NL193340C - Farmaceutisch preparaat voor parenterale toediening gevormd uit een vetemulsie. - Google Patents
Farmaceutisch preparaat voor parenterale toediening gevormd uit een vetemulsie. Download PDFInfo
- Publication number
- NL193340C NL193340C NL8802657A NL8802657A NL193340C NL 193340 C NL193340 C NL 193340C NL 8802657 A NL8802657 A NL 8802657A NL 8802657 A NL8802657 A NL 8802657A NL 193340 C NL193340 C NL 193340C
- Authority
- NL
- Netherlands
- Prior art keywords
- sample
- emulsion
- drug
- dexamethasone
- active compound
- Prior art date
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- HYVJNYYVNIYMDK-QSEXIABDSA-N triarachidonin Chemical compound CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)OCC(OC(=O)CCC\C=C/C\C=C/C\C=C/C\C=C/CCCCC)COC(=O)CCC\C=C/C\C=C/C\C=C/C\C=C/CCCCC HYVJNYYVNIYMDK-QSEXIABDSA-N 0.000 description 1
- 150000005691 triesters Chemical class 0.000 description 1
- 229940081852 trilinolein Drugs 0.000 description 1
- 229940113164 trimyristin Drugs 0.000 description 1
- 229960001947 tripalmitin Drugs 0.000 description 1
- 235000015112 vegetable and seed oil Nutrition 0.000 description 1
- 239000008158 vegetable oil Substances 0.000 description 1
- 239000003981 vehicle Substances 0.000 description 1
- 229940088594 vitamin Drugs 0.000 description 1
- 239000011782 vitamin Substances 0.000 description 1
- 229930003231 vitamin Natural products 0.000 description 1
- 235000013343 vitamin Nutrition 0.000 description 1
- GVJHHUAWPYXKBD-IEOSBIPESA-N α-tocopherol Chemical compound OC1=C(C)C(C)=C2O[C@@](CCC[C@H](C)CCC[C@H](C)CCCC(C)C)(C)CCC2=C1C GVJHHUAWPYXKBD-IEOSBIPESA-N 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Dispersion Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Materials For Medical Uses (AREA)
- Lubricants (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP27277087 | 1987-10-28 | ||
| JP27277087 | 1987-10-28 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NL8802657A NL8802657A (nl) | 1989-05-16 |
| NL193340B NL193340B (nl) | 1999-03-01 |
| NL193340C true NL193340C (nl) | 1999-07-02 |
Family
ID=17518498
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL8802657A NL193340C (nl) | 1987-10-28 | 1988-10-28 | Farmaceutisch preparaat voor parenterale toediening gevormd uit een vetemulsie. |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0315079B1 (de) |
| KR (1) | KR960013281B1 (de) |
| CN (1) | CN1048182C (de) |
| AT (1) | ATE119031T1 (de) |
| AU (1) | AU623342B2 (de) |
| BE (1) | BE1001760A5 (de) |
| CA (1) | CA1333993C (de) |
| CH (1) | CH677605A5 (de) |
| DE (1) | DE3853191T2 (de) |
| ES (1) | ES2012561A6 (de) |
| FR (1) | FR2622442B1 (de) |
| GB (1) | GB2211408B (de) |
| IL (1) | IL88076A (de) |
| IT (1) | IT1224596B (de) |
| NL (1) | NL193340C (de) |
Families Citing this family (41)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR0148748B1 (ko) | 1988-09-16 | 1998-08-17 | 장 크라메르, 한스 루돌프 하우스 | 사이클로스포린을 함유하는 약학조성물 |
