NO20015362L - Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse derav - Google Patents
Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse deravInfo
- Publication number
- NO20015362L NO20015362L NO20015362A NO20015362A NO20015362L NO 20015362 L NO20015362 L NO 20015362L NO 20015362 A NO20015362 A NO 20015362A NO 20015362 A NO20015362 A NO 20015362A NO 20015362 L NO20015362 L NO 20015362L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- heterocyclic substituted
- substituted benzimidazoles
- benzimidazoles
- heterocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/10—Antiepileptics; Anticonvulsants for petit-mal
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/18—Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Communicable Diseases (AREA)
- Psychology (AREA)
- Cardiology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Oncology (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19920936A DE19920936A1 (de) | 1999-05-07 | 1999-05-07 | Heterozyklisch substituierte Benzimidazole, deren Herstellung und Anwendung |
PCT/EP2000/003813 WO2000068206A1 (de) | 1999-05-07 | 2000-04-27 | Heterozyklisch substituierte benzimidazole, deren herstellung und anwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20015362D0 NO20015362D0 (no) | 2001-11-02 |
NO20015362L true NO20015362L (no) | 2001-11-02 |
Family
ID=7907219
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20015362A NO20015362L (no) | 1999-05-07 | 2001-11-02 | Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse derav |
Country Status (27)
Country | Link |
---|---|
US (1) | US6696437B1 (no) |
EP (1) | EP1177178B1 (no) |
JP (1) | JP4004737B2 (no) |
KR (1) | KR20010112477A (no) |
CN (1) | CN1353695A (no) |
AR (1) | AR029161A1 (no) |
AT (1) | ATE286029T1 (no) |
AU (1) | AU4558400A (no) |
BG (1) | BG106035A (no) |
BR (1) | BR0010342A (no) |
CA (1) | CA2371645C (no) |
CO (1) | CO5170517A1 (no) |
DE (2) | DE19920936A1 (no) |
DK (1) | DK1177178T3 (no) |
ES (1) | ES2235869T3 (no) |
HK (1) | HK1046281A1 (no) |
HU (1) | HUP0202970A2 (no) |
IL (1) | IL146147A0 (no) |
MY (1) | MY122771A (no) |
NO (1) | NO20015362L (no) |
PL (1) | PL351558A1 (no) |
PT (1) | PT1177178E (no) |
SK (1) | SK15962001A3 (no) |
TR (1) | TR200103221T2 (no) |
UA (1) | UA68436C2 (no) |
WO (1) | WO2000068206A1 (no) |
ZA (1) | ZA200108609B (no) |
Families Citing this family (78)
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BR9915013A (pt) | 1998-11-03 | 2001-08-07 | Basf Ag | Composto, uso dos mesmos, processo para preparar os mesmos, droga, e, método para detecção in vitro para inibidores parp |
ATE265998T1 (de) * | 2000-03-20 | 2004-05-15 | N Gene Res Lab Inc | Propancarbonsäure-amidoxim derivate, ein verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen, die diese entahlten |
ATE369853T1 (de) | 2001-03-12 | 2007-09-15 | Avanir Pharmaceuticals | Benzimidazolderivate zur ige-modulierung und zellproliferationshemmung |
AU2002312371A1 (en) | 2001-06-13 | 2002-12-23 | Roland W. Burli | Aryl-benzimidazole compounds having antiinfective activity |
US7642278B2 (en) | 2001-07-03 | 2010-01-05 | Novartis Vaccines And Diagnostics, Inc. | Indazole benzimidazole compounds |
