NO20051193L - Vanilloidreseptorligander, fremgangsmate for fremstilling og anvendelse av disse. - Google Patents
Vanilloidreseptorligander, fremgangsmate for fremstilling og anvendelse av disse.Info
- Publication number
- NO20051193L NO20051193L NO20051193A NO20051193A NO20051193L NO 20051193 L NO20051193 L NO 20051193L NO 20051193 A NO20051193 A NO 20051193A NO 20051193 A NO20051193 A NO 20051193A NO 20051193 L NO20051193 L NO 20051193L
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- Prior art keywords
- inflammatory
- disorders
- pain
- headache
- general
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- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
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Abstract
Forbindelser som har generell Btruktur (I) YX^ og preparater som inneholder slike, for behandling av akutt inClammatorisk og neuropatisk smerte, dental smerte, generell hodepine, migrene, "duster"- hodepine, blandede vaskulære og ikke- vaskulsre syndromer, spenningshodepine, generell inflamrnaejon, artritt, reumat- iske sykdommer, osteoartritt, inflamma- toriske tarmlidelser, inflammatoriske øyelideleer, inflammatoriske eller ustabile blxrelidelser, psoriasis, hud- plager med inflammatoriske konponenter, kroniske inflammatoriske tilstander, inflammatorisk smerte og tilhørende hyperalgesi og allodyni, neuropatisk smerte og tilhørende hyperalgesi og allodyni, diabetisk neuropatisk smerte, kausalgi, sympatisk vedvarende smerte, deafferenteringseyndromer, astma, epitelvevsskade eller dysfunksjon, herpes simplex, forstyrrelser i visceral motilitet i respiratoriske, genitourinare, gastrointestinale eller vaskulære områder, sår, brannsår, allergiske hudreaksjoner, pruritt, vitiligo, generelle gastrointestinale lidelser, gastrisk ulcer, duodenalt
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- 2003-08-08 WO PCT/US2003/025191 patent/WO2004014871A1/en active Application Filing
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- 2005-03-07 NO NO20051193A patent/NO20051193L/no not_active Application Discontinuation
- 2005-08-01 US US11/195,134 patent/US7148221B2/en not_active Expired - Fee Related
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PL376372A1 (en) | 2005-12-27 |
US7332511B2 (en) | 2008-02-19 |
EP1546116A1 (en) | 2005-06-29 |
RS20050161A (en) | 2007-09-21 |
JP4555082B2 (ja) | 2010-09-29 |
KR20050055694A (ko) | 2005-06-13 |
US7144888B2 (en) | 2006-12-05 |
EA010380B1 (ru) | 2008-08-29 |
US20050272777A1 (en) | 2005-12-08 |
MXPA05001456A (es) | 2005-06-06 |
WO2004014871A8 (en) | 2005-04-07 |
TW200410945A (en) | 2004-07-01 |
AR041191A1 (es) | 2005-05-04 |
CA2493667A1 (en) | 2004-02-19 |
NZ537952A (en) | 2008-04-30 |
CN1694873A (zh) | 2005-11-09 |
EP2270006A1 (en) | 2011-01-05 |
US7148221B2 (en) | 2006-12-12 |
EP1717220A2 (en) | 2006-11-02 |
AU2003264047B2 (en) | 2008-06-26 |
EA200500168A1 (ru) | 2005-08-25 |
US20040082780A1 (en) | 2004-04-29 |
IL166396A0 (en) | 2006-01-15 |
AU2003264047A1 (en) | 2004-02-25 |
ZA200501332B (en) | 2007-04-25 |
JP2006504670A (ja) | 2006-02-09 |
US20050277631A1 (en) | 2005-12-15 |
BR0313255A (pt) | 2005-07-12 |
EP1717220A3 (en) | 2007-08-22 |
AU2008202517A1 (en) | 2008-06-26 |
WO2004014871A1 (en) | 2004-02-19 |
CA2493667C (en) | 2010-04-27 |
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