NL8001919A - Werkwijze voor het bereiden van beta-lactamaseremmers. - Google Patents

Werkwijze voor het bereiden van beta-lactamaseremmers. Download PDF

Info

Publication number
NL8001919A
NL8001919A NL8001919A NL8001919A NL8001919A NL 8001919 A NL8001919 A NL 8001919A NL 8001919 A NL8001919 A NL 8001919A NL 8001919 A NL8001919 A NL 8001919A NL 8001919 A NL8001919 A NL 8001919A
Authority
NL
Netherlands
Prior art keywords
formula
compound
group
meaning
benzyl
Prior art date
Application number
NL8001919A
Other languages
English (en)
Dutch (nl)
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NL8001919A publication Critical patent/NL8001919A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568—Four-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Cephalosporin Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NL8001919A 1979-04-06 1980-04-01 Werkwijze voor het bereiden van beta-lactamaseremmers. NL8001919A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7912168 1979-04-06
GB7912168 1979-04-06

Publications (1)

Publication Number Publication Date
NL8001919A true NL8001919A (nl) 1980-10-08

Family

ID=10504396

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8001919A NL8001919A (nl) 1979-04-06 1980-04-01 Werkwijze voor het bereiden van beta-lactamaseremmers.

Country Status (24)

Country Link
US (1) US4269771A (cs)
JP (1) JPS55139385A (cs)
AT (1) AT369371B (cs)
AU (1) AU536673B2 (cs)
BE (1) BE882621A (cs)
CA (1) CA1148143A (cs)
CH (1) CH645645A5 (cs)
CS (1) CS219273B2 (cs)
DE (1) DE3012975A1 (cs)
DK (1) DK144180A (cs)
FI (1) FI801080A7 (cs)
FR (1) FR2453162A1 (cs)
GB (1) GB2048857B (cs)
GR (1) GR66673B (cs)
HU (1) HU182118B (cs)
IE (1) IE49656B1 (cs)
IL (1) IL59760A (cs)
IT (1) IT1196407B (cs)
LU (1) LU82320A1 (cs)
NL (1) NL8001919A (cs)
SE (1) SE8002600L (cs)
SU (1) SU1152524A3 (cs)
YU (1) YU93880A (cs)
ZA (1) ZA802000B (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4500457A (en) * 1977-05-09 1985-02-19 Ciba-Geigy Corporation Process for preparing thia-aza compounds with a beta-lactam ring
AT365594B (de) * 1978-11-24 1982-01-25 Erba Farmitalia Verfahren zur herstellung von neuen 7-oxo-4-thia1-aza-bicyclo-(3,2,0)heptanderivaten
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
US4347183A (en) * 1981-02-02 1982-08-31 Schering Corporation Process for the synthesis of penems and carbapenems
US4508649A (en) * 1981-12-11 1985-04-02 Farmitalia Carlo Erba Process for preparing optically active penems
NO831160L (no) * 1982-04-08 1983-10-10 Erba Farmitalia Fremstilling av substituerte penem-derivater
GB8321677D0 (en) * 1983-08-11 1983-09-14 Erba Farmitalia Preparation of penems
US6720445B2 (en) 2000-12-21 2004-04-13 Beacon Laboratories, Inc. Acetyloxymethyl esters and methods for using the same

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3905965A (en) * 1969-10-17 1975-09-16 Roussel Uclaf Process of total synthesis of cephalosporin derivatives and intermediates
US4053468A (en) * 1976-02-25 1977-10-11 Smithkline Corporation Process for preparing 7-oxo cephalosporins and 6-oxo penicillins
LU77306A1 (cs) 1977-05-09 1979-01-18
EP0000636A1 (en) * 1977-07-13 1979-02-07 Glaxo Group Limited Penem compounds, processes for their preparation, their use in pharmaceutical compositions and azetidinones used in their preparation
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
US4155912A (en) * 1977-12-14 1979-05-22 Bristol-Myers Company 2-Methylpenem-3-carboxylic acid antibiotics
EP0003415A3 (en) * 1978-01-20 1979-08-22 Glaxo Group Limited Beta-lactam compounds, processes for their preparation,compositions containing them and intermediates of use in their preparation
GB2014574A (en) * 1978-02-16 1979-08-30 Glaxo Group Ltd Lactam Compounds
JPS5559193A (en) * 1978-09-20 1980-05-02 Glaxo Group Ltd Bblactam compound

Also Published As

Publication number Publication date
CA1148143A (en) 1983-06-14
DK144180A (da) 1980-10-07
YU93880A (en) 1983-02-28
IT8021099A0 (it) 1980-04-01
CH645645A5 (de) 1984-10-15
ZA802000B (en) 1981-04-29
DE3012975A1 (de) 1980-10-23
GR66673B (cs) 1981-04-08
IE800668L (en) 1980-10-06
SE8002600L (sv) 1980-10-07
AU536673B2 (en) 1984-05-17
FR2453162A1 (fr) 1980-10-31
IE49656B1 (en) 1985-11-13
IL59760A (en) 1983-07-31
IL59760A0 (en) 1980-06-30
GB2048857B (en) 1983-05-25
AU5701580A (en) 1980-10-09
BE882621A (fr) 1980-10-03
CS219273B2 (en) 1983-03-25
US4269771A (en) 1981-05-26
GB2048857A (en) 1980-12-17
AT369371B (de) 1982-12-27
JPS55139385A (en) 1980-10-31
HU182118B (en) 1983-12-28
LU82320A1 (fr) 1980-07-02
SU1152524A3 (en) 1985-04-23
IT1196407B (it) 1988-11-16
FI801080A7 (fi) 1981-01-01
ATA177480A (de) 1982-05-15

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BV The patent application has lapsed