NO20021528L - Kinuklidinforbindelser og medikamenter inneholdende de samme som den aktive bestanddel - Google Patents

Kinuklidinforbindelser og medikamenter inneholdende de samme som den aktive bestanddel

Info

Publication number
NO20021528L
NO20021528L NO20021528A NO20021528A NO20021528L NO 20021528 L NO20021528 L NO 20021528L NO 20021528 A NO20021528 A NO 20021528A NO 20021528 A NO20021528 A NO 20021528A NO 20021528 L NO20021528 L NO 20021528L
Authority
NO
Norway
Prior art keywords
optionally substituted
chain
substituted
denotes
represented
Prior art date
Application number
NO20021528A
Other languages
English (en)
Other versions
NO20021528D0 (no
NO328218B1 (no
Inventor
Toshimi Okada
Nobuyuki Kurusu
Keigo Tanaka
Kazuki Miyazaki
Daisuke Shinmyo
Hiroyuki Sugumi
Hironori Ikuta
Hironobu Hiyoshi
Takao Saeki
Mamoru Yanagimachi
Masashi Ito
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of NO20021528D0 publication Critical patent/NO20021528D0/no
Publication of NO20021528L publication Critical patent/NO20021528L/no
Publication of NO328218B1 publication Critical patent/NO328218B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20021528A 1999-09-28 2002-03-26 Kinuklidinforbindelser, anvendelse derav, fremgangsmater for fremstilling derav, og medisinske preparater omfattende slike NO328218B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP27390599 1999-09-28
JP2000179352 2000-06-15
PCT/JP2000/006665 WO2001023383A1 (fr) 1999-09-28 2000-09-27 Composes de quinuclidine et medicaments contenant ces composes comme principe actif

Publications (3)

Publication Number Publication Date
NO20021528D0 NO20021528D0 (no) 2002-03-26
NO20021528L true NO20021528L (no) 2002-05-28
NO328218B1 NO328218B1 (no) 2010-01-11

Family

ID=26550809

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20021528A NO328218B1 (no) 1999-09-28 2002-03-26 Kinuklidinforbindelser, anvendelse derav, fremgangsmater for fremstilling derav, og medisinske preparater omfattende slike

Country Status (20)

Country Link
US (1) US6599917B1 (no)
EP (1) EP1217001B1 (no)
JP (1) JP4206212B2 (no)
KR (1) KR100694687B1 (no)
CN (1) CN100334085C (no)
AT (1) ATE312100T1 (no)
AU (1) AU782114B2 (no)
BR (1) BR0014331A (no)
CA (1) CA2385995C (no)
DE (1) DE60024651T2 (no)
DK (1) DK1217001T3 (no)
ES (1) ES2252063T3 (no)
HU (1) HUP0203514A3 (no)
IL (2) IL148631A0 (no)
MX (1) MXPA02003167A (no)
NO (1) NO328218B1 (no)
NZ (1) NZ517788A (no)
RU (1) RU2266905C2 (no)
TW (1) TWI282794B (no)
WO (1) WO2001023383A1 (no)