EP1401831A1 (en) | 2001-07-03 | 2004-03-31 | Chiron Corporation | Indazole benzimidazole compounds as tyrosine and serine/threonine kinase inhibitors |
RU2004126671A (ru) * | 2002-02-06 | 2005-04-10 | Вертекс Фармасьютикалз Инкорпорейтед (Us) | Гетероарилсоединения, полезные в качестве ингибиторов gsk-3 |
DE10227668A1 (de) * | 2002-06-20 | 2004-01-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Arzneimittel zur Behandlung des systemic inflammatory response syndrome |
ATE405658T1 (de) | 2002-07-26 | 2008-09-15 | Basf Plant Science Gmbh | Neue selektionsverfahren |
ATE425753T1 (de) | 2002-08-02 | 2009-04-15 | Genesoft Pharmaceuticals Inc | Biaryl-verbindungen mit antiinfektiver wirkung |
EP1531674B1 (en) | 2002-08-19 | 2014-06-18 | Lorus Therapeutics Inc. | 2,4,5-trisubstituted imidazoles and their use as anti-microbial agents |
AU2003270426A1 (en) | 2002-09-12 | 2004-04-30 | Avanir Pharmaceuticals | PHENYL-INDOLE COMPOUNDS FOR MODULATING IgE AND INHIBITING CELLULAR PROLIFERATION |
TWI276631B (en) | 2002-09-12 | 2007-03-21 | Avanir Pharmaceuticals | Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation |
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EP1562931A2 (en) | 2002-10-25 | 2005-08-17 | Genesoft Pharmaceuticals, Inc. | Anti-infective biaryl compounds |
ES2376166T3 (es) | 2002-11-22 | 2012-03-09 | Mitsubishi Tanabe Pharma Corporation | Compuestos de isoquinolina y su uso medicinal. |
AU2003297822A1 (en) | 2002-12-10 | 2004-06-30 | Oscient Pharmaceuticals Corporation | Antibacterial compounds having a (pyrrole carboxamide)-(benzamide)-(imidazole carboxamide) motif |
SE0301371D0 (sv) * | 2003-05-09 | 2003-05-09 | Astrazeneca Ab | New Compounds |
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JP4767857B2 (ja) * | 2003-09-30 | 2011-09-07 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ベンゾイミダゾール化合物 |
DE602004020364D1 (de) * | 2003-09-30 | 2009-05-14 | Janssen Pharmaceutica Nv | Benzoimidazolverbindungen |
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FR2862971B1 (fr) * | 2003-11-28 | 2006-03-24 | Sod Conseils Rech Applic | Nouveaux derives de benzimidazole et d'imidazo-pyridine et leur utilisation en tant que medicament |
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CN111417395A (zh) | 2017-10-30 | 2020-07-14 | 艾普托斯生物科学公司 | 用于治疗癌症的芳基咪唑 |
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ZA885929B (en) * | 1987-08-25 | 1989-04-26 | Oxi Gene Inc | Agents for use in tumor or cancer cell killing therapy |
DK0841924T3 (da) * | 1995-08-02 | 2003-02-10 | Univ Newcastle Ventures Ltd | Benzimidazolforbindelser |
EP2223920A3 (en) * | 1996-06-19 | 2011-09-28 | Aventis Pharma Limited | Substituted azabicyclic compounds |
BR9915013A (pt) * | 1998-11-03 | 2001-08-07 | Basf Ag | Composto, uso dos mesmos, processo para preparar os mesmos, droga, e, método para detecção in vitro para inibidores parp |
BR9915381A (pt) * | 1998-11-17 | 2001-08-14 | Basf Ag | Uso de um composto, e, composto |
HUP0200749A3 (en) * | 1998-11-27 | 2003-03-28 | Basf Ag | Substituted benzimidazoles and their use as parp inhibitors and process for their preparation |
