PT95522A - Processo para a preparacao de novos compostos tetraciclicos com accao anti-alergica e anti-asmatica e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de novos compostos tetraciclicos com accao anti-alergica e anti-asmatica e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT95522A PT95522A PT95522A PT9552290A PT95522A PT 95522 A PT95522 A PT 95522A PT 95522 A PT95522 A PT 95522A PT 9552290 A PT9552290 A PT 9552290A PT 95522 A PT95522 A PT 95522A
- Authority
- PT
- Portugal
- Prior art keywords
- asmatic
- allergic
- contain
- action
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP26059289 | 1989-10-05 | ||
JP8151390 | 1990-03-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
PT95522A true PT95522A (pt) | 1991-08-14 |
PT95522B PT95522B (pt) | 1997-08-29 |
Family
ID=26422533
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT95522A PT95522B (pt) | 1989-10-05 | 1990-10-04 | Processo para a preparacao de novos compostos tetraciclicos com accao anti-alergica e anti-asmatica e de composicoes farmaceuticas que os contem |
Country Status (11)
Country | Link |
---|---|
US (2) | US5362725A (pt) |
EP (2) | EP0421823A3 (pt) |
KR (1) | KR910007934A (pt) |
CN (1) | CN1030607C (pt) |
CA (1) | CA2026925A1 (pt) |
HU (1) | HUT57771A (pt) |
IE (1) | IE903557A1 (pt) |
NO (1) | NO175781C (pt) |
PT (1) | PT95522B (pt) |
RU (1) | RU2048469C1 (pt) |
TW (1) | TW206227B (pt) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5476848A (en) * | 1989-10-05 | 1995-12-19 | Sankyo Company, Limited | 14B(R) isomers of novel tetracyclic compounds having anti-allergic and anti-asthmatic activities, and their use |
JPH04211071A (ja) * | 1990-03-05 | 1992-08-03 | Hokuriku Seiyaku Co Ltd | 多環式化合物 |
US5470851A (en) * | 1990-06-27 | 1995-11-28 | Sankyo Company, Limited | Thiazolidinecarboxylic acid amide derivatives and their therapeutic uses |
EP0539164A1 (en) * | 1991-10-23 | 1993-04-28 | Sankyo Company Limited | Nitrogen-containing tetracyclic compounds having anti-allergic and anti-asthmatic activities, their preparation and use |
PL183618B1 (pl) * | 1994-11-02 | 2002-06-28 | Janssen Pharmaceutica Nv | Nowy związek, pochodna podstawionej tetracyklicznej oksazepiny lub tiazepiny, kompozycja farmaceutyczna i sposób wytwarzania pochodnej podstawionej tetracyklicznej oksazepiny lub tiazepiny |
US5552399A (en) * | 1994-11-02 | 1996-09-03 | Janssen Pharmaceutica N.V. | Substituted tetracyclic azepine derivatives |
HU221608B (hu) * | 1996-04-12 | 2002-11-28 | Janssen Pharmaceutica N.V. | Izoxazolidinszármazékok |
KR100422254B1 (ko) * | 1996-04-17 | 2004-05-24 | 삼성중공업 주식회사 | 복합지지형수중익선의몰수체 |
EP1017695A4 (en) * | 1997-09-26 | 2002-01-16 | Univ Monash | RESOLUTION OF OPTICALLY ACTIVE COMPOUNDS |
US6187770B1 (en) | 1998-03-17 | 2001-02-13 | Novo Nordisk A/S | N-substituted azaheterocyclic compounds |
US7355042B2 (en) * | 2001-10-16 | 2008-04-08 | Hypnion, Inc. | Treatment of CNS disorders using CNS target modulators |
UA83666C2 (ru) * | 2003-07-10 | 2008-08-11 | Н.В. Органон | Способ получения энантиомерно чистого миртазапина |
JP2009018992A (ja) * | 2007-07-10 | 2009-01-29 | Sumitomo Chemical Co Ltd | 光学活性ミルタザピンの製造方法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL179906C (nl) * | 1974-02-09 | 1986-12-01 | Akzo Nv | Werkwijze voor het bereiden van 1,2,3,4,10,14b-hexahydrodibenzo(c,f)pyrazino (1,2-a)azepine derivaten. |
US4217452A (en) * | 1974-02-09 | 1980-08-12 | Akzona Incorporated | Synthesis for the preparation of tetracyclic compounds |
NL189199C (nl) * | 1975-04-05 | 1993-02-01 | Akzo Nv | Werkwijze ter bereiding van farmaceutische preparaten met werking op het centraal zenuwstelsel op basis van benz(aryl)azepinederivaten, de verkregen gevormde farmaceutische preparaten, alsmede werkwijze ter bereiding van de toe te passen benz(aryl)azepinederivaten. |
ZA784475B (en) * | 1977-10-05 | 1979-07-25 | Ciba Geigy Ag | Piperazinopyrrolobenzodiazepines |
US4271073A (en) * | 1979-11-29 | 1981-06-02 | Cassella Aktiengesellschaft | 6-Substituted-9-(2-hydroxyethyl)-1,2,3,4-tetrahydro carbazol-1-one |
US5049637A (en) * | 1987-04-10 | 1991-09-17 | Monash University | 1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino-[1,2-a]azepino derivatives and 10-aza, 10-oxa and 10-thia analogues |
-
1990
- 1990-10-04 CA CA002026925A patent/CA2026925A1/en not_active Abandoned
- 1990-10-04 NO NO904308A patent/NO175781C/no unknown
- 1990-10-04 IE IE355790A patent/IE903557A1/en unknown
- 1990-10-04 RU SU904831552A patent/RU2048469C1/ru active
- 1990-10-04 TW TW079108315A patent/TW206227B/zh active
- 1990-10-04 PT PT95522A patent/PT95522B/pt not_active IP Right Cessation
- 1990-10-05 EP EP19900310979 patent/EP0421823A3/en not_active Ceased
- 1990-10-05 HU HU906353A patent/HUT57771A/hu unknown
- 1990-10-05 KR KR1019900015834A patent/KR910007934A/ko not_active Application Discontinuation
- 1990-10-05 CN CN90109208A patent/CN1030607C/zh not_active Expired - Fee Related
- 1990-10-05 EP EP19920201652 patent/EP0505014A3/en not_active Withdrawn
-
1992
- 1992-10-15 US US07/962,037 patent/US5362725A/en not_active Expired - Fee Related
-
1994
- 1994-06-28 US US08/267,274 patent/US5461051A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP0505014A2 (en) | 1992-09-23 |
US5461051A (en) | 1995-10-24 |
CN1051360A (zh) | 1991-05-15 |
NO904308L (no) | 1991-04-08 |
EP0421823A3 (en) | 1991-12-18 |
EP0505014A3 (en) | 1993-01-13 |
NO175781C (no) | 1994-12-07 |
TW206227B (pt) | 1993-05-21 |
US5362725A (en) | 1994-11-08 |
CN1030607C (zh) | 1996-01-03 |
CA2026925A1 (en) | 1991-04-06 |
HU906353D0 (en) | 1991-04-29 |
RU2048469C1 (ru) | 1995-11-20 |
EP0421823A2 (en) | 1991-04-10 |
NO175781B (no) | 1994-08-29 |
HUT57771A (en) | 1991-12-30 |
NO904308D0 (no) | 1990-10-04 |
IE903557A1 (en) | 1991-04-10 |
PT95522B (pt) | 1997-08-29 |
KR910007934A (ko) | 1991-05-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
BB1A | Laying open of patent application |
Effective date: 19910313 |
|
MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19981130 |