FR16C1023I1 - Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile - Google Patents

Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile

Info

Publication number
FR16C1023I1
FR16C1023I1 FR16C1023C FR16C1023C FR16C1023I1 FR 16C1023 I1 FR16C1023 I1 FR 16C1023I1 FR 16C1023 C FR16C1023 C FR 16C1023C FR 16C1023 C FR16C1023 C FR 16C1023C FR 16C1023 I1 FR16C1023 I1 FR 16C1023I1
Authority
FR
France
Prior art keywords
amino
cyanoethenyl
dimethylphenyl
pyrimidinyl
benzonitrile
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR16C1023C
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38091637&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR16C1023(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from MYPI20043578A external-priority patent/MY169670A/en
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Publication of FR16C1023I1 publication Critical patent/FR16C1023I1/fr
Active legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Hybrid Cells (AREA)
FR16C1023C 2004-09-02 2016-12-20 Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile Active FR16C1023I1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
MYPI20043578A MY169670A (en) 2003-09-03 2004-09-02 Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (fr) 2003-09-03 2004-09-03 Combinaisons d'une pyrimidine renfermant nnrti avec des inhibiteurs de rt
EP05101467 2005-02-25

Publications (1)

Publication Number Publication Date
FR16C1023I1 true FR16C1023I1 (fr) 2017-02-03

Family

ID=38091637

Family Applications (2)

Application Number Title Priority Date Filing Date
FR16C1023C Active FR16C1023I1 (fr) 2004-09-02 2016-12-20 Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile
FR16C1025C Active FR16C1025I1 (fr) 2004-09-02 2016-12-20 Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR16C1025C Active FR16C1025I1 (fr) 2004-09-02 2016-12-20 Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile

Country Status (21)

Country Link
EP (1) EP1632232B3 (fr)
JP (1) JP4912309B2 (fr)
CN (1) CN104586850A (fr)
AT (1) ATE508748T1 (fr)
BR (1) BRPI0514871A (fr)
CY (3) CY1112249T1 (fr)
DK (1) DK1632232T6 (fr)
EA (1) EA013686B1 (fr)
ES (1) ES2371442T7 (fr)
FR (2) FR16C1023I1 (fr)
HK (1) HK1210029A1 (fr)
HU (2) HUS1600061I1 (fr)
IL (1) IL181650A (fr)
LT (2) LTPA2016043I1 (fr)
ME (1) ME01246B (fr)
MX (1) MX2007002595A (fr)
NI (1) NI200700068A (fr)
NO (3) NO340654B1 (fr)
PT (1) PT1632232E (fr)
RS (1) RS51923B2 (fr)
SI (1) SI1632232T1 (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
TWI458483B (zh) * 2006-01-20 2014-11-01 Tibotec Pharm Ltd Ｈｉｖ感染之長期治療
AR065720A1 (es) 2007-03-14 2009-06-24 Tibotec Pharm Ltd Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso.
KR101923103B1 (ko) 2010-11-19 2018-11-28 길리애드 사이언시즈, 인코포레이티드 릴피비린 hcl 및 테노포비어 디소프록실 푸마레이트를 포함하는 치료 조성물
KR101879468B1 (ko) * 2011-04-15 2018-07-17 엠큐어 파마슈티컬즈 리미티드 릴피비린 중간체의 제조를 위한 공정
WO2013087794A1 (fr) 2011-12-14 2013-06-20 Sandoz Ag Polymorphe de chlorhydrate de rilpivirine et son utilisation à titre d'antiviral
EP2628732A1 (fr) 2012-02-20 2013-08-21 Sandoz AG Nouvelle forme cristalline d'hydrochlorure de rilpivirine
EP2604593A1 (fr) 2011-12-14 2013-06-19 Sandoz AG Polymorphe du chlorhydrate de rilpivirine et son utilisation comme antiviral
WO2013153161A2 (fr) 2012-04-11 2013-10-17 Sandoz Ag Nouveau polymorphe de chlorhydrate de rilpivirine
WO2013153162A1 (fr) 2012-04-11 2013-10-17 Sandoz Ag Polymorphe de chlorhydrate de rilpivirine
CN103570688B (zh) * 2012-07-19 2016-06-08 中国科学院上海药物研究所 2，5-二氨甲基吡嗪类化合物、其药物组合物、制备方法和用途
GR1008965B (el) * 2015-12-02 2017-02-28 Φαρματεν Ανωνυμος Βιομηχανικη Και Εμπορικη Εταιρεια Φαρμακευτικων Ιατρικων Και Καλλυντικων Προϊοντων Φαρμακευτικο σκευασμα που περιλαμβανει δαρουναβιρη και μεθοδος παρασκευης αυτου
RU2616267C1 (ru) * 2016-01-25 2017-04-13 Закрытое Акционерное Общество "БИОКОМ" Твердая лекарственная форма индинавира немедленного высвобождения и способ ее получения
DK3528791T3 (da) * 2016-10-24 2024-01-29 Janssen Sciences Ireland Unlimited Co Dispergible sammensætninger
WO2019003150A2 (fr) * 2017-06-30 2019-01-03 Viiv Healthcare Company Association, utilisations et schémas thérapeutiques
CN114392241B (zh) * 2022-01-10 2023-07-25 安徽贝克生物制药有限公司 一种利匹韦林片及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6307543B1 (en) * 1998-09-10 2001-10-23 Silicon Image, Inc. Bi-directional data transfer using two pair of differential lines as a single additional differential pair
JO3429B1 (ar) * 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv مشتقات برميدينات مثبطة فيروس الايدز
MY169670A (en) * 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
BR0313545B1 (pt) * 2002-08-09 2021-07-27 Janssen Pharmaceutica Nv processos para a preparação de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2-pirimidinil]amino]benzonitrila
WO2004050068A1 (fr) * 2002-11-29 2004-06-17 Janssen Pharmaceutica N.V. Compositions pharmaceutiques comprenant un compose medicamenteux respectivement basique, tensioactif et base respectivement acide hydrosoluble et tolerable physiologiquement
CA2513527C (fr) * 2003-02-07 2012-08-14 Janssen Pharmaceutica N.V. Derives de pyrimidine utilises dans la prevention des infections par le vih

