PT95919A - Processo para a prearacao de 5,11-dihidro-6h-dipirido{3,2-b:2',3'-e}{1,4}diazepinas e de composicoes farmaceuticas que os contem - Google Patents

Processo para a prearacao de 5,11-dihidro-6h-dipirido{3,2-b:2',3'-e}{1,4}diazepinas e de composicoes farmaceuticas que os contem

Info

Publication number
PT95919A
PT95919A PT95919A PT9591990A PT95919A PT 95919 A PT95919 A PT 95919A PT 95919 A PT95919 A PT 95919A PT 9591990 A PT9591990 A PT 9591990A PT 95919 A PT95919 A PT 95919A
Authority
PT
Portugal
Prior art keywords
dipirid
diazepines
dihydro
contain
pharmaceutical compositions
Prior art date
Application number
PT95919A
Other languages
English (en)
Other versions
PT95919B (pt
Inventor
Guenther Schmidt
Wolfhard Engel
Wolfgang Eberlein
Gunter Trummlitz
Original Assignee
Thomae Gmbh Dr K
Boehringer Ingelheim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27412005&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT95919(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Thomae Gmbh Dr K, Boehringer Ingelheim Ltd filed Critical Thomae Gmbh Dr K
Publication of PT95919A publication Critical patent/PT95919A/pt
Publication of PT95919B publication Critical patent/PT95919B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT95919A 1989-11-17 1990-11-16 Processo para a prearacao de 5,11-dihidro-6h-dipirido{3,2-b:2',3'-e}{1,4}diazepinas e de composicoes farmaceuticas que os contem PT95919B (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US43892389A 1989-11-17 1989-11-17
US57900190A 1990-09-06 1990-09-06
US60039090A 1990-10-19 1990-10-19

Publications (2)

Publication Number Publication Date
PT95919A true PT95919A (pt) 1991-09-13
PT95919B PT95919B (pt) 1998-01-30

Family

ID=27412005

Family Applications (1)

Application Number Title Priority Date Filing Date
PT95919A PT95919B (pt) 1989-11-17 1990-11-16 Processo para a prearacao de 5,11-dihidro-6h-dipirido{3,2-b:2',3'-e}{1,4}diazepinas e de composicoes farmaceuticas que os contem

Country Status (21)