| US6007840A (en) * | 1988-09-16 | 1999-12-28 | Novartis Ag | Pharmaceutical compositions comprising cyclosporins |
| ES2052016T3 (es) * | 1988-09-29 | 1994-07-01 | Shiseido Co Ltd | Composicion emulsionada. |
| JP2785981B2 (ja) * | 1989-11-20 | 1998-08-13 | 株式会社資生堂 | 乳化組成物 |
| TW211015B (de) * | 1990-01-11 | 1993-08-11 | Nippon Shinyaku Co Ltd | |
| AU665931B2 (en) * | 1990-11-06 | 1996-01-25 | Nippon Shinyaku Co. Ltd. | Lyophilized preparation and production thereof |
| US6262022B1 (en) | 1992-06-25 | 2001-07-17 | Novartis Ag | Pharmaceutical compositions containing cyclosporin as the active agent |
| IL101387A (en) * | 1992-03-26 | 1999-11-30 | Pharmos Ltd | Emulsion with enhanced topical and/or transdermal systemic effect utilizing submicron oil droplets |
| BR9201168A (pt) * | 1992-04-02 | 1994-04-12 | Zerbini E J Fundacao | Microemulsoes usadas como velculo para carregar quimioterapicos as celulas neoplasicas |
| HK1004520A1 (en) | 1992-05-13 | 1998-11-27 | Novartis Ag | Ophthalmic compositions containing a cyclosporin |
| PT589843E (pt) | 1992-09-25 | 2002-04-29 | Novartis Ag | Composicoes farmaceuticas contendo ciclosporinas |
| US6113921A (en) * | 1993-03-23 | 2000-09-05 | Pharmos Corp. | Topical and transdermal delivery system utilizing submicron oil spheres |
| US5576016A (en) * | 1993-05-18 | 1996-11-19 | Pharmos Corporation | Solid fat nanoemulsions as drug delivery vehicles |
| US5961970A (en) * | 1993-10-29 | 1999-10-05 | Pharmos Corporation | Submicron emulsions as vaccine adjuvants |
| FI963297L (fi) * | 1994-02-25 | 1996-10-18 | Takeda Chemical Industries Ltd | Antifungaalisia triatsolijohdannaisia sisältävät emulsiot |
| US5851510A (en) * | 1994-05-16 | 1998-12-22 | The Board Of Regents Of The University Of Michigan | Hepatocyte-selective oil-in-water emulsion |
| SK164796A3 (en) | 1994-11-03 | 1997-06-04 | Dresden Arzneimittel | Novel cyclosporine preparation forms for oral administration of and process for producing them |
| EP0808154B1 (de) * | 1995-02-06 | 2000-12-20 | Elan Pharma International Limited | Formulierungen von verbindungen als nanopartikel dispergiert in verdaubaren ölen oder fettsäuren |
| DE19544507B4 (de) | 1995-11-29 | 2007-11-15 | Novartis Ag | Cyclosporin enthaltende Präparate |
| GB9601120D0 (en) | 1996-01-19 | 1996-03-20 | Sandoz Ltd | Organic compounds |
| JP3136352B2 (ja) * | 1996-01-22 | 2001-02-19 | 参天製薬株式会社 | 角結膜疾患治療剤 |
| TR199802769T2 (xx) * | 1996-07-02 | 1999-04-21 | Novartis Consumer Health S.A. | Terpenoid bileşikler ile antihistaminik bileşiklerin bir kombinasyonunu ihtiva eden topikal bileşim. |
| SK285019B6 (sk) | 1997-01-30 | 2006-04-06 | Novartis Ag | Tvrdá želatínová tobolka |
| US6537561B1 (en) | 1997-02-27 | 2003-03-25 | Nippon Shinyaku Co., Ltd. | Fat emulsion for oral administration |
| IL121647A (en) * | 1997-08-28 | 2001-07-24 | Pharmateam Dev Ltd | Pharmaceutical compositions for the treatment of ocular inflammation comprising dexamethasone palmitate |
