NI200700068A - Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo - Google Patents

Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo

Info

Publication number
NI200700068A
NI200700068A NI200700068A NI200700068A NI200700068A NI 200700068 A NI200700068 A NI 200700068A NI 200700068 A NI200700068 A NI 200700068A NI 200700068 A NI200700068 A NI 200700068A NI 200700068 A NI200700068 A NI 200700068A
Authority
NI
Nicaragua
Prior art keywords
amino
cyanoethenyl
benzonitrile
dimethylphenyl
pyrimidinyl
Prior art date
Application number
NI200700068A
Other languages
English (en)
Spanish (es)
Inventor
Theodoor Agnes Stevens Paul
Peeters Jozef
Petrus Gerebern Vandecruys Roger
Elisabeth Stappers Alfred
Herman Copmans Alex
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38091637&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NI200700068(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from MYPI20043578A external-priority patent/MY169670A/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NI200700068A publication Critical patent/NI200700068A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Hybrid Cells (AREA)
NI200700068A 2004-09-02 2007-03-01 Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo NI200700068A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
MYPI20043578A MY169670A (en) 2003-09-03 2004-09-02 Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors
EP05101467 2005-02-25

Publications (1)

Publication Number Publication Date
NI200700068A true NI200700068A (es) 2016-09-29

Family

ID=38091637

Family Applications (1)

Application Number Title Priority Date Filing Date
NI200700068A NI200700068A (es) 2004-09-02 2007-03-01 Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo

Country Status (23)

Country Link
EP (1) EP1632232B3 (https=)
JP (1) JP4912309B2 (https=)
KR (1) KR101284361B1 (https=)
CN (1) CN104586850A (https=)
AT (1) ATE508748T1 (https=)
BR (1) BRPI0514871A (https=)
CY (3) CY1112249T1 (https=)
DK (1) DK1632232T6 (https=)
EA (1) EA013686B1 (https=)
ES (1) ES2371442T7 (https=)
FR (2) FR16C1023I2 (https=)
HK (1) HK1210029A1 (https=)
HU (2) HUS1600061I1 (https=)
IL (1) IL181650A (https=)
LT (2) LTC1632232I2 (https=)
ME (1) ME01246B (https=)
MX (1) MX2007002595A (https=)
NI (1) NI200700068A (https=)
NO (3) NO340654B1 (https=)
PL (1) PL1632232T6 (https=)
PT (1) PT1632232E (https=)
RS (1) RS51923B2 (https=)
SI (1) SI1632232T1 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
PT1981506E (pt) * 2006-01-20 2013-06-25 Janssen R & D Ireland Tratamento a longo prazo da infeção pelo vih com tmc278
AR065720A1 (es) 2007-03-14 2009-06-24 Tibotec Pharm Ltd Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso.
JP2014500261A (ja) * 2010-11-19 2014-01-09 ギリアード サイエンシーズ, インコーポレイテッド リルピビリンHClおよびフマル酸テノホビルジソプロキシルを含有する治療用組成物
KR101879468B1 (ko) * 2011-04-15 2018-07-17 엠큐어 파마슈티컬즈 리미티드 릴피비린 중간체의 제조를 위한 공정
EP2604593A1 (en) 2011-12-14 2013-06-19 Sandoz AG Polymorph of Rilpivirine hydrochloride and its use as antiviral
WO2013087794A1 (en) 2011-12-14 2013-06-20 Sandoz Ag Polymorph of rilpivirine hydrochloride and its use as antiviral
EP2628732A1 (en) 2012-02-20 2013-08-21 Sandoz AG Novel crystalline form of rilpivirine hydrochloride
WO2013153162A1 (en) 2012-04-11 2013-10-17 Sandoz Ag Polymorph of rilpivirine hydrochloride
WO2013153161A2 (en) 2012-04-11 2013-10-17 Sandoz Ag Novel polymorph of rilpivirine hydrochloride
CN103570688B (zh) * 2012-07-19 2016-06-08 中国科学院上海药物研究所 2,5-二氨甲基吡嗪类化合物、其药物组合物、制备方法和用途
GR1008965B (el) * 2015-12-02 2017-02-28 Φαρματεν Ανωνυμος Βιομηχανικη Και Εμπορικη Εταιρεια Φαρμακευτικων Ιατρικων Και Καλλυντικων Προϊοντων Φαρμακευτικο σκευασμα που περιλαμβανει δαρουναβιρη και μεθοδος παρασκευης αυτου
RU2616267C1 (ru) * 2016-01-25 2017-04-13 Закрытое Акционерное Общество "БИОКОМ" Твердая лекарственная форма индинавира немедленного высвобождения и способ ее получения
US11065198B2 (en) * 2016-10-24 2021-07-20 Janssen Sciences Ireland Unlimited Company Dispersible compositions
CN110958883A (zh) * 2017-06-30 2020-04-03 Viiv保健公司 组合及其用途和疗法
CN114392241B (zh) * 2022-01-10 2023-07-25 安徽贝克生物制药有限公司 一种利匹韦林片及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6307543B1 (en) * 1998-09-10 2001-10-23 Silicon Image, Inc. Bi-directional data transfer using two pair of differential lines as a single additional differential pair
MY169670A (en) * 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
JO3429B1 (ar) * 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv مشتقات برميدينات مثبطة فيروس الايدز
DK1529032T3 (da) * 2002-08-09 2013-07-08 Janssen Pharmaceutica Nv Fremgangsmåder til fremstilling af 4-4-4-(2-cyanoethenyl)-2,6-dimethylphenyl)amino)-2-pyrimidinyl)aminobenzonitrill
WO2004050068A1 (en) * 2002-11-29 2004-06-17 Janssen Pharmaceutica N.V. Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base
BRPI0407329A (pt) * 2003-02-07 2006-01-10 Janssen Pharmaceutica Nv Derivados de pirimidina para a prevenção de infecção de hiv

