NO20024281L - Indolderivater, fremgangsmÕte for fremstilling av de samme og anvendelse derav - Google Patents

Indolderivater, fremgangsmÕte for fremstilling av de samme og anvendelse derav

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Publication number
NO20024281L
NO20024281L NO20024281A NO20024281A NO20024281L NO 20024281 L NO20024281 L NO 20024281L NO 20024281 A NO20024281 A NO 20024281A NO 20024281 A NO20024281 A NO 20024281A NO 20024281 L NO20024281 L NO 20024281L
Authority
NO
Norway
Prior art keywords
diseases
allergic
urticaria
inflammation
general formula
Prior art date
Application number
NO20024281A
Other languages
English (en)
Norwegian (no)
Other versions
NO20024281D0 (no
Inventor
Kazushiki Torisu
Kaoru Kobayashi
Fumio Nambu
Original Assignee
Ono Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co
Publication of NO20024281D0 publication Critical patent/NO20024281D0/no
Publication of NO20024281L publication Critical patent/NO20024281L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/22—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an aralkyl radical attached to the ring nitrogen atom
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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  • Oncology (AREA)
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  • Neurosurgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
NO20024281A 2000-03-09 2002-09-06 Indolderivater, fremgangsmÕte for fremstilling av de samme og anvendelse derav NO20024281L (no)

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JP2000064696 2000-03-09
JP2000231857 2000-07-31
PCT/JP2001/001817 WO2001066520A1 (fr) 2000-03-09 2001-03-08 Derives indole, procede de preparation de ces derives et leur utilisation

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NO20024281L true NO20024281L (no) 2002-11-08

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RU2002123882A (ru) 2004-03-20
US6743793B2 (en) 2004-06-01
US20030176400A1 (en) 2003-09-18
JP4292742B2 (ja) 2009-07-08
KR20030010589A (ko) 2003-02-05
NZ521192A (en) 2005-01-28
EP1262475A4 (de) 2005-01-05
CN1179945C (zh) 2004-12-15
US20040180885A1 (en) 2004-09-16
CN1427824A (zh) 2003-07-02
WO2001066520A1 (fr) 2001-09-13
US7098234B2 (en) 2006-08-29
HUP0301493A2 (hu) 2003-08-28
RU2259998C2 (ru) 2005-09-10
CA2402174A1 (en) 2001-09-13
BR0109050A (pt) 2004-04-27
NO20024281D0 (no) 2002-09-06
MXPA02008801A (es) 2003-07-07
EP1262475A1 (de) 2002-12-04
AU2001241068A1 (en) 2001-09-17

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