NO174053C - Analogifremgangsmåte for fremstilling av terapeutisk aktive R(-) 3-kinuklidinol-derivater - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktive R(-) 3-kinuklidinol-derivater

Info

Publication number
NO174053C
NO174053C NO902710A NO902710A NO174053C NO 174053 C NO174053 C NO 174053C NO 902710 A NO902710 A NO 902710A NO 902710 A NO902710 A NO 902710A NO 174053 C NO174053 C NO 174053C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
analogous process
quinuclidinol derivatives
quinuclidinol
Prior art date
Application number
NO902710A
Other languages
English (en)
Other versions
NO174053B (no
NO902710D0 (no
NO902710L (no
Inventor
Enzo Cereda
Arturo Donetti
Giuseppe Bietti
Antonio Schiavone
Giovanni Battista Schiavi
Henri Nico Doods
Original Assignee
Boehringer Ingelheim Italia
Angeli Inst Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Italia, Angeli Inst Spa filed Critical Boehringer Ingelheim Italia
Publication of NO902710D0 publication Critical patent/NO902710D0/no
Publication of NO902710L publication Critical patent/NO902710L/no
Publication of NO174053B publication Critical patent/NO174053B/no
Publication of NO174053C publication Critical patent/NO174053C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
NO902710A 1989-06-20 1990-06-19 Analogifremgangsmåte for fremstilling av terapeutisk aktive R(-) 3-kinuklidinol-derivater NO174053C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8920929A IT1230881B (it) 1989-06-20 1989-06-20 Derivati del r(-) 3-chinuclidinolo

Publications (4)

Publication Number Publication Date
NO902710D0 NO902710D0 (no) 1990-06-19
NO902710L NO902710L (no) 1990-12-21
NO174053B NO174053B (no) 1993-11-29
NO174053C true NO174053C (no) 1994-03-16

Family

ID=11174223

Family Applications (1)

Application Number Title Priority Date Filing Date
NO902710A NO174053C (no) 1989-06-20 1990-06-19 Analogifremgangsmåte for fremstilling av terapeutisk aktive R(-) 3-kinuklidinol-derivater

Country Status (19)

Country Link
US (1) US5164386A (no)
EP (1) EP0404737A3 (no)
JP (1) JPH0331279A (no)
KR (1) KR910000720A (no)
AU (1) AU634787B2 (no)
CA (1) CA2019251A1 (no)
DD (1) DD300105A5 (no)
FI (1) FI94131C (no)
HU (1) HUT54151A (no)
IE (1) IE902208A1 (no)
IL (1) IL94763A (no)
IT (1) IT1230881B (no)
NO (1) NO174053C (no)
NZ (1) NZ234157A (no)
PL (1) PL164218B1 (no)
PT (1) PT94408A (no)
RU (1) RU2034843C1 (no)
YU (1) YU47356B (no)
ZA (1) ZA904736B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9106571D0 (en) * 1991-03-27 1991-05-15 Erba Carlo Spa Derivatives of substituted imidazol-2-one and process for their preparation
US5202318A (en) * 1990-05-14 1993-04-13 Syntex (U.S.A.) Inc. Tricyclic compounds acting at serotonin receptor subtypes
AU7618991A (en) * 1990-05-14 1991-11-14 Syntex (U.S.A.) Inc. Novel tricyclic compounds
WO1992012151A1 (en) * 1991-01-10 1992-07-23 Pfizer Inc. N-alkyl quinuclidinium salts as substance p antagonists
US5340826A (en) * 1993-02-04 1994-08-23 Pfizer Inc. Pharmaceutical agents for treatment of urinary incontinence
US7214686B2 (en) * 1997-06-30 2007-05-08 Targacept, Inc. Pharmaceutical compositions and methods for effecting dopamine release
JP4295985B2 (ja) 2000-12-28 2009-07-15 ラボラトリオス・アルミラル・ソシエダッド・アノニマ 新規なキヌクリジン誘導体およびそれを含む医薬組成物
CA3178035A1 (en) 2012-12-24 2014-07-03 Neurogastrx, Inc. Methods for treating gi tract disorders
WO2015200369A1 (en) 2014-06-24 2015-12-30 Neurogastrx, Inc. Prodrugs of metopimazine
KR102423577B1 (ko) 2017-04-07 2022-07-21 삼성전자주식회사 가전기기
US10836757B1 (en) 2020-04-02 2020-11-17 Neurogastrx, Inc. Polymorphic forms of metopimazine

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3290316A (en) * 1962-08-03 1966-12-06 Hoffmann La Roche Alpha-3-pyridylmandelic acid and derivatives thereof
WO1985001048A1 (en) * 1983-08-26 1985-03-14 Sandoz Ag Aromatic esters or amides of carboxylic acid and sulfonic acid
CA1307790C (en) * 1987-08-04 1992-09-22 Ian Anthony Cliffe Ethers
ZA886585B (en) * 1987-09-08 1990-05-30 Lilly Co Eli Specific 5-ht,antagonists
US4921982A (en) * 1988-07-21 1990-05-01 Eli Lilly And Company 5-halo-2,3-dihydro-2,2-dimethylbenzofuran-7-carboxylic acids useful as intermediates for 5-HT3 antagonists
IT1231413B (it) * 1987-09-23 1991-12-04 Angeli Inst Spa Derivati dell'acido benzimidazolin-2-osso-1-carbossilico utili come antagonisti dei recettori 5-ht
US4975437A (en) * 1989-12-14 1990-12-04 Marion Laboratories, Inc. Isomers of 1-azabicyclo(2.2.2)oct-3-yl 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-5-nitropyridine-3-carboxylate

Also Published As

Publication number Publication date
HU903908D0 (en) 1990-11-28
PT94408A (pt) 1991-02-08
YU47356B (sh) 1995-01-31
EP0404737A3 (en) 1992-03-11
US5164386A (en) 1992-11-17
IT8920929A0 (it) 1989-06-20
FI903077A0 (fi) 1990-06-19
AU634787B2 (en) 1993-03-04
JPH0331279A (ja) 1991-02-12
NO174053B (no) 1993-11-29
AU5764990A (en) 1991-01-03
IL94763A0 (en) 1991-04-15
IT1230881B (it) 1991-11-08
HUT54151A (en) 1991-01-28
NO902710D0 (no) 1990-06-19
IL94763A (en) 1994-08-26
DD300105A5 (de) 1992-05-21
CA2019251A1 (en) 1990-12-20
NO902710L (no) 1990-12-21
FI94131C (fi) 1995-07-25
ZA904736B (en) 1992-02-26
EP0404737A2 (en) 1990-12-27
PL285669A1 (en) 1991-03-11
FI94131B (fi) 1995-04-13
RU2034843C1 (ru) 1995-05-10
IE902208L (en) 1990-12-20
KR910000720A (ko) 1991-01-30
YU120290A (sh) 1992-12-21
NZ234157A (en) 1992-09-25
IE902208A1 (en) 1991-01-02
PL164218B1 (pl) 1994-07-29

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