Also Published As

Publication number Publication date
FR16C1023I1 (fr) 2017-02-03
PT1632232E (pt) 2011-08-02
CY2016050I1 (el) 2017-07-12
FR16C1025I1 (fr) 2017-02-03
CY2016051I1 (el) 2017-07-12
NO2017065I1 (no) 2017-11-21
NO20071745L (no) 2007-04-02
EP1632232B1 (en) 2011-05-11
DK1632232T3 (da) 2011-08-22
CY1112249T1 (el) 2015-12-09
EA013686B1 (ru) 2010-06-30
RS51923B (sr) 2012-02-29
DK1632232T6 (da) 2022-04-19
HUS1600061I1 (hu) 2017-01-30
MX2007002595A (es) 2007-04-25
ES2371442T3 (es) 2012-01-02
BRPI0514871A (pt) 2008-06-24
KR20070074555A (ko) 2007-07-12
CN104586850A (zh) 2015-05-06
KR101284361B1 (ko) 2013-07-15
NO2017063I1 (no) 2017-11-21
NO340654B1 (no) 2017-05-22
LTC1632232I2 (lt) 2024-09-10
PL1632232T6 (pl) 2022-06-27
FR16C1023I2 (fr) 2025-11-21
EP1632232A1 (en) 2006-03-08
ME01246B (me) 2013-06-20
HUS1600060I1 (hu) 2017-01-30
LTPA2016042I1 (lt) 2017-01-10
EA200700536A1 (ru) 2007-08-31
JP4912309B2 (ja) 2012-04-11
ES2371442T7 (es) 2022-05-12
FR16C1025I2 (fr) 2025-11-21
RS51923B2 (sr) 2022-05-31
JP2008511592A (ja) 2008-04-17
HK1210029A1 (en) 2016-04-15
LTPA2016043I1 (lt) 2017-01-10
PL1632232T3 (pl) 2011-10-31
ATE508748T1 (de) 2011-05-15
SI1632232T1 (sl) 2011-09-30
EP1632232B3 (en) 2022-03-30
IL181650A (en) 2012-08-30
IL181650A0 (en) 2007-07-04

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