NI200700068A - Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo - Google Patents

Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo

Info

Publication number
NI200700068A
NI200700068A NI200700068A NI200700068A NI200700068A NI 200700068 A NI200700068 A NI 200700068A NI 200700068 A NI200700068 A NI 200700068A NI 200700068 A NI200700068 A NI 200700068A NI 200700068 A NI200700068 A NI 200700068A
Authority
NI
Nicaragua
Prior art keywords
amino
cyanoethenyl
benzonitrile
dimethylphenyl
pyrimidinyl
Prior art date
Application number
NI200700068A
Other languages
English (en)
Inventor
Theodoor Agnes Stevens Paul
Peeters Jozef
Petrus Gerebern Vandecruys Roger
Elisabeth Stappers Alfred
Herman Copmans Alex
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38091637&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NI200700068(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from MYPI20043578A external-priority patent/MY169670A/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NI200700068A publication Critical patent/NI200700068A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Hybrid Cells (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)

Abstract

La presente invención se relaciona con la sal fumarato de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2-pirimidinil] amino] benzonitrilo, composiciones farmacéuticas que comprenden como ingrediente activo a la sal y con procedimiento para su preparación.
NI200700068A 2004-09-02 2007-03-01 Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo NI200700068A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
MYPI20043578A MY169670A (en) 2003-09-03 2004-09-02 Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors
EP05101467 2005-02-25

Publications (1)

Publication Number Publication Date
NI200700068A true NI200700068A (es) 2016-09-29

Family

ID=38091637

Family Applications (1)

Application Number Title Priority Date Filing Date
NI200700068A NI200700068A (es) 2004-09-02 2007-03-01 Clorhidrato de 4-[[4-[[4-(2-cianoetenil)-2,6- dimetilfenil]amino]-2- pirimidinil]amino] benzonitrilo

Country Status (21)

