and furo pyrimidine derivatives |
| US5620978A (en) | 1994-01-03 | 1997-04-15 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon, Eugene Oregon | 8-aza, 6-aza and 6,8-diaza-1,4-dihydroquinoxaline-2,3-diones and the use thereof as antagonists for the glycine/NMDA receptor |
| FR2750862B1 (fr) | 1996-07-12 | 1998-10-16 | Dupin Jean Pierre | Utilisation d'heterocycles diazotes fusionnes avec un systeme aromatique ou heteroaromatique pour le traitement des maladies thrombo-emboliques |
-
2002
- 2002-03-25 KR KR10-2003-7012460A patent/KR20030083755A/ko not_active Application Discontinuation
- 2002-03-25 PL PL02363907A patent/PL363907A1/xx not_active Application Discontinuation
- 2002-03-25 CZ CZ20032561A patent/CZ20032561A3/cs unknown
- 2002-03-25 CN CNA028073495A patent/CN1500089A/zh active Pending
- 2002-03-25 SK SK1195-2003A patent/SK11952003A3/sk unknown
- 2002-03-25 EP EP02730062A patent/EP1377576A2/en not_active Withdrawn
- 2002-03-25 IL IL15781502A patent/IL157815A0/xx unknown
- 2002-03-25 JP JP2002576207A patent/JP4205430B2/ja not_active Expired - Fee Related
- 2002-03-25 MX MXPA03008754A patent/MXPA03008754A/es not_active Application Discontinuation
- 2002-03-25 BR BR0208338-8A patent/BR0208338A/pt not_active IP Right Cessation
- 2002-03-25 RU RU2003130221/04A patent/RU2003130221A/ru not_active Application Discontinuation
- 2002-03-25 CA CA002441599A patent/CA2441599A1/en not_active Abandoned
- 2002-03-25 US US10/469,756 patent/US7915264B2/en not_active Expired - Fee Related
- 2002-03-25 HU HU0303623A patent/HUP0303623A2/hu unknown
- 2002-03-25 WO PCT/EP2002/003332 patent/WO2002076946A2/en not_active Application Discontinuation
- 2002-03-26 PE PE2002000241A patent/PE20021161A1/es not_active Application Discontinuation
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2003
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Also Published As
| Publication number | Publication date |
|---|---|
| JP4205430B2 (ja) | 2009-01-07 |
| SK11952003A3 (sk) | 2004-03-02 |
| HUP0303623A2 (hu) | 2004-03-01 |
| CA2441599A1 (en) | 2002-10-03 |
| PE20021161A1 (es) | 2003-02-21 |
| BR0208338A (pt) | 2004-03-09 |
| NO20034122D0 (no) | 2003-09-16 |
| CZ20032561A3 (cs) | 2003-12-17 |
| WO2002076946A3 (en) | 2002-12-27 |
| US7915264B2 (en) | 2011-03-29 |
| JP2004528312A (ja) | 2004-09-16 |
| RU2003130221A (ru) | 2005-04-10 |
| KR20030083755A (ko) | 2003-10-30 |
| CN1500089A (zh) | 2004-05-26 |
| US20040138454A1 (en) | 2004-07-15 |
| NO20034122L (no) | 2003-09-16 |
| MXPA03008754A (es) | 2004-02-18 |
| PL363907A1 (en) | 2004-11-29 |
| IL157815A0 (en) | 2004-03-28 |
| WO2002076946A2 (en) | 2002-10-03 |
| EP1377576A2 (en) | 2004-01-07 |
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