| GR20020100012A (el) * | 2002-01-16 | 2003-09-24 | Αγγελικη Κουρουνακη | Το γουαιαζουλενιο για χρηση στην προληψη ή θεραπεια καθε τυπου υπερχοληστερολαιμιας, υπερλιπιδαιμιας και καθε διαταραχη λιπιδιων, σε ανθρωπους και ζωα |
| CN1297271C (zh) * | 2003-09-30 | 2007-01-31 | 昆明紫健生物技术有限公司 | 草乌甲素脂肪乳输液及其生产方法 |
| CN100386085C (zh) * | 2003-12-17 | 2008-05-07 | 昆明紫健生物技术有限公司 | 一种防治肿瘤的脂肪乳输液及生产方法 |
| US7871632B2 (en) * | 2004-07-12 | 2011-01-18 | Adventrx Pharmaceuticals, Inc. | Compositions for delivering highly water soluble drugs |
| US20080274195A1 (en) | 2005-07-18 | 2008-11-06 | University Of Massachusetts Lowell | Compositions and Methods for Making and Using Nanoemulsions |
| US9486408B2 (en) | 2005-12-01 | 2016-11-08 | University Of Massachusetts Lowell | Botulinum nanoemulsions |
| SG177184A1 (en) | 2006-12-01 | 2012-01-30 | Anterios Inc | Amphiphilic entity nanoparticles |
| SG179457A1 (en) | 2006-12-01 | 2012-04-27 | Anterios Inc | Peptide nanoparticles and uses therefor |
| CN101765423B (zh) | 2007-05-31 | 2014-08-06 | 安特里奥公司 | 核酸纳米粒子和其用途 |
| WO2010079037A2 (de) * | 2008-12-18 | 2010-07-15 | Basf Se | Wässrige dispersion umfassend pestizidpartikel und amphiphil |
| DE102010021688A1 (de) * | 2010-05-27 | 2011-12-01 | Qineva Gmbh & Co. Kg | Verfahren zur Herstellung eines micellaren Wirkstoffkonzentrats |
| JP6166480B2 (ja) * | 2013-12-11 | 2017-07-19 | ヘルス−エバー バイオテック カンパニー リミテッド | カロテノイドの医薬組成物 |
| CN105483076B (zh) | 2015-12-23 | 2019-01-25 | 中国科学院生物物理研究所 | 一种脂肪体的制备方法及其应用 |
| MX2019005833A (es) | 2016-11-21 | 2019-10-30 | Eirion Therapeutics Inc | Administracion transdermica de agentes grandes. |
| WO2023178519A1 (zh) * | 2022-03-22 | 2023-09-28 | 乐普（北京）医疗器械股份有限公司 | 一种药物涂层、药物球囊及药物球囊制备方法与应用 |
| CN115919759B (zh) * | 2022-12-27 | 2025-03-18 | 沈阳药科大学 | 一种低聚集体眼用纳米制剂及其制备方法和用途 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2502951B1 (fr) * | 1981-04-06 | 1985-12-06 | Sandoz Sa | Compositions pharmaceutiques topiques sous forme d'une micro-emulsion |
| DE3225848A1 (de) * | 1982-07-07 | 1984-01-19 | Schering AG, 1000 Berlin und 4709 Bergkamen | Kortikoidhaltige zubereitung zur topischen applikation |
| DE3225706C2 (de) * | 1982-07-09 | 1984-04-26 | A. Nattermann & Cie GmbH, 5000 Köln | Flüssige Wirkstofformulierungen in Form von Konzentraten für Mikroemulsionen |
| JPS59193814A (ja) * | 1983-04-20 | 1984-11-02 | Ajinomoto Co Inc | アミノ酸含有脂肪乳剤 |
| JPS60231609A (ja) * | 1984-04-28 | 1985-11-18 | Terumo Corp | リポソ−ム製剤 |
| DE3421468A1 (de) * | 1984-06-08 | 1985-12-19 | Dr. Rentschler Arzneimittel Gmbh & Co, 7958 Laupheim | Lipidnanopellets als traegersystem fuer arzneimittel zur peroralen anwendung |
| DK482685D0 (da) * | 1984-10-22 | 1985-10-21 | Hope Nat Medical Center | Fremgangsmaade til tilfoersel af micellulaere partikler, der indkapslerbilleddannende og kemoterapeutiske midler, til tumorer i et legeme |
