NO320844B1 - Celecoxibpreparat, fremgangsmate for fremstilling av dette og av farmasoytisk preparat som omfatter det og anvendelse av celeboxibpreparatet for fremstilling av preparat og medikament. - Google Patents
Celecoxibpreparat, fremgangsmate for fremstilling av dette og av farmasoytisk preparat som omfatter det og anvendelse av celeboxibpreparatet for fremstilling av preparat og medikament. Download PDFInfo
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- NO320844B1 NO320844B1 NO20013855A NO20013855A NO320844B1 NO 320844 B1 NO320844 B1 NO 320844B1 NO 20013855 A NO20013855 A NO 20013855A NO 20013855 A NO20013855 A NO 20013855A NO 320844 B1 NO320844 B1 NO 320844B1
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/58—One oxygen atom, e.g. butenolide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurosurgery (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Virology (AREA)
- Endocrinology (AREA)
- Ophthalmology & Optometry (AREA)
- Diabetes (AREA)
- Molecular Biology (AREA)
- Urology & Nephrology (AREA)
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US16985699P | 1999-12-08 | 1999-12-08 | |
PCT/US2000/032435 WO2001042221A1 (en) | 1999-12-08 | 2000-12-06 | Solid-state form of celecoxib having enhanced bioavailability |
US09/730,663 US6964978B2 (en) | 1999-12-08 | 2000-12-06 | Solid-state form of celecoxib having enhanced bioavailability |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20013855D0 NO20013855D0 (no) | 2001-08-08 |
NO20013855L NO20013855L (no) | 2001-10-05 |
NO320844B1 true NO320844B1 (no) | 2006-02-06 |
Family
ID=26865450
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20013855A NO320844B1 (no) | 1999-12-08 | 2001-08-08 | Celecoxibpreparat, fremgangsmate for fremstilling av dette og av farmasoytisk preparat som omfatter det og anvendelse av celeboxibpreparatet for fremstilling av preparat og medikament. |
Country Status (20)
Country | Link |
---|---|
US (3) | US6964978B2 (de) |
EP (1) | EP1150959B1 (de) |
JP (1) | JP2004500358A (de) |
CN (1) | CN1376146B (de) |
AT (1) | ATE387431T1 (de) |
AU (1) | AU784572B2 (de) |
BR (1) | BR0008058A (de) |
CA (1) | CA2362673A1 (de) |
CY (1) | CY1107389T1 (de) |
DE (1) | DE60038162T2 (de) |
DK (1) | DK1150959T3 (de) |
EA (1) | EA003612B1 (de) |
ES (1) | ES2299441T3 (de) |
HU (1) | HUP0201450A3 (de) |
IL (2) | IL144761A0 (de) |
NO (1) | NO320844B1 (de) |
NZ (1) | NZ513964A (de) |
PL (1) | PL203262B1 (de) |
SK (1) | SK12682001A3 (de) |
WO (1) | WO2001042221A1 (de) |
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NZ513964A (en) * | 1999-12-08 | 2004-01-30 | Pharmacia Corp | Solid-state form of celecoxib having enhanced bioavailability |
EP1712222A3 (de) | 1999-12-23 | 2012-06-20 | Pfizer Products Inc. | Arzneizusammensetzung mit erhöhter Arzneistoffkonzentration |
US6589557B2 (en) | 2000-06-15 | 2003-07-08 | Acusphere, Inc. | Porous celecoxib matrices and methods of manufacture thereof |
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TWI256305B (en) * | 2000-08-18 | 2006-06-11 | Pharmacia Corp | Oral fast-melt pharmaceutical composition of a cyclooxygenase-2 inhibitor and process for preparing the same |