Also Published As

Publication number Publication date
IL181650A (en) 2012-08-30
HK1210029A1 (en) 2016-04-15
EA013686B1 (ru) 2010-06-30
ATE508748T1 (de) 2011-05-15
JP2008511592A (ja) 2008-04-17
HUS1600061I1 (hu) 2017-01-30
EP1632232B3 (fr) 2022-03-30
NO340654B1 (no) 2017-05-22
LTPA2016042I1 (lt) 2017-01-10
DK1632232T3 (da) 2011-08-22
BRPI0514871A (pt) 2008-06-24
EP1632232B1 (fr) 2011-05-11
MX2007002595A (es) 2007-04-25
CY1112249T1 (el) 2015-12-09
EA200700536A1 (ru) 2007-08-31
ES2371442T7 (es) 2022-05-12
RS51923B2 (sr) 2022-05-31
RS51923B (en) 2012-02-29
IL181650A0 (en) 2007-07-04
HUS1600060I1 (hu) 2017-01-30
EP1632232A1 (fr) 2006-03-08
NO2017063I1 (no) 2017-11-21
CN104586850A (zh) 2015-05-06
NO20071745L (no) 2007-04-02
CY2016051I1 (el) 2017-07-12
ME01246B (fr) 2013-06-20
SI1632232T1 (sl) 2011-09-30
ES2371442T3 (es) 2012-01-02
DK1632232T6 (da) 2022-04-19
FR16C1025I1 (fr) 2017-02-03
NI200700068A (es) 2016-09-29
JP4912309B2 (ja) 2012-04-11
LTPA2016043I1 (lt) 2017-01-10
PT1632232E (pt) 2011-08-02
NO2017065I1 (no) 2017-11-21
CY2016050I1 (el) 2017-07-12

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