| US4753788A (en) * | 1985-01-31 | 1988-06-28 | Vestar Research Inc. | Method for preparing small vesicles using microemulsification |
| IL78929A0 (en) * | 1985-07-29 | 1986-09-30 | Abbott Lab | Microemulsion compositions for parenteral administration |
| US5023271A (en) * | 1985-08-13 | 1991-06-11 | California Biotechnology Inc. | Pharmaceutical microemulsions |
| JPS6348214A (ja) * | 1986-08-18 | 1988-02-29 | Morishita Seiyaku Kk | １−〔２−（２，４−ジクロロフエニル）−３−メチル−１−ペンテニル〕−１ｈ−イミダゾ−ルを含有する水中油型脂肪乳剤 |
| FR2608942B1 (fr) * | 1986-12-31 | 1991-01-11 | Centre Nat Rech Scient | Procede de preparation de systemes colloidaux dispersibles d'une substance, sous forme de nanocapsules |
-
1988
- 1988-10-18 IL IL88076A patent/IL88076A/xx not_active IP Right Cessation
- 1988-10-26 GB GB8825024A patent/GB2211408B/en not_active Expired - Fee Related
- 1988-10-27 ES ES8803282A patent/ES2012561A6/es not_active Expired - Fee Related
- 1988-10-27 CN CN88107466A patent/CN1048182C/zh not_active Expired - Fee Related
- 1988-10-27 BE BE8801239A patent/BE1001760A5/fr not_active IP Right Cessation
- 1988-10-27 IT IT8848502A patent/IT1224596B/it active
- 1988-10-28 AU AU24472/88A patent/AU623342B2/en not_active Ceased
- 1988-10-28 CH CH4018/88A patent/CH677605A5/fr not_active IP Right Cessation
- 1988-10-28 CA CA000581659A patent/CA1333993C/en not_active Expired - Fee Related
- 1988-10-28 AT AT88118025T patent/ATE119031T1/de not_active IP Right Cessation
- 1988-10-28 NL NL8802657A patent/NL193340C/nl not_active IP Right Cessation
- 1988-10-28 EP EP88118025A patent/EP0315079B1/de not_active Expired - Lifetime
- 1988-10-28 FR FR8814209A patent/FR2622442B1/fr not_active Expired - Fee Related
- 1988-10-28 KR KR1019880014049A patent/KR960013281B1/ko not_active Expired - Fee Related
- 1988-10-28 DE DE3853191T patent/DE3853191T2/de not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CN1042080A (zh) | 1990-05-16 |
| CA1333993C (en) | 1995-01-17 |
| GB8825024D0 (en) | 1988-11-30 |
| DE3853191T2 (de) | 1995-10-19 |
| ATE119031T1 (de) | 1995-03-15 |
| ES2012561A6 (es) | 1990-04-01 |
| BE1001760A5 (fr) | 1990-02-27 |
| EP0315079A1 (de) | 1989-05-10 |
| FR2622442A1 (fr) | 1989-05-05 |
| KR890006225A (ko) | 1989-06-12 |
| FR2622442B1 (fr) | 1993-10-22 |
| GB2211408A (en) | 1989-07-05 |
| AU2447288A (en) | 1989-05-04 |
| IL88076A0 (en) | 1989-06-30 |
| IT8848502A0 (it) | 1988-10-27 |
| IL88076A (en) | 1993-01-14 |
| AU623342B2 (en) | 1992-05-14 |
| IT1224596B (it) | 1990-10-04 |
| NL8802657A (nl) | 1989-05-16 |
| CH677605A5 (de) | 1991-06-14 |
| EP0315079B1 (de) | 1995-03-01 |
| DE3853191D1 (de) | 1995-04-06 |
| KR960013281B1 (ko) | 1996-10-02 |
| CN1048182C (zh) | 2000-01-12 |
| GB2211408B (en) | 1992-04-15 |
| NL193340B (nl) | 1999-03-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A1B | A search report has been drawn up | ||
| BC | A request for examination has been filed | ||
| V1 | Lapsed because of non-payment of the annual fee |
Effective date: 20050501 |