BR0210518A (pt) | 2001-06-22 | 2004-06-22 | Pfizer Prod Inc | Composições farmacêuticas de dispersões de drogas e polìmeros neutros |
EP1469832B2 (de) | 2002-02-01 | 2016-10-26 | Bend Research, Inc. | Pharmazeutische zusammensetzungen amorpher dispersionen von wirkstoffen und lipophiler mikrophasenbildender materialien |
US20100311701A1 (en) * | 2002-02-15 | 2010-12-09 | Transform Pharmaceuticals, Inc | Pharmaceutical Co-Crystal Compositions |
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AU2003267231A1 (en) * | 2002-09-20 | 2004-04-08 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions with improved dissolution |
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EP2339328A3 (de) | 2002-12-30 | 2011-07-13 | Transform Pharmaceuticals, Inc. | Pharmazeutische kokristallisierte Celecoxib-Zusammensetzungen |
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US20070060629A1 (en) * | 2003-10-17 | 2007-03-15 | Yasuhiro Imanishi | Large conductance calcium-activated k channel opener |
CA2551254A1 (en) * | 2003-12-31 | 2005-07-21 | Pfizer Products Inc. | Stabilized pharmaceutical solid compositions of low-solubility drugs, poloxamers, and stabilizing polymers |
WO2005065657A2 (en) * | 2003-12-31 | 2005-07-21 | Pfizer Products Inc. | Solid compositions of low-solubility drugs and poloxamers |
FR2879075B1 (fr) * | 2004-12-15 | 2007-01-19 | Adisseo France Sas Soc Par Act | Procede de preparation de granules de principe actif hydrophile par extrusion |
FR2881049B1 (fr) * | 2005-01-24 | 2008-12-26 | Vetoquinol Sa Sa | Medicament destine a etre administre par voie orale comprenant un inhibiteur de la cyclo-oxygenase-2, et son procede de preparation |
ATE480229T1 (de) * | 2005-05-24 | 2010-09-15 | Flamel Tech Sa | Orale pharmazeutische zusammensetzung zur behandlung einer cox-2-vermittelten erkrankung |
CA2671200A1 (en) * | 2006-07-21 | 2008-01-24 | Lab International Srl | Hydrophilic abuse deterrent delivery system |
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WO2008085674A1 (en) * | 2007-01-04 | 2008-07-17 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions comprising celecoxib co-crystals |
US20100233272A1 (en) * | 2007-11-15 | 2010-09-16 | Leah Elizabeth Appel | Dosage forms comprising celecoxib providing both rapid and sustained pain relief |
EP2105130A1 (de) * | 2008-03-25 | 2009-09-30 | Ratiopharm GmbH | Pharmazeutische Formulierung und Verfahren zu deren Herstellung |
EP2133068A1 (de) * | 2008-06-13 | 2009-12-16 | Ratiopharm GmbH | Verfahren zur Auswahl eines geeigneten Hilfsstoffs für die Herstellung von festen Dispersionen für pharmazeutische Formulierungen |
CN102238941A (zh) * | 2008-09-17 | 2011-11-09 | 迈兰实验室公司 | 颗粒、制备它们的方法和包含它们的药物产品 |
EP2442794A1 (de) * | 2009-06-19 | 2012-04-25 | Nanoform Hungary Ltd. | Nanopartikelförmige telmisartanzusammensetzungen und verfahren für ihre herstellung |
WO2010150144A2 (en) | 2009-06-25 | 2010-12-29 | Wockhardt Research Centre | Low dose pharmaceutical compositions of celecoxib |
WO2011055233A2 (en) | 2009-11-03 | 2011-05-12 | Actavis Group Ptc Ehf | Improved process for preparing celecoxib polymorph |
US20110213159A1 (en) * | 2010-03-01 | 2011-09-01 | Vamsee Krishna Muppidi | Process for preparation of celecoxib crystalline form |
