ATE360617T1 - Benzoheterocyclische verbindungen verwendbar als vasopressin- oder oxytocin-modulatoren - Google Patents

Benzoheterocyclische verbindungen verwendbar als vasopressin- oder oxytocin-modulatoren

Info

Publication number
ATE360617T1
ATE360617T1 AT02007987T AT02007987T ATE360617T1 AT E360617 T1 ATE360617 T1 AT E360617T1 AT 02007987 T AT02007987 T AT 02007987T AT 02007987 T AT02007987 T AT 02007987T AT E360617 T1 ATE360617 T1 AT E360617T1
Authority
AT
Austria
Prior art keywords
vasopressin
benzohetrocyclic
oxytocin
compounds usable
activity
Prior art date
Application number
AT02007987T
Other languages
English (en)
Inventor
Hidenori Ogawa
Kazumi Kondo
Hiroshi Yamashita
Keizo Kan
Takayuki Matsuzaki
Tomoichi Shinohara
Kokuwajima-Aha-Maehama
Yoshihisa Tanada
Muneaki Kurimura
Michiaki Tominaga
Yoichi Yabuuchi
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Application granted granted Critical
Publication of ATE360617T1 publication Critical patent/ATE360617T1/de

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    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
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    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
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    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
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AT02007987T 1994-06-15 1995-06-07 Benzoheterocyclische verbindungen verwendbar als vasopressin- oder oxytocin-modulatoren ATE360617T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP13235594 1994-06-15
JP7072795 1995-03-03

Publications (1)

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ATE360617T1 true ATE360617T1 (de) 2007-05-15

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AT95921112T ATE239710T1 (de) 1994-06-15 1995-06-07 Benzoheterocyclische derivate verwendbar als vasopressin- oder oxytocin-modulatoren
AT02007987T ATE360617T1 (de) 1994-06-15 1995-06-07 Benzoheterocyclische verbindungen verwendbar als vasopressin- oder oxytocin-modulatoren

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AT95921112T ATE239710T1 (de) 1994-06-15 1995-06-07 Benzoheterocyclische derivate verwendbar als vasopressin- oder oxytocin-modulatoren

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US (3) US6096735A (de)
EP (2) EP1221440B1 (de)
JP (1) JP2000351768A (de)
KR (1) KR100433375B1 (de)
CN (2) CN1104418C (de)
AT (2) ATE239710T1 (de)
CA (1) CA2192928C (de)
DE (2) DE69535486T2 (de)
DK (2) DK1221440T3 (de)
ES (2) ES2199251T3 (de)
MX (1) MX9606510A (de)
PT (2) PT1221440E (de)
TW (1) TW467899B (de)
WO (1) WO1995034540A1 (de)

Families Citing this family (74)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW359669B (en) * 1995-12-15 1999-06-01 Otsuka Pharma Co Ltd Benzazepine derivatives
AUPO395396A0 (en) * 1996-12-02 1997-01-02 Fujisawa Pharmaceutical Co., Ltd. Benzamide derivatives
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MX9606510A (es) 1997-03-29
DE69530690T2 (de) 2004-03-18
PT765314E (pt) 2003-09-30
AU690283B2 (en) 1998-04-23
TW467899B (en) 2001-12-11
CN1313280A (zh) 2001-09-19
US6642223B2 (en) 2003-11-04
EP1221440B1 (de) 2007-04-25
ATE239710T1 (de) 2003-05-15
CA2192928A1 (en) 1995-12-21
EP1221440A1 (de) 2002-07-10
ES2284741T3 (es) 2007-11-16
CN100384825C (zh) 2008-04-30
ES2199251T3 (es) 2004-02-16
CN1104418C (zh) 2003-04-02
WO1995034540A1 (en) 1995-12-21
KR970703317A (ko) 1997-07-03
DE69535486D1 (de) 2007-06-06
KR100433375B1 (ko) 2005-09-23
DE69535486T2 (de) 2008-04-10
DK0765314T3 (da) 2003-08-25
EP0765314A1 (de) 1997-04-02
JP2000351768A (ja) 2000-12-19
CN1150799A (zh) 1997-05-28
US6335327B1 (en) 2002-01-01
EP0765314B1 (de) 2003-05-07
PT1221440E (pt) 2007-07-20
AU2629395A (en) 1996-01-05
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US20020049194A1 (en) 2002-04-25
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