NO326375B1 - Vedvarende frigivelsesformuleringer av oksymorfon samt fast doseringsform inneholdende slike. - Google Patents
Vedvarende frigivelsesformuleringer av oksymorfon samt fast doseringsform inneholdende slike. Download PDFInfo
- Publication number
- NO326375B1 NO326375B1 NO20031019A NO20031019A NO326375B1 NO 326375 B1 NO326375 B1 NO 326375B1 NO 20031019 A NO20031019 A NO 20031019A NO 20031019 A NO20031019 A NO 20031019A NO 326375 B1 NO326375 B1 NO 326375B1
- Authority
- NO
- Norway
- Prior art keywords
- sustained release
- release formulation
- oxymorphone
- delivery system
- amount
- Prior art date
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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US32935201P | 2001-10-15 | 2001-10-15 | |
PCT/US2002/021403 WO2003004033A1 (en) | 2001-07-06 | 2002-07-03 | Sustained release formulations of oxymorphone |
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NO20031019D0 NO20031019D0 (no) | 2003-03-05 |
NO20031019L NO20031019L (no) | 2003-05-05 |
NO326375B1 true NO326375B1 (no) | 2008-11-17 |
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NO20031019A NO326375B1 (no) | 2001-07-06 | 2003-03-05 | Vedvarende frigivelsesformuleringer av oksymorfon samt fast doseringsform inneholdende slike. |
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US (3) | US20030129234A1 (pl) |
EP (2) | EP1404331B1 (pl) |
KR (1) | KR20030048026A (pl) |
AT (1) | ATE376832T1 (pl) |
BR (2) | BR0205722A (pl) |
DE (1) | DE60223254T2 (pl) |
DK (1) | DK1404331T3 (pl) |
ES (1) | ES2292775T3 (pl) |
HK (1) | HK1064921A1 (pl) |
NO (1) | NO326375B1 (pl) |
PL (2) | PL208484B1 (pl) |
WO (2) | WO2003004033A1 (pl) |
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US5478577A (en) * | 1993-11-23 | 1995-12-26 | Euroceltique, S.A. | Method of treating pain by administering 24 hour oral opioid formulations exhibiting rapid rate of initial rise of plasma drug level |
CN100356907C (zh) * | 2001-06-08 | 2007-12-26 | 恩德制药公司 | 利用丙烯酸酯聚合物的控释剂型和其制备方法 |
EP1404331B1 (en) * | 2001-07-06 | 2007-10-31 | Penwest Pharmaceuticals Co. | Sustained release formulations of oxymorphone |
US8329216B2 (en) * | 2001-07-06 | 2012-12-11 | Endo Pharmaceuticals Inc. | Oxymorphone controlled release formulations |
US20030130297A1 (en) * | 2001-07-06 | 2003-07-10 | Endo Pharmaceuticals, Inc. | Oral administration of 6-hydroxy-oxymorphone for use as an analgesic |
US20030068375A1 (en) | 2001-08-06 | 2003-04-10 | Curtis Wright | Pharmaceutical formulation containing gelling agent |
CA2459976A1 (en) * | 2001-09-26 | 2003-04-03 | Penwest Pharmaceuticals Company | Opioid formulations having reduced potential for abuse |
US7776314B2 (en) | 2002-06-17 | 2010-08-17 | Grunenthal Gmbh | Abuse-proofed dosage system |
US8557291B2 (en) | 2002-07-05 | 2013-10-15 | Collegium Pharmaceutical, Inc. | Abuse-deterrent pharmaceutical compositions of opioids and other drugs |
US10004729B2 (en) | 2002-07-05 | 2018-06-26 | Collegium Pharmaceutical, Inc. | Tamper-resistant pharmaceutical compositions of opioids and other drugs |
US8840928B2 (en) | 2002-07-05 | 2014-09-23 | Collegium Pharmaceutical, Inc. | Tamper-resistant pharmaceutical compositions of opioids and other drugs |
EP1594467A4 (en) | 2002-07-05 | 2008-10-22 | Collegium Pharmaceutical Inc | MISUSE OF PHARMACEUTICAL COMPOSITIONS OF OPIOIDES AND OTHER MEDICAMENTS |
EP1646367A4 (en) * | 2003-07-21 | 2011-06-15 | Nesher Solutions Ltd | ORAL DOSAGE FORMS WITH CONTROLLED RELEASE ON GELLAN RUBBER BASE A NEW PLATFORM TECHNOLOGY FOR MAGNETIC RETENTION |
DE102005005446A1 (de) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Bruchfeste Darreichungsformen mit retardierter Freisetzung |
DE10361596A1 (de) | 2003-12-24 | 2005-09-29 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform |
DE10336400A1 (de) | 2003-08-06 | 2005-03-24 | Grünenthal GmbH | Gegen Missbrauch gesicherte Darreichungsform |
US20070048228A1 (en) | 2003-08-06 | 2007-03-01 | Elisabeth Arkenau-Maric | Abuse-proofed dosage form |
EP1765292B1 (en) | 2004-06-12 | 2017-10-04 | Collegium Pharmaceutical, Inc. | Abuse-deterrent drug formulations |
DE102004032049A1 (de) | 2004-07-01 | 2006-01-19 | Grünenthal GmbH | Gegen Missbrauch gesicherte, orale Darreichungsform |
DE102005005449A1 (de) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform |
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- 2002-07-03 KR KR10-2003-7003334A patent/KR20030048026A/ko not_active Application Discontinuation
- 2002-07-03 ES ES02744835T patent/ES2292775T3/es not_active Expired - Lifetime
- 2002-07-03 EP EP02748085A patent/EP1404332A1/en not_active Withdrawn
- 2002-07-03 AT AT02744835T patent/ATE376832T1/de active
- 2002-07-03 WO PCT/US2002/021354 patent/WO2003004029A1/en not_active Application Discontinuation
-
2003
- 2003-03-05 NO NO20031019A patent/NO326375B1/no not_active IP Right Cessation
-
2004
- 2004-09-23 HK HK04107358A patent/HK1064921A1/xx not_active IP Right Cessation
-
2007
- 2007-08-13 US US11/891,775 patent/US20080050431A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
PL207748B1 (pl) | 2011-01-31 |
BR0210855A (pt) | 2006-10-24 |
ATE376832T1 (de) | 2007-11-15 |
KR20030048026A (ko) | 2003-06-18 |
US7276250B2 (en) | 2007-10-02 |
US20030129234A1 (en) | 2003-07-10 |
WO2003004033A1 (en) | 2003-01-16 |
US20030129230A1 (en) | 2003-07-10 |
DK1404331T3 (da) | 2008-01-28 |
HK1064921A1 (en) | 2005-02-08 |
DE60223254D1 (de) | 2007-12-13 |
PL366430A1 (pl) | 2005-01-24 |
NO20031019D0 (no) | 2003-03-05 |
BR0205722A (pt) | 2005-04-05 |
EP1404331A1 (en) | 2004-04-07 |
ES2292775T3 (es) | 2008-03-16 |
US20080050431A1 (en) | 2008-02-28 |
EP1404332A1 (en) | 2004-04-07 |
NO20031019L (no) | 2003-05-05 |
WO2003004029A1 (en) | 2003-01-16 |
PL208484B1 (pl) | 2011-05-31 |
DE60223254T2 (de) | 2008-08-14 |
PL367277A1 (pl) | 2005-02-21 |
EP1404331B1 (en) | 2007-10-31 |
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Legal Events
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MM1K | Lapsed by not paying the annual fees |