CN102764264A (zh) * | 2012-07-25 | 2012-11-07 | 杭州和泽医药科技有限公司 | 一种具高溶出度的塞来昔布固体组合物、制备方法及应用 |
CN103655478A (zh) * | 2012-09-26 | 2014-03-26 | 北京星昊医药股份有限公司 | 一种塞来昔布固体分散体及其制备方法和应用 |
EP2919767B1 (de) * | 2012-11-14 | 2020-04-01 | Abon Pharmaceuticals, LLC | System zur transmukosalen verabreichung von arzneimitteln |
WO2015016256A1 (ja) * | 2013-07-30 | 2015-02-05 | ライオン株式会社 | 錠剤 |
US10493089B2 (en) * | 2014-04-03 | 2019-12-03 | Sandoz Ag | Solid composition comprising amorphous sofosbuvir |
CN114209707A (zh) * | 2015-05-28 | 2022-03-22 | 瑞迪博士实验室有限公司 | 用于治疗疼痛的塞来昔布口服组合物 |
CA2999215A1 (en) * | 2015-10-07 | 2017-04-13 | Sandoz Ag | Solid pharmaceutical composition comprising amorphous sofosbuvir |
HUP1500618A2 (en) | 2015-12-16 | 2017-06-28 | Druggability Tech Ip Holdco Ltd | Complexes of celecoxib and its salts and derivatives, process for the preparation thereof and pharmaceutical composition containing them |
WO2018031577A1 (en) * | 2016-08-09 | 2018-02-15 | Autotelic Llc | Fixed dose combination for pain relief without edema |
US10736905B1 (en) | 2016-09-09 | 2020-08-11 | Shahin Fatholahi | Nefopam dosage forms and methods of treatment |
KR102002906B1 (ko) * | 2016-10-18 | 2019-07-23 | 경동제약 주식회사 | 셀레콕시브를 포함하는 정제 |
AU2017376257A1 (en) * | 2016-12-14 | 2019-06-13 | Druggability Technologies Ip Holdco Limited | Pharmaceutical composition containing celecoxib |
US11446311B2 (en) | 2017-09-08 | 2022-09-20 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
US10736874B1 (en) | 2017-09-08 | 2020-08-11 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
WO2020214791A1 (en) * | 2019-04-18 | 2020-10-22 | Nangenex Nanotechnology Incorporated | Celecoxib compositions and methods for their use |
CN111505058A (zh) * | 2020-03-05 | 2020-08-07 | 艾普康(香港)有限公司 | 乳房炎检测分析仪 |
CN112358492B (zh) * | 2020-11-13 | 2022-04-15 | 兰州大学 | 碳硼烷基塞来昔布及其制备和在头颈癌硼中子俘获治疗药物中的应用 |
KR102459968B1 (ko) * | 2022-01-21 | 2022-10-27 | 주식회사 큐어팜텍 | 기능성 약물이 함유된 생분해성 수지 제조방법 및 이에 의해 제조된 생분해성 수지 |
CN116942630B (zh) * | 2023-09-19 | 2023-12-26 | 北京福元医药股份有限公司 | 一种塞来昔布胶囊剂及其制备方法 |
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WO1998019708A2 (en) | 1996-11-04 | 1998-05-14 | Union Carbide Chemicals & Plastics Technology Corporation | Method for enhancing the solubility of substantially water-insoluble compounds |
KR100187959B1 (ko) * | 1997-03-31 | 1999-06-01 | 윤재승 | 저융점 무정형 세푸록심 악세틸의 제조방법 |
SE9802333D0 (sv) * | 1998-06-29 | 1998-06-29 | Astra Pharma Prod | Novel combination |
EP1126841B1 (de) * | 1998-11-02 | 2004-12-15 | Merck & Co., Inc. | Zusammensetzungen aus einem 5ht1b/1d agonisten und einem selektiven cox-2 hemmer zur behandlung von migräne |
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CA2360354A1 (en) | 1999-01-14 | 2000-07-20 | Sophie-Dorothee Clas | Synthesis of 4-[(5-substituted or unsubstituted phenyl)-3-substituted-1h-pyrazol-1-yl] benzenesulfonamides |
AU4308300A (en) | 1999-05-03 | 2000-11-17 | Dr. Reddy's Research Foundation | Pyrazoles having antiinflammatory activity |
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GB9920558D0 (en) | 1999-08-31 | 1999-11-03 | Bradford Particle Design Ltd | Methods for particle formation and their products |
