NO20080468L - Diazepinokinoliner, synteser av disse samt intermediater - Google Patents
Diazepinokinoliner, synteser av disse samt intermediaterInfo
- Publication number
- NO20080468L NO20080468L NO20080468A NO20080468A NO20080468L NO 20080468 L NO20080468 L NO 20080468L NO 20080468 A NO20080468 A NO 20080468A NO 20080468 A NO20080468 A NO 20080468A NO 20080468 L NO20080468 L NO 20080468L
- Authority
- NO
- Norway
- Prior art keywords
- intermediates
- diazepinoquinolines
- syntheses
- agonists
- synthesis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Hematology (AREA)
- Addiction (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Diabetes (AREA)
- Pregnancy & Childbirth (AREA)
- Child & Adolescent Psychology (AREA)
- Obesity (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Foreliggende oppfinnelse angår metoder for syntese av forbindelser med formel (I) som er anvendelige som 5HT2C-agonister eller partielle agonister, derivater derav og mellomprodukter dertil.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70250905P | 2005-07-26 | 2005-07-26 | |
PCT/US2006/028655 WO2007016029A2 (en) | 2005-07-26 | 2006-07-24 | Diazepinoquinolines, synthesis thereof, and intermediates thereto |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20080468L true NO20080468L (no) | 2008-02-22 |
Family
ID=37603396
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20080468A NO20080468L (no) | 2005-07-26 | 2008-01-25 | Diazepinokinoliner, synteser av disse samt intermediater |
Country Status (20)
Country | Link |
---|---|
US (1) | US7671196B2 (no) |
EP (1) | EP1907390A2 (no) |
JP (1) | JP2009502925A (no) |
KR (1) | KR20080030682A (no) |
CN (1) | CN101268076A (no) |
AR (1) | AR054849A1 (no) |
AU (1) | AU2006276010A1 (no) |
BR (1) | BRPI0614154A2 (no) |
CA (1) | CA2616161A1 (no) |
CR (1) | CR9670A (no) |
EC (1) | ECSP088151A (no) |
GT (1) | GT200600326A (no) |
IL (1) | IL188896A0 (no) |
MX (1) | MX2008001030A (no) |
NO (1) | NO20080468L (no) |
PE (1) | PE20070238A1 (no) |
RU (1) | RU2008102884A (no) |
SA (1) | SA06270241B1 (no) |
TW (1) | TW200738713A (no) |
WO (1) | WO2007016029A2 (no) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GT200500317A (es) * | 2004-11-05 | 2006-10-27 | Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos | |
AR054849A1 (es) | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
AR060088A1 (es) * | 2006-03-24 | 2008-05-21 | Wyeth Corp | Metodos para tratar trastornos cognitivos y otros afines |
CA2644662A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | New therapeutic combinations for the treatment of depression |
EP1998782A2 (en) * | 2006-03-24 | 2008-12-10 | Wyeth a Corporation of the State of Delaware | Methods for modulating bladder function |
WO2007112000A2 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | Treatment of pain |
CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
CN103204858A (zh) * | 2013-03-20 | 2013-07-17 | 广州科瑞生物技术有限公司 | 基于酒石酸拆分合成工艺制备新型手性抗焦虑症药物 |
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AR051946A1 (es) * | 2004-11-05 | 2007-02-21 | Wyeth Corp | Formulaciones de derivados de [1,4] diazepina [6,7,1-ij] quinolina |
EP1714963A1 (en) | 2005-04-19 | 2006-10-25 | IPCA Laboratories Limited | Process for the Preparation of Valsartan and its Intermediates |
AR054849A1 (es) | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
AR056695A1 (es) * | 2005-10-17 | 2007-10-17 | Wyeth Corp | Tetrahidroquinolinas, su sintesis e intermediarios |
TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
CA2644639A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | New therapeutic combinations for the treatment or prevention of psychotic disorders |
EP1998782A2 (en) * | 2006-03-24 | 2008-12-10 | Wyeth a Corporation of the State of Delaware | Methods for modulating bladder function |
CA2644662A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | New therapeutic combinations for the treatment of depression |
AR060088A1 (es) * | 2006-03-24 | 2008-05-21 | Wyeth Corp | Metodos para tratar trastornos cognitivos y otros afines |
WO2007112000A2 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | Treatment of pain |
CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
-
2006
- 2006-07-19 AR ARP060103086A patent/AR054849A1/es unknown
- 2006-07-24 RU RU2008102884/04A patent/RU2008102884A/ru not_active Application Discontinuation
- 2006-07-24 CN CNA2006800341809A patent/CN101268076A/zh active Pending
- 2006-07-24 WO PCT/US2006/028655 patent/WO2007016029A2/en active Application Filing
- 2006-07-24 BR BRPI0614154-4A patent/BRPI0614154A2/pt not_active Application Discontinuation
- 2006-07-24 PE PE2006000891A patent/PE20070238A1/es not_active Application Discontinuation
- 2006-07-24 CA CA002616161A patent/CA2616161A1/en not_active Abandoned
- 2006-07-24 JP JP2008524026A patent/JP2009502925A/ja not_active Withdrawn
- 2006-07-24 AU AU2006276010A patent/AU2006276010A1/en not_active Abandoned
- 2006-07-24 US US11/491,590 patent/US7671196B2/en not_active Expired - Fee Related
- 2006-07-24 MX MX2008001030A patent/MX2008001030A/es not_active Application Discontinuation
- 2006-07-24 GT GT200600326A patent/GT200600326A/es unknown
- 2006-07-24 KR KR1020087004478A patent/KR20080030682A/ko not_active Application Discontinuation
- 2006-07-24 TW TW095126932A patent/TW200738713A/zh unknown
- 2006-07-24 EP EP06788294A patent/EP1907390A2/en not_active Withdrawn
- 2006-07-26 SA SA06270241A patent/SA06270241B1/ar unknown
-
2008
- 2008-01-17 CR CR9670A patent/CR9670A/es not_active Application Discontinuation
- 2008-01-21 IL IL188896A patent/IL188896A0/en unknown
- 2008-01-25 NO NO20080468A patent/NO20080468L/no not_active Application Discontinuation
- 2008-01-30 EC EC2008008151A patent/ECSP088151A/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP1907390A2 (en) | 2008-04-09 |
AR054849A1 (es) | 2007-07-18 |
GT200600326A (es) | 2007-03-14 |
CA2616161A1 (en) | 2007-02-08 |
KR20080030682A (ko) | 2008-04-04 |
JP2009502925A (ja) | 2009-01-29 |
CR9670A (es) | 2008-07-29 |
PE20070238A1 (es) | 2007-03-26 |
WO2007016029A3 (en) | 2007-05-18 |
RU2008102884A (ru) | 2009-09-10 |
TW200738713A (en) | 2007-10-16 |
CN101268076A (zh) | 2008-09-17 |
ECSP088151A (es) | 2008-02-20 |
BRPI0614154A2 (pt) | 2011-03-15 |
SA06270241B1 (ar) | 2009-09-02 |
US20070027142A1 (en) | 2007-02-01 |
AU2006276010A1 (en) | 2007-02-08 |
US7671196B2 (en) | 2010-03-02 |
WO2007016029A2 (en) | 2007-02-08 |
IL188896A0 (en) | 2008-04-13 |
MX2008001030A (es) | 2008-03-19 |
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