NI201100102A - 3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas. - Google Patents

3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas.

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Publication number
NI201100102A
NI201100102A NI201100102A NI201100102A NI201100102A NI 201100102 A NI201100102 A NI 201100102A NI 201100102 A NI201100102 A NI 201100102A NI 201100102 A NI201100102 A NI 201100102A NI 201100102 A NI201100102 A NI 201100102A
Authority
NI
Nicaragua
Prior art keywords
aminociclopentancarboxamide
receptor modulators
chemokines receptor
chemokines
compound
Prior art date
Application number
NI201100102A
Other languages
English (en)
Spanish (es)
Inventor
Venkateswaran Devraj Rajesh
Joseph Rogier Donald Jr
Huang Wei
Owen Hughes Robert
Isidro Trujillo John
Ronald Turner Steve
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NI201100102A publication Critical patent/NI201100102A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Nutrition Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Transplantation (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
NI201100102A 2008-11-26 2011-05-24 3 - aminociclopentancarboxamida como moduladores del receptor de quimioquinas. NI201100102A (es)

Applications Claiming Priority (1)

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US11805308P 2008-11-26 2008-11-26

Publications (1)

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NI201100102A true NI201100102A (es) 2011-09-27

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EP (1) EP2370442B9 (https=)
JP (1) JP5108153B2 (https=)
KR (1) KR101374412B1 (https=)
CN (1) CN102227429B (https=)
AP (1) AP3113A (https=)
AU (1) AU2009321221B2 (https=)
BR (1) BRPI0920936A2 (https=)
CA (1) CA2743030C (https=)
CL (1) CL2011001223A1 (https=)
CO (1) CO6361921A2 (https=)
CR (1) CR20110275A (https=)
CU (1) CU24022B1 (https=)
CY (1) CY1114020T1 (https=)
DK (1) DK2370442T5 (https=)
DO (1) DOP2011000154A (https=)
EA (1) EA020470B1 (https=)
EC (1) ECSP11011081A (https=)
ES (1) ES2415430T3 (https=)
GE (1) GEP20146064B (https=)
HR (1) HRP20130409T2 (https=)
IL (1) IL212732A (https=)
MA (1) MA32834B1 (https=)
ME (1) ME01144B (https=)
MX (1) MX2011005526A (https=)
MY (1) MY152557A (https=)
NI (1) NI201100102A (https=)
NZ (1) NZ592919A (https=)
PE (1) PE20110831A1 (https=)
PL (1) PL2370442T3 (https=)
PT (1) PT2370442E (https=)
RS (1) RS52810B8 (https=)
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EP2370442B9 (en) * 2008-11-26 2013-09-04 Pfizer Inc. 3-Aminocyclopentanecarboxamides as chemokine receptor modulators
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WO2016010131A1 (ja) * 2014-07-17 2016-01-21 参天製薬株式会社 加齢黄斑変性の予防または治療剤
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TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲(江蘇)醫藥有限公司 環戊烷化合物

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AU2009321221A1 (en) 2010-06-03
PT2370442E (pt) 2013-06-27
US20110144129A1 (en) 2011-06-16
EP2370442B1 (en) 2013-04-24
EP2370442A1 (en) 2011-10-05
US8293903B2 (en) 2012-10-23
ES2415430T3 (es) 2013-07-25
JP2012509931A (ja) 2012-04-26
KR20110075036A (ko) 2011-07-05
JP5108153B2 (ja) 2012-12-26
TN2011000254A1 (fr) 2012-12-17
DK2370442T5 (da) 2013-09-23
CL2011001223A1 (es) 2011-09-02
EA020470B1 (ru) 2014-11-28
AP3113A (en) 2015-01-31
US20130197008A1 (en) 2013-08-01
CN102227429A (zh) 2011-10-26
HRP20130409T1 (en) 2013-06-30
ES2415430T9 (es) 2013-11-25
NZ592919A (en) 2013-05-31
ZA201104069B (en) 2012-02-29
HRP20130409T2 (hr) 2013-11-22
CY1114020T1 (el) 2016-07-27
HK1161261A1 (en) 2012-08-24
CA2743030C (en) 2013-10-22
CR20110275A (es) 2011-07-01
CU24022B1 (es) 2014-07-30
CN102227429B (zh) 2014-05-28
SI2370442T1 (sl) 2013-06-28
RS52810B (sr) 2013-10-31
SV2011003923A (es) 2011-07-28
GEP20146064B (en) 2014-03-25
IL212732A0 (en) 2011-07-31
AU2009321221B2 (en) 2013-04-04
IL212732A (en) 2016-06-30
UA99978C2 (en) 2012-10-25
BRPI0920936A2 (pt) 2020-08-11
RS52810B8 (sr) 2019-08-30
KR101374412B1 (ko) 2014-03-17
DOP2011000154A (es) 2011-07-31
CA2743030A1 (en) 2010-06-03
ME01144B (me) 2013-03-20
MA32834B1 (fr) 2011-11-01
MX2011005526A (es) 2011-06-06
CO6361921A2 (es) 2012-01-20
WO2010061329A1 (en) 2010-06-03
EP2370442B9 (en) 2013-09-04
DK2370442T3 (da) 2013-06-17
US8946413B2 (en) 2015-02-03
CU20110121A7 (es) 2013-05-31
MY152557A (en) 2014-10-31
RS52810B9 (sr) 2019-06-28
ECSP11011081A (es) 2011-12-30
EA201170721A1 (ru) 2011-12-30
PL2370442T3 (pl) 2013-08-30
AP2011005732A0 (en) 2011-06-30
PE20110831A1 (es) 2011-11-20

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