NO175478C - Analogifremgangsmåte for fremstilling av terapeutisk aktive diazepin-derivater - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktive diazepin-derivater

Info

Publication number
NO175478C
NO175478C NO904986A NO904986A NO175478C NO 175478 C NO175478 C NO 175478C NO 904986 A NO904986 A NO 904986A NO 904986 A NO904986 A NO 904986A NO 175478 C NO175478 C NO 175478C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
analogous process
diazepine derivatives
diazepine
Prior art date
Application number
NO904986A
Other languages
English (en)
Other versions
NO904986D0 (no
NO904986L (no
NO175478B (no
Inventor
Karl D Hargrave
Wolfhard Engel
Gunter Trummlitz
Wolfgang Eberlein
Gunther Schmidt
Original Assignee
Boehringer Ingelheim Pharma
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27412005&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO175478(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma, Thomae Gmbh Dr K filed Critical Boehringer Ingelheim Pharma
Publication of NO904986D0 publication Critical patent/NO904986D0/no
Publication of NO904986L publication Critical patent/NO904986L/no
Publication of NO175478B publication Critical patent/NO175478B/no
Publication of NO175478C publication Critical patent/NO175478C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO904986A 1989-11-17 1990-11-16 Analogifremgangsmåte for fremstilling av terapeutisk aktive diazepin-derivater NO175478C (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US43892389A 1989-11-17 1989-11-17
US57900190A 1990-09-06 1990-09-06
US60039090A 1990-10-19 1990-10-19

Publications (4)

Publication Number Publication Date
NO904986D0 NO904986D0 (no) 1990-11-16
NO904986L NO904986L (no) 1991-05-21
NO175478B NO175478B (no) 1994-07-11
NO175478C true NO175478C (no) 1994-10-19

Family

ID=27412005

Family Applications (2)

Application Number Title Priority Date Filing Date
NO904986A NO175478C (no) 1989-11-17 1990-11-16 Analogifremgangsmåte for fremstilling av terapeutisk aktive diazepin-derivater
NO1999013C NO1999013I1 (no) 1989-11-17 1999-06-29 Nevirapin

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO1999013C NO1999013I1 (no) 1989-11-17 1999-06-29 Nevirapin

Country Status (21)