-
1999
- 1999-05-07 DE DE19920936A patent/DE19920936A1/de not_active Withdrawn
-
2000
- 2000-04-27 HU HU0202970A patent/HUP0202970A2/hu unknown
- 2000-04-27 CA CA002371645A patent/CA2371645C/en not_active Expired - Fee Related
- 2000-04-27 CN CN00808364A patent/CN1353695A/zh active Pending
- 2000-04-27 AU AU45584/00A patent/AU4558400A/en not_active Abandoned
- 2000-04-27 DK DK00927088T patent/DK1177178T3/da active
- 2000-04-27 ES ES00927088T patent/ES2235869T3/es not_active Expired - Lifetime
- 2000-04-27 DE DE50009118T patent/DE50009118D1/de not_active Expired - Lifetime
- 2000-04-27 AT AT00927088T patent/ATE286029T1/de active
- 2000-04-27 TR TR2001/03221T patent/TR200103221T2/xx unknown
- 2000-04-27 BR BR0010342-0A patent/BR0010342A/pt not_active IP Right Cessation
- 2000-04-27 PT PT00927088T patent/PT1177178E/pt unknown
- 2000-04-27 EP EP00927088A patent/EP1177178B1/de not_active Expired - Lifetime
- 2000-04-27 UA UA2001128419A patent/UA68436C2/uk unknown
- 2000-04-27 JP JP2000617186A patent/JP4004737B2/ja not_active Expired - Fee Related
- 2000-04-27 KR KR1020017014145A patent/KR20010112477A/ko not_active Application Discontinuation
- 2000-04-27 IL IL14614700A patent/IL146147A0/xx unknown
- 2000-04-27 PL PL00351558A patent/PL351558A1/xx not_active Application Discontinuation
- 2000-04-27 SK SK1596-2001A patent/SK15962001A3/sk unknown
- 2000-04-27 US US09/959,632 patent/US6696437B1/en not_active Expired - Lifetime
- 2000-04-27 WO PCT/EP2000/003813 patent/WO2000068206A1/de not_active Application Discontinuation
- 2000-05-05 CO CO00032472A patent/CO5170517A1/es not_active Application Discontinuation
- 2000-05-05 AR ARP000102178A patent/AR029161A1/es unknown
- 2000-05-05 MY MYPI20001934A patent/MY122771A/en unknown
-
2001
- 2001-10-19 ZA ZA200108609A patent/ZA200108609B/en unknown
- 2001-10-22 BG BG106035A patent/BG106035A/xx unknown
- 2001-11-02 NO NO20015362A patent/NO20015362L/no not_active Application Discontinuation
-
2002
- 2002-10-30 HK HK02107871.7A patent/HK1046281A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
DE50009118D1 (de) | 2005-02-03 |
IL146147A0 (en) | 2002-07-25 |
NO20015362D0 (no) | 2001-11-02 |
HUP0202970A2 (hu) | 2002-12-28 |
MY122771A (en) | 2006-05-31 |
CA2371645A1 (en) | 2000-11-16 |
TR200103221T2 (tr) | 2002-04-22 |
SK15962001A3 (sk) | 2002-06-04 |
US6696437B1 (en) | 2004-02-24 |
JP2002544199A (ja) | 2002-12-24 |
EP1177178B1 (de) | 2004-12-29 |
CA2371645C (en) | 2007-04-17 |
CO5170517A1 (es) | 2002-06-27 |
ATE286029T1 (de) | 2005-01-15 |
BG106035A (en) | 2002-06-28 |
AU4558400A (en) | 2000-11-21 |
UA68436C2 (en) | 2004-08-16 |
PL351558A1 (en) | 2003-05-05 |
AR029161A1 (es) | 2003-06-18 |
DE19920936A1 (de) | 2000-11-09 |
EP1177178A1 (de) | 2002-02-06 |
JP4004737B2 (ja) | 2007-11-07 |
KR20010112477A (ko) | 2001-12-20 |
CN1353695A (zh) | 2002-06-12 |
HK1046281A1 (zh) | 2003-01-03 |
BR0010342A (pt) | 2002-05-28 |
PT1177178E (pt) | 2005-05-31 |
WO2000068206A1 (de) | 2000-11-16 |
DK1177178T3 (da) | 2005-05-02 |
ZA200108609B (en) | 2002-10-21 |
ES2235869T3 (es) | 2005-07-16 |
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