NO20090457L - Oksazolidon derivativer som PR modulatorer - Google Patents

Oksazolidon derivativer som PR modulatorer

Info

Publication number
NO20090457L
NO20090457L NO20090457A NO20090457A NO20090457L NO 20090457 L NO20090457 L NO 20090457L NO 20090457 A NO20090457 A NO 20090457A NO 20090457 A NO20090457 A NO 20090457A NO 20090457 L NO20090457 L NO 20090457L
Authority
NO
Norway
Prior art keywords
hormone
compounds
treatment
modulators
intake
Prior art date
Application number
NO20090457A
Other languages
English (en)
Norwegian (no)
Inventor
Andrew Fensome
Ronald Charles Bernotas
Casey Cameron Mccomas
Michael Anthony Marella
Gavin David Heffernan
Edward George Melenski
Thomas Joseph Commons
Jr Richard Page Woodworth
Michael Byron Webb
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NO20090457L publication Critical patent/NO20090457L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/48Nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/06Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing isoquinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20090457A 2006-08-15 2009-01-29 Oksazolidon derivativer som PR modulatorer NO20090457L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83789806P 2006-08-15 2006-08-15
PCT/US2007/017931 WO2008021331A2 (en) 2006-08-15 2007-08-13 Oxazolidone derivatives as pr modulators

Publications (1)

Publication Number Publication Date
NO20090457L true NO20090457L (no) 2009-04-27

Family

ID=39082681

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090457A NO20090457L (no) 2006-08-15 2009-01-29 Oksazolidon derivativer som PR modulatorer

Country Status (22)

Country Link
US (1) US7618990B2 (es)
EP (1) EP2054410A2 (es)
JP (1) JP2010500409A (es)
KR (1) KR20090039774A (es)
CN (1) CN101501031B (es)
AR (1) AR062327A1 (es)
AU (1) AU2007284599B2 (es)
BR (1) BRPI0716622A2 (es)
CA (1) CA2659208A1 (es)
CR (1) CR10617A (es)
GT (1) GT200900032A (es)
IL (1) IL196886A0 (es)
MX (1) MX2009001698A (es)
NO (1) NO20090457L (es)
NZ (1) NZ574753A (es)
PE (1) PE20070753A1 (es)
RU (1) RU2009105113A (es)
SA (1) SA07280440B1 (es)
SV (1) SV2009003168A (es)
TW (1) TW200815428A (es)
WO (1) WO2008021331A2 (es)
ZA (1) ZA200901055B (es)

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* Cited by examiner, † Cited by third party
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WO2008112495A1 (en) * 2007-03-09 2008-09-18 Wyeth Synthesis and characterization of polymorph form iii of 4-(2,(4,4-dimethyl-2-oxooxazolidin-3-yl)thiazol-4-yl)benzonitrile
PE20081803A1 (es) * 2007-03-09 2008-12-11 Wyeth Corp Sintesis y caracterizacion de la forma ii polimorfica de 4-(2-(4,4-dimetil-2-oxooxazolidin-3-il)tiazol-4-il)benzonitrilo
CN101525310B (zh) * 2009-04-21 2019-04-16 大连九信精细化工有限公司 1-苯甲酰基-3-(2-羟基-1,1-二甲基乙基)硫脲的合成方法
AU2011312490B2 (en) * 2010-09-28 2015-06-25 Radius Pharmaceuticals, Inc. Selective androgen receptor modulators
US9120818B2 (en) * 2010-12-14 2015-09-01 Merck Sharp & Dohme Corp. Process and intermediates for preparing macrolactams
JP6663866B2 (ja) * 2014-07-03 2020-03-13 セルジーン クオンティセル リサーチ,インク. リジン特異的なデメチラーゼ−1の阻害剤

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Also Published As

Publication number Publication date
US7618990B2 (en) 2009-11-17
KR20090039774A (ko) 2009-04-22
SA07280440B1 (ar) 2010-10-20
PE20070753A1 (es) 2008-08-14
IL196886A0 (en) 2009-11-18
GT200900032A (es) 2011-03-29
AU2007284599B2 (en) 2011-07-21
RU2009105113A (ru) 2010-09-27
AU2007284599A1 (en) 2008-02-21
EP2054410A2 (en) 2009-05-06
CN101501031B (zh) 2012-02-01
WO2008021331A3 (en) 2008-05-22
TW200815428A (en) 2008-04-01
US20080045556A1 (en) 2008-02-21
JP2010500409A (ja) 2010-01-07
ZA200901055B (en) 2009-12-30
CA2659208A1 (en) 2008-02-21
WO2008021331A2 (en) 2008-02-21
AR062327A1 (es) 2008-10-29
CR10617A (es) 2009-03-12
CN101501031A (zh) 2009-08-05
NZ574753A (en) 2011-04-29
MX2009001698A (es) 2009-02-25
SV2009003168A (es) 2010-01-14
BRPI0716622A2 (pt) 2013-10-08

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