NL1017414C1 - Werkwijze voor de bereiding van Citalopram. - Google Patents

Werkwijze voor de bereiding van Citalopram. Download PDF

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Publication number
NL1017414C1
NL1017414C1 NL1017414A NL1017414A NL1017414C1 NL 1017414 C1 NL1017414 C1 NL 1017414C1 NL 1017414 A NL1017414 A NL 1017414A NL 1017414 A NL1017414 A NL 1017414A NL 1017414 C1 NL1017414 C1 NL 1017414C1
Authority
NL
Netherlands
Prior art keywords
formula
compound
citalopram
acid
prepared
Prior art date
Application number
NL1017414A
Other languages
English (en)
Dutch (nl)
Inventor
Hans Petersen
Michael Harold Rock
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8159208&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NL1017414(C1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Application granted granted Critical
Publication of NL1017414C1 publication Critical patent/NL1017414C1/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Steroid Compounds (AREA)
  • Furan Compounds (AREA)
NL1017414A 2000-02-24 2001-02-21 Werkwijze voor de bereiding van Citalopram. NL1017414C1 (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK200000296 2000-02-24
DKPA200000296 2000-02-24

Publications (1)

Publication Number Publication Date
NL1017414C1 true NL1017414C1 (nl) 2001-03-15

Family

ID=8159208

Family Applications (1)

Application Number Title Priority Date Filing Date
NL1017414A NL1017414C1 (nl) 2000-02-24 2001-02-21 Werkwijze voor de bereiding van Citalopram.

Country Status (29)

Country Link
US (3) US20020004604A1 (https=)
EP (1) EP1259500A1 (https=)
JP (1) JP2003524009A (https=)
KR (1) KR20020080438A (https=)
CN (1) CN1161350C (https=)
AU (1) AU2001235357A1 (https=)
BE (1) BE1012921A6 (https=)
BG (1) BG107015A (https=)
BR (1) BR0108947A (https=)
CA (1) CA2400682A1 (https=)
EA (1) EA005593B1 (https=)
FR (1) FR2805813A1 (https=)
GR (1) GR20010100097A (https=)
HK (1) HK1054378B (https=)
HR (1) HRP20020743A2 (https=)
HU (1) HUP0300078A3 (https=)
IE (1) IES20010143A2 (https=)
IL (1) IL151339A0 (https=)
IS (1) IS6512A (https=)
IT (1) ITMI20010385A1 (https=)
MX (1) MXPA02008230A (https=)
NL (1) NL1017414C1 (https=)
NO (1) NO20024007L (https=)
PL (1) PL357178A1 (https=)
SK (1) SK13662002A3 (https=)
TR (1) TR200202048T2 (https=)
UA (1) UA71059C2 (https=)
WO (1) WO2001062754A1 (https=)
ZA (2) ZA200206255B (https=)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
DK1173431T4 (da) 1999-04-14 2010-01-04 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
ITMI991581A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
HRP20020344B1 (hr) 1999-10-25 2010-10-31 H. Lundbeck A/S Način priprave citaloprama
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
HUP0203635A3 (en) 1999-12-28 2005-02-28 Lundbeck & Co As H Method for the preparation of citalopram
PT1246813E (pt) 1999-12-30 2004-02-27 Lundbeck & Co As H Metodo para a preparacao de citalopram
CN1195749C (zh) * 2000-01-14 2005-04-06 H.隆德贝克有限公司 制备5－氰基2－苯并[c]呋喃酮的方法
US6433196B1 (en) 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017417C1 (nl) 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en) 2000-03-07 2000-04-26 Resolution Chemicals Limited Process for the preparation of citalopram
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
KR20020080481A (ko) 2000-03-13 2002-10-23 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
CN1427835A (zh) 2000-03-13 2003-07-02 H·隆德贝克有限公司 5－取代的1－(4－氟苯基)－1,3－二氢异苯并呋喃的分步烷基化
TR200202155T2 (tr) 2000-03-14 2002-12-23 H. Lundbeck A/S Sitalopramin preparasyon metodu
DE10190485T1 (de) * 2000-03-16 2002-03-21 Lundbeck & Co As H Verfahren zur Herstellung von 5-Cyano-1-(4-fluorphenyl)-1,3-dihydroisobenzofuranen
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
CA2354877C (en) 2000-08-18 2006-05-02 H. Lundbeck A/S Method for the preparation of citalopram
WO2001045483A2 (en) 2000-12-22 2001-06-28 H. Lundbeck A/S Method for the preparation of pure citalopram
DK1281707T3 (da) * 2001-08-02 2005-05-02 Infosint Sa Fremgangsmåde til fremstilling af 5-substituerede isobenzenfuraner
WO2004016602A1 (en) * 2002-08-14 2004-02-26 Natco Pharma Limited Process for the preparation of high purity citalopram and its pharmaceutically acceptable salts
US8539533B2 (en) * 2003-03-07 2013-09-17 Siemens Enterprise Communications, Inc. System and method for digital personal video stream manager
WO2004085416A1 (en) * 2003-03-24 2004-10-07 Hetero Drugs Limited Novel crystalline forms of (s)-citalopram oxalate
CN100569765C (zh) 2003-12-19 2009-12-16 杭州民生药业集团有限公司 西酞普兰中间体晶体碱
JP2006176490A (ja) * 2004-11-29 2006-07-06 Sumitomo Chemical Co Ltd ５−フタランカルボニトリル及びシタロプラムの製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
UA62985C2 (en) * 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
DK1173431T4 (da) * 1999-04-14 2010-01-04 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
US6310222B1 (en) * 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) * 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate

Also Published As

Publication number Publication date
BR0108947A (pt) 2003-06-03
CN1161350C (zh) 2004-08-11
HUP0300078A2 (en) 2003-05-28
UA71059C2 (uk) 2004-11-15
HK1054378B (zh) 2005-04-29
ZA200206255B (en) 2003-10-20
CN1404475A (zh) 2003-03-19
JP2003524009A (ja) 2003-08-12
AU2001235357A1 (en) 2001-09-03
IL151339A0 (en) 2003-04-10
FR2805813A1 (fr) 2001-09-07
EA200200900A1 (ru) 2003-02-27
IES20010143A2 (en) 2001-07-25
US20030114692A1 (en) 2003-06-19
HUP0300078A3 (en) 2005-02-28
US20030083508A1 (en) 2003-05-01
TR200202048T2 (tr) 2003-01-21
BE1012921A6 (fr) 2001-05-08
CA2400682A1 (en) 2001-08-30
SK13662002A3 (sk) 2003-01-09
PL357178A1 (en) 2004-07-26
KR20020080438A (ko) 2002-10-23
US20020004604A1 (en) 2002-01-10
IS6512A (is) 2002-08-20
GR20010100097A (el) 2001-10-31
EA005593B1 (ru) 2005-04-28
HK1054378A1 (en) 2003-11-28
NO20024007D0 (no) 2002-08-22
BG107015A (bg) 2003-05-30
ITMI20010385A1 (it) 2002-08-26
ZA200206699B (en) 2003-11-21
WO2001062754A1 (en) 2001-08-30
EP1259500A1 (en) 2002-11-27
MXPA02008230A (es) 2003-05-23
HRP20020743A2 (en) 2003-12-31
NO20024007L (no) 2002-10-07

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Publication Publication Date Title
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Legal Events

Date Code Title Description
VD2 Discontinued due to expiration of the term of protection

Effective date: 20070221