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TW200526631A (en) * 2003-10-07 2005-08-16 Renovis Inc Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
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US8106066B2 (en) 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
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TW201111385A (en) 2009-08-27 2011-04-01 Biocryst Pharm Inc Heterocyclic compounds as janus kinase inhibitors
US8420661B2 (en) * 2010-04-13 2013-04-16 Hoffmann-La Roche Inc. Arylethynyl derivatives
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SI3141542T1 (sl) 2011-12-28 2020-11-30 Global Blood Therapeutics, Inc. Substituirane spojine benzaldehida in metode njihove uporabe pri povečanju oksigenacije tkiva
WO2013102145A1 (en) 2011-12-28 2013-07-04 Global Blood Therapeutics, Inc. Substituted heteroaryl aldehyde compounds and methods for their use in increasing tissue oxygenation
WO2014060381A1 (de) 2012-10-18 2014-04-24 Bayer Cropscience Ag Heterocyclische verbindungen als schädlingsbekämpfungsmittel
EP2914587A1 (de) 2012-10-31 2015-09-09 Bayer CropScience AG Neue heterocylische verbindungen als schädlingsbekämpfungsmittel
US9604999B2 (en) 2013-03-15 2017-03-28 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
US8952171B2 (en) 2013-03-15 2015-02-10 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
CN105073728A (zh) 2013-03-15 2015-11-18 全球血液疗法股份有限公司 化合物及其用于调节血红蛋白的用途
WO2014145040A1 (en) 2013-03-15 2014-09-18 Global Blood Therapeutics, Inc. Substituted aldehyde compounds and methods for their use in increasing tissue oxygenation
US9458139B2 (en) 2013-03-15 2016-10-04 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
US20140274961A1 (en) 2013-03-15 2014-09-18 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
KR101971385B1 (ko) 2013-03-15 2019-04-22 글로벌 블러드 테라퓨틱스, 인크. 헤모글로빈 조정을 위한 화합물 및 이의 용도
US9802900B2 (en) 2013-03-15 2017-10-31 Global Blood Therapeutics, Inc. Bicyclic heteroaryl compounds and uses thereof for the modulation of hemoglobin
US10266551B2 (en) 2013-03-15 2019-04-23 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
CN105246477A (zh) 2013-03-15 2016-01-13 全球血液疗法股份有限公司 化合物及其用于调节血红蛋白的用途
US9422279B2 (en) 2013-03-15 2016-08-23 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
EA202092627A1 (ru) 2013-11-18 2021-09-30 Глобал Блад Терапьютикс, Инк. Соединения и их применения для модуляции гемоглобина
EA028529B1 (ru) 2014-02-07 2017-11-30 Глобал Блад Терапьютикс, Инк. Кристаллические полиморфные формы свободного основания 2-гидрокси-6-((2-(1-изопропил-1н-пиразол-5-ил)пиридин-3-ил)метокси)бензальдегида
MA41841A (fr) 2015-03-30 2018-02-06 Global Blood Therapeutics Inc Composés aldéhyde pour le traitement de la fibrose pulmonaire, de l'hypoxie, et de maladies auto-immunes et des tissus conjonctifs
AU2016273751B2 (en) 2015-06-03 2020-04-02 F. Hoffmann-La Roche Ag Ethynyl derivatives
MX2018006832A (es) 2015-12-04 2018-11-09 Global Blood Therapeutics Inc Regimenes de dosificacion de 2-hidroxi-6-((2-(1-isopropil-1h-piraz ol-5-il)-piridin-3-il)-metoxi)-benzaldehido.
TWI663160B (zh) 2016-05-12 2019-06-21 全球血液治療公司 用於合成2-羥基-6-((2-(1-異丙基-1h-吡唑-5-基)-吡啶-3-基)甲氧基)苯甲醛之方法
TWI778983B (zh) 2016-10-12 2022-10-01 美商全球血液治療公司 包含2-羥基-6-((2-(1-異丙基-1h-吡唑-5-基)吡啶-3-基)甲氧基)-苯甲醛之片劑
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Also Published As

Publication number Publication date
DE60024651T2 (de) 2006-09-28
KR20020034197A (ko) 2002-05-08
AU782114B2 (en) 2005-07-07
IL148631A (en) 2010-04-29
CN1377349A (zh) 2002-10-30
HUP0203514A3 (en) 2004-01-28
NZ517788A (en) 2003-11-28
AU7446400A (en) 2001-04-30
DE60024651D1 (de) 2006-01-12
TWI282794B (en) 2007-06-21
ES2252063T3 (es) 2006-05-16
JP4206212B2 (ja) 2009-01-07
CA2385995C (en) 2009-06-16
KR100694687B1 (ko) 2007-03-13
CN100334085C (zh) 2007-08-29
HUP0203514A2 (hu) 2003-03-28
WO2001023383A1 (fr) 2001-04-05
EP1217001A4 (en) 2002-12-18
EP1217001B1 (en) 2005-12-07
ATE312100T1 (de) 2005-12-15
NO20021528D0 (no) 2002-03-26
DK1217001T3 (da) 2006-03-20
EP1217001A1 (en) 2002-06-26
MXPA02003167A (es) 2003-10-06
IL148631A0 (en) 2002-09-12
BR0014331A (pt) 2003-06-10
RU2266905C2 (ru) 2005-12-27
CA2385995A1 (en) 2001-04-05
US6599917B1 (en) 2003-07-29
NO328218B1 (no) 2010-01-11

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Legal Events

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