NZ513964A (en) * | 1999-12-08 | 2004-01-30 | Pharmacia Corp | Solid-state form of celecoxib having enhanced bioavailability |
WO2004041243A2 (en) * | 2002-05-13 | 2004-05-21 | Pharmacia Corporation | Stable amorphous celecoxib composite and process therefor |
-
2000
- 2000-12-06 NZ NZ513964A patent/NZ513964A/xx not_active IP Right Cessation
- 2000-12-06 EP EP00982255A patent/EP1150959B1/de not_active Revoked
- 2000-12-06 DK DK00982255T patent/DK1150959T3/da active
- 2000-12-06 SK SK1268-2001A patent/SK12682001A3/sk not_active Application Discontinuation
- 2000-12-06 AT AT00982255T patent/ATE387431T1/de active
- 2000-12-06 HU HU0201450A patent/HUP0201450A3/hu unknown
- 2000-12-06 CA CA002362673A patent/CA2362673A1/en not_active Abandoned
- 2000-12-06 BR BR0008058-6A patent/BR0008058A/pt not_active Application Discontinuation
- 2000-12-06 IL IL14476100A patent/IL144761A0/xx active IP Right Grant
- 2000-12-06 US US09/730,663 patent/US6964978B2/en not_active Expired - Lifetime
- 2000-12-06 DE DE60038162T patent/DE60038162T2/de not_active Expired - Lifetime
- 2000-12-06 WO PCT/US2000/032435 patent/WO2001042221A1/en active IP Right Grant
- 2000-12-06 EA EA200100873A patent/EA003612B1/ru not_active IP Right Cessation
- 2000-12-06 PL PL349223A patent/PL203262B1/pl not_active IP Right Cessation
- 2000-12-06 CN CN008056358A patent/CN1376146B/zh not_active Expired - Fee Related
- 2000-12-06 ES ES00982255T patent/ES2299441T3/es not_active Expired - Lifetime
- 2000-12-06 JP JP2001543522A patent/JP2004500358A/ja active Pending
- 2000-12-06 AU AU19311/01A patent/AU784572B2/en not_active Ceased
-
2001
- 2001-08-06 IL IL144761A patent/IL144761A/en unknown
- 2001-08-08 NO NO20013855A patent/NO320844B1/no not_active IP Right Cessation
-
2005
- 2005-07-26 US US11/189,659 patent/US7220867B2/en not_active Expired - Lifetime
-
2007
- 2007-05-04 US US11/744,603 patent/US20070202160A1/en not_active Abandoned
-
2008
- 2008-04-10 CY CY20081100393T patent/CY1107389T1/el unknown
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DK1150959T3 (da) | 2008-06-02 |
AU1931101A (en) | 2001-06-18 |
HUP0201450A3 (en) | 2003-02-28 |
US20070202160A1 (en) | 2007-08-30 |
DE60038162T2 (de) | 2009-02-26 |
PL349223A1 (en) | 2002-07-01 |
IL144761A (en) | 2007-07-24 |
WO2001042221A1 (en) | 2001-06-14 |
EA200100873A1 (ru) | 2002-02-28 |
EA003612B1 (ru) | 2003-06-26 |
PL203262B1 (pl) | 2009-09-30 |
AU784572B2 (en) | 2006-05-04 |
BR0008058A (pt) | 2002-03-26 |
HUP0201450A2 (hu) | 2002-12-28 |
US7220867B2 (en) | 2007-05-22 |
US20050267190A1 (en) | 2005-12-01 |
CN1376146B (zh) | 2011-04-06 |
NZ513964A (en) | 2004-01-30 |
US20020006951A1 (en) | 2002-01-17 |
US6964978B2 (en) | 2005-11-15 |
ES2299441T3 (es) | 2008-06-01 |
EP1150959A1 (de) | 2001-11-07 |
NO20013855L (no) | 2001-10-05 |
DE60038162D1 (de) | 2008-04-10 |
CA2362673A1 (en) | 2001-06-14 |
ATE387431T1 (de) | 2008-03-15 |
CN1376146A (zh) | 2002-10-23 |
NO20013855D0 (no) | 2001-08-08 |
IL144761A0 (en) | 2002-08-14 |
EP1150959B1 (de) | 2008-02-27 |
CY1107389T1 (el) | 2012-12-19 |
JP2004500358A (ja) | 2004-01-08 |
SK12682001A3 (sk) | 2002-07-02 |
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