Country Link
EP (1) EP0429987B1 (pt)
AP (1) AP179A (pt)
AT (1) ATE177744T1 (pt)
AU (1) AU630251B2 (pt)
CA (1) CA2030056C (pt)
DE (2) DE19975051I2 (pt)
DK (1) DK0429987T3 (pt)
ES (1) ES2130114T3 (pt)
FI (1) FI94529C (pt)
GR (1) GR3030100T3 (pt)
HK (1) HK1011025A1 (pt)
IE (1) IE904141A1 (pt)
IL (1) IL96367A (pt)
LU (1) LU90393I2 (pt)
NL (1) NL990022I2 (pt)
NO (2) NO175478C (pt)
NZ (1) NZ236105A (pt)
OA (1) OA09852A (pt)
PT (1) PT95919B (pt)
RU (1) RU2040527C1 (pt)
UA (1) UA34420C2 (pt)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
GB9109557D0 (en) * 1991-05-02 1991-06-26 Wellcome Found Chemical compounds
US5200522A (en) * 1991-06-11 1993-04-06 Boehringer Ingelheim Pharmaceuticals, Inc. Method for preparing 3-amino-2-chloro-4-alkylpyridines
AU652656B2 (en) * 1991-06-11 1994-09-01 Boehringer Ingelheim Pharmaceuticals, Inc. Method for the preparation of 3-amino-2-chloro-4-alkylpyridines
DE4138908A1 (de) * 1991-11-27 1993-06-03 Bayer Ag 6-thiono-dibenz(b,e)azepine
DE4138853A1 (de) * 1991-11-27 1993-06-03 Bayer Ag 5,6-dihydro-dibenz(b,e)azepin-6,11-dion-11- oxime
ATE170512T1 (de) * 1992-11-18 1998-09-15 Boehringer Ingelheim Pharma Verbesserte methode zur herstellung von 4-alkyl-3-amino-2-chlor-pyridinen
WO1994017075A1 (en) * 1993-01-20 1994-08-04 A. Menarini Industrie Farmaceutiche Riunite S.R.L. Diazepin derivatives and antiviral compositions
DE4333697A1 (de) * 1993-10-02 1995-04-06 Merck Patent Gmbh Verfahren zur Herstellung von 3-Aminopyridinen aus 3-Nitropyridinen
DE4403311C1 (de) * 1994-02-03 1995-04-20 Boehringer Ingelheim Kg Verfahren zur Herstellung von Nevirapine (11-Cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3,2-b:2',3'-e][1,4-diazepin]-6-on)
ES2118575T3 (es) * 1994-02-18 1998-09-16 Boehringer Ingelheim Pharma 2-heteroaril-5,11-dihidro-6h-dipirido(3,2-b:2',3'-e)(1,4)diazepinas y su uso en la prevencion o tratamiento de la infeccion con hiv.
US5917033A (en) * 1995-10-31 1999-06-29 University Of Medicine & Dentistry Of New Jersey Structure based design of inhibitors of HIV-1 reverse transcriptase
US5747488A (en) * 1996-01-30 1998-05-05 Boehringer Ingelheim Pharmaceuticals, Inc. 2-aryl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-E! 1, 4!diazepines and their use in the treatment of HIV infection
ES2265666T3 (es) * 1997-08-25 2007-02-16 Boehringer Ingelheim Pharmaceuticals Inc. Suspension farmaceutica que comprende hemihidrato de nevirapina.
DE10023492A1 (de) * 2000-05-09 2001-11-22 Schering Ag Aza- und Polyazanthranylamide und deren Verwendung als Arzneimittel
US6995162B2 (en) 2001-01-12 2006-02-07 Amgen Inc. Substituted alkylamine derivatives and methods of use
US7102009B2 (en) 2001-01-12 2006-09-05 Amgen Inc. Substituted amine derivatives and methods of use
US7105682B2 (en) 2001-01-12 2006-09-12 Amgen Inc. Substituted amine derivatives and methods of use
US6878714B2 (en) 2001-01-12 2005-04-12 Amgen Inc. Substituted alkylamine derivatives and methods of use
US7307088B2 (en) 2002-07-09 2007-12-11 Amgen Inc. Substituted anthranilic amide derivatives and methods of use
AU2005263577C1 (en) 2004-07-16 2010-08-26 Proteosys Ag Muscarinic antagonists with PARP and SiR modulating activity as cytoprotective agents
US8247556B2 (en) 2005-10-21 2012-08-21 Amgen Inc. Method for preparing 6-substituted-7-aza-indoles
WO2008154234A2 (en) 2007-06-08 2008-12-18 Boehringer Ingelheim International Gmbh Extended release formulation of nevirapine
EP2379080A1 (en) 2009-01-13 2011-10-26 ProteoSys AG Pirenzepine as otoprotective agent
WO2016083276A1 (de) 2014-11-25 2016-06-02 Bayer Pharma Aktiengesellschaft Substituierte pyridobenzodiazepinon-derivate und ihre verwendung
EP3153157A1 (en) 2015-10-09 2017-04-12 Teva Pharmaceutical Works Private Limited Company Pharmaceutical composition for prolonged release of nevirapine
CN107382848A (zh) * 2017-07-15 2017-11-24 河北蓝泰化工科技有限公司 一种烟酰胺化合物及其制备方法和应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA783570A (en) * 1968-04-23 Schmidt Gunther 5,6-dihydro-6-oxo-11h-pyrido (2,3-b) (1,4)-benzodiazepines
CA554134A (en) * 1958-03-11 Hoffmann Karl Thia-aza-cycloheptadiene compounds and process for their manufacture
CA658624A (en) * 1963-02-26 Schmutz Jean Diazepine derivatives
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3726908A1 (de) * 1987-08-13 1989-02-23 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3735895A1 (de) * 1987-10-23 1989-05-03 Thomae Gmbh Dr K Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
EP0393604B1 (en) * 1989-04-20 1997-12-29 Boehringer Ingelheim Pharmaceuticals Inc. 6,11-Dihydro-5H-pyrido(2,3-b)(1,5,)benzodiazepin-5-ones and thiones and their use in the prevention or treatment of AIDS
EP0393529B1 (en) * 1989-04-20 1993-06-30 Boehringer Ingelheim Pharmaceuticals Inc. 5,11-dihydro-6H-dipyrido [3,2-b:2',3'-e][1,4]diazepin-6-ones and their use in the prevention or treatment of AIDS
CA2019812C (en) * 1989-06-28 2000-11-21 Gunther Schmidt (Deceased) Novel 5,11-dihydro-6h-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-ones and their use in the prevention or treatment of aids

Also Published As

Publication number Publication date
EP0429987A3 (en) 1992-01-22
HK1011025A1 (en) 1999-07-02
NZ236105A (en) 1994-04-27
NO904986L (no) 1991-05-21
CA2030056A1 (en) 1991-05-18
AP179A (en) 1992-04-30
FI94529C (fi) 1995-09-25
EP0429987A2 (en) 1991-06-05
IE904141A1 (en) 1991-05-22
FI94529B (fi) 1995-06-15
DE19975051I2 (de) 2004-05-06
GR3030100T3 (en) 1999-07-30
NO175478B (no) 1994-07-11
CA2030056C (en) 1995-10-17
PT95919B (pt) 1998-01-30
DK0429987T3 (da) 1999-10-11
AU6673290A (en) 1991-05-23
ES2130114T3 (es) 1999-07-01
RU2040527C1 (ru) 1995-07-25
LU90393I2 (fr) 1999-06-30
NO904986D0 (no) 1990-11-16
FI905674A (fi) 1991-05-18
FI905674A0 (fi) 1990-11-16
AU630251B2 (en) 1992-10-22
NL990022I1 (nl) 1999-10-01
UA34420C2 (uk) 2001-03-15
NO1999013I1 (no) 1999-06-29
DE69033003D1 (de) 1999-04-22
NL990022I2 (nl) 2007-11-01
DE69033003T2 (de) 1999-09-16
OA09852A (en) 1994-08-15
NO175478C (no) 1994-10-19
EP0429987B1 (en) 1999-03-17
IL96367A (en) 1997-02-18
AP9000224A0 (en) 1991-01-31
ATE177744T1 (de) 1999-04-15

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Legal Events

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BB1A Laying open of patent application

Effective date: 19910405

FG3A Patent granted, date of granting

Effective date: 19971022

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19990430

NF3A Restitutio in integrum

Free format text: 19991111 RESTITUTIO IN INTEGRUM

PC4A Transfer of assignment

Owner name: BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG, DE

Effective date: 20111213

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Effective date: 20121022