Country Link
EP (1) EP1632232B3 (es)
JP (1) JP4912309B2 (es)
CN (1) CN104586850A (es)
AT (1) ATE508748T1 (es)
BR (1) BRPI0514871A (es)
CY (3) CY1112249T1 (es)
DK (1) DK1632232T6 (es)
EA (1) EA013686B1 (es)
ES (1) ES2371442T7 (es)
FR (2) FR16C1023I1 (es)
HK (1) HK1210029A1 (es)
HU (2) HUS1600060I1 (es)
IL (1) IL181650A (es)
LT (2) LTPA2016042I1 (es)
ME (1) ME01246B (es)
MX (1) MX2007002595A (es)
NI (1) NI200700068A (es)
NO (3) NO340654B1 (es)
PT (1) PT1632232E (es)
RS (1) RS51923B2 (es)
SI (1) SI1632232T1 (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
SI1981506T1 (sl) * 2006-01-20 2013-08-30 Janssen R&D Ireland Dolgoročno zdravljenje infekcije HIV s TCM278
AR065720A1 (es) 2007-03-14 2009-06-24 Tibotec Pharm Ltd Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso.
AU2011329642B2 (en) 2010-11-19 2016-08-11 Gilead Sciences, Inc. Therapeutic compositions comprising rilpivirine HCl and tenofovir disoproxil fumarate
JP5870183B2 (ja) * 2011-04-15 2016-02-24 エムキュア ファーマシューティカルズ リミテッド リルピビリン中間体の合成方法
EP2628732A1 (en) 2012-02-20 2013-08-21 Sandoz AG Novel crystalline form of rilpivirine hydrochloride
EP2604593A1 (en) 2011-12-14 2013-06-19 Sandoz AG Polymorph of Rilpivirine hydrochloride and its use as antiviral
WO2013087794A1 (en) 2011-12-14 2013-06-20 Sandoz Ag Polymorph of rilpivirine hydrochloride and its use as antiviral
WO2013153162A1 (en) 2012-04-11 2013-10-17 Sandoz Ag Polymorph of rilpivirine hydrochloride
WO2013153161A2 (en) 2012-04-11 2013-10-17 Sandoz Ag Novel polymorph of rilpivirine hydrochloride
CN103570688B (zh) * 2012-07-19 2016-06-08 中国科学院上海药物研究所 2，5-二氨甲基吡嗪类化合物、其药物组合物、制备方法和用途
GR1008965B (el) * 2015-12-02 2017-02-28 Φαρματεν Ανωνυμος Βιομηχανικη Και Εμπορικη Εταιρεια Φαρμακευτικων Ιατρικων Και Καλλυντικων Προϊοντων Φαρμακευτικο σκευασμα που περιλαμβανει δαρουναβιρη και μεθοδος παρασκευης αυτου
RU2616267C1 (ru) * 2016-01-25 2017-04-13 Закрытое Акционерное Общество "БИОКОМ" Твердая лекарственная форма индинавира немедленного высвобождения и способ ее получения
HUE064823T2 (hu) * 2016-10-24 2024-04-28 Janssen Sciences Ireland Unlimited Co Diszpergálható készítmények
CN114392241B (zh) * 2022-01-10 2023-07-25 安徽贝克生物制药有限公司 一种利匹韦林片及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6307543B1 (en) * 1998-09-10 2001-10-23 Silicon Image, Inc. Bi-directional data transfer using two pair of differential lines as a single additional differential pair
JO3429B1 (ar) * 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv مشتقات برميدينات مثبطة فيروس الايدز
MY169670A (en) * 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
CN102225902B (zh) * 2002-08-09 2013-04-24 詹森药业有限公司 制备4-[[4-[[4-(2-氰基乙烯基)-2,6-二甲基苯基]氨基]-2-嘧啶基]氨基]苄腈的方法
AU2002350719A1 (en) * 2002-11-29 2004-06-23 Janssen Pharmaceutica N.V. Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base
CL2004000192A1 (es) * 2003-02-07 2005-03-18 Janssen Pharmaceutica Nv Uso de compuestos derivados de 2-aminopirimidina para preparar un medicamento para la prevencion de una infeccion por vih relaciones sexuales o un contacto intimo en la pareja.

Also Published As

Publication number Publication date
CY2016051I1 (el) 2017-07-12
NO2017063I1 (no) 2017-11-21
PT1632232E (pt) 2011-08-02
EP1632232A1 (en) 2006-03-08
BRPI0514871A (pt) 2008-06-24
NO2017065I1 (no) 2017-11-21
EA013686B1 (ru) 2010-06-30
EA200700536A1 (ru) 2007-08-31
LTPA2016043I1 (lt) 2017-01-10
DK1632232T3 (da) 2011-08-22
JP2008511592A (ja) 2008-04-17
SI1632232T1 (sl) 2011-09-30
EP1632232B1 (en) 2011-05-11
CY2016050I1 (el) 2017-07-12
ME01246B (me) 2013-06-20
MX2007002595A (es) 2007-04-25
ES2371442T3 (es) 2012-01-02
HUS1600060I1 (hu) 2017-01-30
EP1632232B3 (en) 2022-03-30
CY1112249T1 (el) 2015-12-09
RS51923B2 (sr) 2022-05-31
RS51923B (en) 2012-02-29
CN104586850A (zh) 2015-05-06
LTPA2016042I1 (lt) 2017-01-10
HUS1600061I1 (hu) 2017-01-30
HK1210029A1 (en) 2016-04-15
IL181650A0 (en) 2007-07-04
FR16C1023I1 (fr) 2017-02-03
IL181650A (en) 2012-08-30
FR16C1025I1 (fr) 2017-02-03
JP4912309B2 (ja) 2012-04-11
NO340654B1 (no) 2017-05-22
ES2371442T7 (es) 2022-05-12
DK1632232T6 (da) 2022-04-19
ATE508748T1 (de) 2011-05-15
NO20071745L (no) 2007-04-02

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