Country Link
EP (1) EP0429987B1 (no)
AP (1) AP179A (no)
AT (1) ATE177744T1 (no)
AU (1) AU630251B2 (no)
CA (1) CA2030056C (no)
DE (2) DE19975051I2 (no)
DK (1) DK0429987T3 (no)
ES (1) ES2130114T3 (no)
FI (1) FI94529C (no)
GR (1) GR3030100T3 (no)
HK (1) HK1011025A1 (no)
IE (1) IE904141A1 (no)
IL (1) IL96367A (no)
LU (1) LU90393I2 (no)
NL (1) NL990022I2 (no)
NO (2) NO175478C (no)
NZ (1) NZ236105A (no)
OA (1) OA09852A (no)
PT (1) PT95919B (no)
RU (1) RU2040527C1 (no)
UA (1) UA34420C2 (no)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
GB9109557D0 (en) * 1991-05-02 1991-06-26 Wellcome Found Chemical compounds
JP3133331B2 (ja) * 1991-06-11 2001-02-05 ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド ３―アミノ―２―クロロ―４―アルキルピリジン類の製造方法
US5200522A (en) * 1991-06-11 1993-04-06 Boehringer Ingelheim Pharmaceuticals, Inc. Method for preparing 3-amino-2-chloro-4-alkylpyridines
DE4138853A1 (de) * 1991-11-27 1993-06-03 Bayer Ag 5,6-dihydro-dibenz(b,e)azepin-6,11-dion-11- oxime
DE4138908A1 (de) * 1991-11-27 1993-06-03 Bayer Ag 6-thiono-dibenz(b,e)azepine
EP0598396B1 (en) * 1992-11-18 1998-09-02 Boehringer Ingelheim Pharmaceuticals Inc. Improved method for the preparation of 3-Amino-2-chloro-4-alkylpyridines
AU5883794A (en) * 1993-01-20 1994-08-15 A. Menarini Industrie Farmaceutiche Riunite S.R.L. Diazepin derivatives and antiviral compositions
DE4333697A1 (de) * 1993-10-02 1995-04-06 Merck Patent Gmbh Verfahren zur Herstellung von 3-Aminopyridinen aus 3-Nitropyridinen
DE4403311C1 (de) * 1994-02-03 1995-04-20 Boehringer Ingelheim Kg Verfahren zur Herstellung von Nevirapine (11-Cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3,2-b:2',3'-e][1,4-diazepin]-6-on)
RU2142464C1 (ru) * 1994-02-18 1999-12-10 Берингер Ингельгейм Фармасьютикалз, Инк. 2-гетероарил-5,11-дигидро-6н-дипиридо[3,2-b:2',3'-e][1,4] диазепин-6-оны, их фармацевтически приемлемые соли, фармацевтическая композиция, обладающая ингибирующей активностью в отношении обратной транскриптазы вич-1
US5917033A (en) * 1995-10-31 1999-06-29 University Of Medicine & Dentistry Of New Jersey Structure based design of inhibitors of HIV-1 reverse transcriptase
US5747488A (en) * 1996-01-30 1998-05-05 Boehringer Ingelheim Pharmaceuticals, Inc. 2-aryl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-E! 1, 4!diazepines and their use in the treatment of HIV infection
US6172059B1 (en) * 1997-08-25 2001-01-09 Boehringer Ingelheim Pharmaceuticals, Inc. Pharmaceutical suspension comprising nevirapine hemihydrate
DE10023492A1 (de) * 2000-05-09 2001-11-22 Schering Ag Aza- und Polyazanthranylamide und deren Verwendung als Arzneimittel
US6878714B2 (en) 2001-01-12 2005-04-12 Amgen Inc. Substituted alkylamine derivatives and methods of use
US7105682B2 (en) 2001-01-12 2006-09-12 Amgen Inc. Substituted amine derivatives and methods of use
US7102009B2 (en) 2001-01-12 2006-09-05 Amgen Inc. Substituted amine derivatives and methods of use
US6995162B2 (en) 2001-01-12 2006-02-07 Amgen Inc. Substituted alkylamine derivatives and methods of use
US7307088B2 (en) 2002-07-09 2007-12-11 Amgen Inc. Substituted anthranilic amide derivatives and methods of use
EP1768674A1 (en) 2004-07-16 2007-04-04 ProteoSys AG Muscarinic antagonists with parp and sir modulating activity as cytoprotective agents
US8247556B2 (en) 2005-10-21 2012-08-21 Amgen Inc. Method for preparing 6-substituted-7-aza-indoles
CN101784263B (zh) 2007-06-08 2012-11-07 贝林格尔.英格海姆国际有限公司 奈韦拉平的延长释放制剂
WO2010081823A1 (en) 2009-01-13 2010-07-22 Proteosys Ag Pirenzepine as otoprotective agent
TW201632520A (zh) 2014-11-25 2016-09-16 拜耳製藥股份有限公司 經取代之吡啶並苯並二氮呯酮衍生物及其用途
EP3153157A1 (en) 2015-10-09 2017-04-12 Teva Pharmaceutical Works Private Limited Company Pharmaceutical composition for prolonged release of nevirapine
CN107382848A (zh) * 2017-07-15 2017-11-24 河北蓝泰化工科技有限公司 一种烟酰胺化合物及其制备方法和应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA554134A (en) * 1958-03-11 Hoffmann Karl Thia-aza-cycloheptadiene compounds and process for their manufacture
CA658624A (en) * 1963-02-26 Schmutz Jean Diazepine derivatives
CA783570A (en) * 1968-04-23 Schmidt Gunther 5,6-dihydro-6-oxo-11h-pyrido (2,3-b) (1,4)-benzodiazepines
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3726908A1 (de) * 1987-08-13 1989-02-23 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3735895A1 (de) * 1987-10-23 1989-05-03 Thomae Gmbh Dr K Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
EP0393529B1 (en) * 1989-04-20 1993-06-30 Boehringer Ingelheim Pharmaceuticals Inc. 5,11-dihydro-6H-dipyrido [3,2-b:2',3'-e][1,4]diazepin-6-ones and their use in the prevention or treatment of AIDS
DE69031845T2 (de) * 1989-04-20 1998-05-07 Boehringer Ingelheim Pharma 6,11-Dihydro-5H-pyrido(2,3-b)(1,5)benzodiazepin-5-one und Thione und ihre Verwendung für die Vorbeugung oder Behandlung von AIDS
ATE103918T1 (de) * 1989-06-28 1994-04-15 Boehringer Ingelheim Pharma 5,11-dihydro-6h-dipyrido(3,2-b:2',3'e>(1,4>diazepin-6-one und -thione und ihre verwendung bei der aids-vorbeugung oder behandlung.

Also Published As

Publication number Publication date
OA09852A (en) 1994-08-15
DE19975051I2 (de) 2004-05-06
NZ236105A (en) 1994-04-27
GR3030100T3 (en) 1999-07-30
LU90393I2 (fr) 1999-06-30
EP0429987B1 (en) 1999-03-17
AU6673290A (en) 1991-05-23
CA2030056A1 (en) 1991-05-18
NL990022I2 (nl) 2007-11-01
NO904986D0 (no) 1990-11-16
FI905674A (fi) 1991-05-18
FI94529B (fi) 1995-06-15
CA2030056C (en) 1995-10-17
NO904986L (no) 1991-05-21
ATE177744T1 (de) 1999-04-15
AP179A (en) 1992-04-30
FI905674A0 (fi) 1990-11-16
DK0429987T3 (da) 1999-10-11
NO1999013I1 (no) 1999-06-29
IL96367A (en) 1997-02-18
PT95919B (pt) 1998-01-30
RU2040527C1 (ru) 1995-07-25
NL990022I1 (nl) 1999-10-01
DE69033003D1 (de) 1999-04-22
PT95919A (pt) 1991-09-13
DE69033003T2 (de) 1999-09-16
HK1011025A1 (en) 1999-07-02
EP0429987A2 (en) 1991-06-05
UA34420C2 (uk) 2001-03-15
ES2130114T3 (es) 1999-07-01
AU630251B2 (en) 1992-10-22
NO175478B (no) 1994-07-11
EP0429987A3 (en) 1992-01-22
FI94529C (fi) 1995-09-25
AP9000224A0 (en) 1991-01-31
IE904141A1 (en) 1991-05-22

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