ECSP088151A - Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas - Google Patents
Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlasInfo
- Publication number
- ECSP088151A ECSP088151A EC2008008151A ECSP088151A ECSP088151A EC SP088151 A ECSP088151 A EC SP088151A EC 2008008151 A EC2008008151 A EC 2008008151A EC SP088151 A ECSP088151 A EC SP088151A EC SP088151 A ECSP088151 A EC SP088151A
- Authority
- EC
- Ecuador
- Prior art keywords
- diazepinoquinolinas
- intermediaries
- synthesis
- same
- agonists
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Anesthesiology (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pregnancy & Childbirth (AREA)
- Addiction (AREA)
- Hematology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a métodos para sintetizar compuestos útiles como agonistas o agonistas parciales de 5HT2C, derivados de los mismos, y a intermediarios para obtenerlos
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70250905P | 2005-07-26 | 2005-07-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP088151A true ECSP088151A (es) | 2008-02-20 |
Family
ID=37603396
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2008008151A ECSP088151A (es) | 2005-07-26 | 2008-01-30 | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
Country Status (20)
Country | Link |
---|---|
US (1) | US7671196B2 (es) |
EP (1) | EP1907390A2 (es) |
JP (1) | JP2009502925A (es) |
KR (1) | KR20080030682A (es) |
CN (1) | CN101268076A (es) |
AR (1) | AR054849A1 (es) |
AU (1) | AU2006276010A1 (es) |
BR (1) | BRPI0614154A2 (es) |
CA (1) | CA2616161A1 (es) |
CR (1) | CR9670A (es) |
EC (1) | ECSP088151A (es) |
GT (1) | GT200600326A (es) |
IL (1) | IL188896A0 (es) |
MX (1) | MX2008001030A (es) |
NO (1) | NO20080468L (es) |
PE (1) | PE20070238A1 (es) |
RU (1) | RU2008102884A (es) |
SA (1) | SA06270241B1 (es) |
TW (1) | TW200738713A (es) |
WO (1) | WO2007016029A2 (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GT200500317A (es) * | 2004-11-05 | 2006-10-27 | Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos | |
AR054849A1 (es) | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
CA2644656A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | Treatment of pain |
US20070225274A1 (en) * | 2006-03-24 | 2007-09-27 | Wyeth | Methods for modulating bladder function |
JP2009531435A (ja) * | 2006-03-24 | 2009-09-03 | ワイス | うつ病の治療用の新規な治療組み合わせ |
CL2007000773A1 (es) * | 2006-03-24 | 2008-01-25 | Wyeth Corp | Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd. |
CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
CN103204858A (zh) * | 2013-03-20 | 2013-07-17 | 广州科瑞生物技术有限公司 | 基于酒石酸拆分合成工艺制备新型手性抗焦虑症药物 |
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AR054849A1 (es) | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
AR056695A1 (es) * | 2005-10-17 | 2007-10-17 | Wyeth Corp | Tetrahidroquinolinas, su sintesis e intermediarios |
TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
BRPI0709129A2 (pt) * | 2006-03-24 | 2011-06-28 | Wyeth Corp | combinações terapêuticas para o tratamento ou prevenção de transtornos psicóticos |
CA2644656A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | Treatment of pain |
JP2009531435A (ja) * | 2006-03-24 | 2009-09-03 | ワイス | うつ病の治療用の新規な治療組み合わせ |
CL2007000773A1 (es) * | 2006-03-24 | 2008-01-25 | Wyeth Corp | Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd. |
US20070225274A1 (en) * | 2006-03-24 | 2007-09-27 | Wyeth | Methods for modulating bladder function |
CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
-
2006
- 2006-07-19 AR ARP060103086A patent/AR054849A1/es unknown
- 2006-07-24 GT GT200600326A patent/GT200600326A/es unknown
- 2006-07-24 WO PCT/US2006/028655 patent/WO2007016029A2/en active Application Filing
- 2006-07-24 PE PE2006000891A patent/PE20070238A1/es not_active Application Discontinuation
- 2006-07-24 US US11/491,590 patent/US7671196B2/en not_active Expired - Fee Related
- 2006-07-24 EP EP06788294A patent/EP1907390A2/en not_active Withdrawn
- 2006-07-24 MX MX2008001030A patent/MX2008001030A/es not_active Application Discontinuation
- 2006-07-24 AU AU2006276010A patent/AU2006276010A1/en not_active Abandoned
- 2006-07-24 CA CA002616161A patent/CA2616161A1/en not_active Abandoned
- 2006-07-24 BR BRPI0614154-4A patent/BRPI0614154A2/pt not_active Application Discontinuation
- 2006-07-24 CN CNA2006800341809A patent/CN101268076A/zh active Pending
- 2006-07-24 TW TW095126932A patent/TW200738713A/zh unknown
- 2006-07-24 JP JP2008524026A patent/JP2009502925A/ja not_active Withdrawn
- 2006-07-24 RU RU2008102884/04A patent/RU2008102884A/ru not_active Application Discontinuation
- 2006-07-24 KR KR1020087004478A patent/KR20080030682A/ko not_active Application Discontinuation
- 2006-07-26 SA SA06270241A patent/SA06270241B1/ar unknown
-
2008
- 2008-01-17 CR CR9670A patent/CR9670A/es not_active Application Discontinuation
- 2008-01-21 IL IL188896A patent/IL188896A0/en unknown
- 2008-01-25 NO NO20080468A patent/NO20080468L/no not_active Application Discontinuation
- 2008-01-30 EC EC2008008151A patent/ECSP088151A/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP1907390A2 (en) | 2008-04-09 |
CA2616161A1 (en) | 2007-02-08 |
AR054849A1 (es) | 2007-07-18 |
BRPI0614154A2 (pt) | 2011-03-15 |
JP2009502925A (ja) | 2009-01-29 |
US7671196B2 (en) | 2010-03-02 |
NO20080468L (no) | 2008-02-22 |
RU2008102884A (ru) | 2009-09-10 |
GT200600326A (es) | 2007-03-14 |
CR9670A (es) | 2008-07-29 |
SA06270241B1 (ar) | 2009-09-02 |
US20070027142A1 (en) | 2007-02-01 |
KR20080030682A (ko) | 2008-04-04 |
AU2006276010A1 (en) | 2007-02-08 |
MX2008001030A (es) | 2008-03-19 |
IL188896A0 (en) | 2008-04-13 |
WO2007016029A2 (en) | 2007-02-08 |
CN101268076A (zh) | 2008-09-17 |
WO2007016029A3 (en) | 2007-05-18 |
TW200738713A (en) | 2007-10-16 |
PE20070238A1 (es) | 2007-03-26 |
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